IP Library Granted Patent US 8,815,241
Granted Patent B2
US 8,815,241 · App. 13/205,328 · Granted Aug 26, 2014

Use of combination of anti-angiogenic substance and c-kit kinase inhibitor

Inventor: Yuji Yamamoto (Ibaraki, JP)
Assignee: Eisai R&D Management Co., Ltd.
C07D215/48A61K31/4709A61K31/404A61K31/517A61K31/47A61K45/06A61K31/519A61K31/502A61K31/5377A61K31/506A61K31/4439A61K31/4409
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 8,815,241
App. No.
13/205,328
Granted
Aug 26, 2014
Kind
B2
Abstract

The object of the present invention is to find a pharmaceutical composition and a method for treating cancer that show an excellent antitumor effect. Combinational use of 4-(3-chloro-4-(cyclopropylaminocarbonyl)aminophenoxy)-7-methoxy-6-quinolinecarboxamide and analogues thereof can result in an excellent antitumor effect when combined with a substance having a c-kit kinase-inhibiting activity.

Claims (2)

1. A method for treating cancer comprising administering to a patient in need thereof an effective amount of 4-(3-chloro-4-(cyclopropylaminocarbonyl)aminophenoxy)-7-methoxy-6-quinolinecarboxamide, or a pharmacologically acceptable salt thereof, and an effective amount of 4-(4-methylipierazine-1-ylmethyl)-N-[4-methyl-3-[4-(3-pyridyl)pyrimidine-2-ylamino]phenyl]benzenamide or a pharmacologically acceptable salt thereof.

2. The method according to claim 1 , wherein a methanesulfonate of 4-(3-chloro-4-(cyclopropylaminocarbonyl)aminophenoxy)-7-methoxy-6-quinolinecarboxamide is administered.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 9, 2011
From: YAMAMOTO, YUJI
To: EISAI R&D MANAGEMENT CO., LTD.
Reel/Frame 026723/0187 →
Priority Claims (1)
JP 2005-322946 · Nov 7, 2005 · national
Continuity (2)
Division 12092539
Related Publication 20110293615A1 · Dec 1, 2011