IP Library Granted Patent US 8,598,135
Granted Patent B2
US 8,598,135 · App. 13/269,091 · Granted Dec 3, 2013

Insulin-like growth factor binding protein 7 for treatment of cancer

Inventors: Michael Green (Boylston, MA); Narendra Wajapeyee (Worcester, MA)
Assignee: University of Massachusetts
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 8,598,135
App. No.
13/269,091
Granted
Dec 3, 2013
Kind
B2
Abstract

Methods of treating a tumor in a subject include identifying a subject having, at risk for, or suspected of having a tumor, and administering to the subject an effective amount of an IGFBP7 agent if the tumor has increased Ras-BRAF-MEK-Erk signaling, is dependent for growth and/or survival upon the Ras-BRAF-MEK-Erk signaling pathway, and/or expresses an activated or oncogenic BRAF or RAS.

Claims (22)

1. A method of treating a tumor in a subject, the method comprising:

identifying a subject having, at risk for, or suspected of having a tumor;

providing a sample comprising a cell from the tumor;

detecting in the sample one or more of:

(i) a level of Ras-BRAF-MEK-Erk signaling;

(ii) dependence of growth or survival of the cell on Ras-BRAF-MEK-Erk signaling; or

(iii) expression of an activated or oncogenic BRAF or RAS;

determining that a cell of the tumor has increased Ras-BRAF-MEK-Erk signaling as compared to a predetermined reference level of Ras-BRAF-MEK-Erk signaling, is dependent for growth and/or survival upon the Ras-BRAF-MEK-Erk signaling pathway, and/or expresses an activated or oncogenic BRAF or RAS; and

administering to the subject an effective amount of an IGFBP7 polypeptide, thereby treating the tumor.

2. The method of claim 1 , wherein the tumor is a cancer.

3. The method of claim 2 , wherein the cancer is a melanoma.

4. The method of claim 2 , wherein the cancer is a carcinoma, breast cancer, ovarian cancer, pancreatic cancer, colon cancer, colorectal carcinoma, or papillary thyroid carcinoma.

5. The method of claim 2 , wherein the cancer expresses an activated or oncogenic BRAF or RAS.

6. The method of claim 2 , wherein the activated or oncogenic BRAF is BRAFV600E.

7. The method of claim 1 , wherein the oncogenic BRAF is BRAFV600E.

8. The method of claim 1 , wherein the IGFBP7 polypeptide consists of a polypeptide at least 80% identical to residues 29 to 282 of SEQ ID NO:1 or to SEQ ID NO:7.

9. The method of claim 8 , wherein the polypeptide is at least 85% identical to residues 29 to 282 of SEQ ID NO:1 or to SEQ ID NO:7.

10. The method of claim 1 , wherein the IGFBP7 polypeptide is administered by introducing to the subject a nucleic acid encoding a polypeptide at least 85% identical to residues 29 to 282 of SEQ ID NO:1 or to SEQ ID NO:7.

11. The method of claim 10 , wherein the nucleic acid is in a viral vector.

12. The method of claim 11 , wherein the viral vector is an adenovirus, adeno-associated virus, retrovirus, or lentivirus vector.

13. The method of claim 1 , wherein the IGFBP7 polypeptide is administered topically, systemically, or locally.

14. The method of claim 13 , wherein the IGFBP7 polypeptide is administered locally by a drug-releasing implant.

Assignments (2)
CONFIRMATORY LICENSE Recorded Sep 26, 2014
From: UNIVERSITY OF MASSACHUSETTS MEDICAL SCHOOL
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 033832/0564 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 9, 2012
From: GREEN, MICHAEL; WAJAPEYEE, NARENDRA
To: UNIVERSITY OF MASSACHUSETTS
Reel/Frame 027676/0614 →
Continuity (4)
Continuation 12209028 · Sep 11, 2008
Provisional Application 60993211 · Sep 11, 2007
Provisional Application 61092230 · Aug 27, 2008
Related Publication 20120094925A1 · Apr 19, 2012