IP Library Granted Patent US 8,865,710
Granted Patent B2
US 8,865,710 · App. 13/320,217 · Granted Oct 21, 2014

Methods of treating proliferative diseases

Inventors: Robert E. Corringham (San Diego, CA); Patrick B. O'Donnell (San Diego, CA); Joyce K. James (San Diego, CA)
Assignee: Ambit Biosciences Corporation
A61K31/429A61K9/4866A61K9/1641A61K9/08A61K9/145
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Quick Facts
Patent No.
US 8,865,710
App. No.
13/320,217
Granted
Oct 21, 2014
Kind
B2
Abstract

Provided herein are methods of administering N-(5-tert-butyl-isoxazol-3-yl)-N′-{4-[7-(2-morpholin-4-yl-ethoxy)imidazo[2,1-b][1,3]benzothiazol-2-yl]phenyl}urea, or a pharmaceutically acceptable salt or solvate thereof, to human patients, including a specific patient population. Specifically, dosing, dosing schedules or dosing regimens are provided herein. Methods of treating proliferative diseases or FLT-3 mediated diseases in humans are also provided.

Claims (7)

1. A spray-dried pharmaceutical composition comprising a compound of Formula I,

or a pharmaceutically acceptable salt or solvate thereof, and hydroxypropyl-β-cyclodextrin.

2. The pharmaceutical composition of claim 1 , wherein the pharmaceutically acceptable salt is a dihydrochloride salt.

3. The pharmaceutical composition of claim 1 , wherein the solvate is a methanol solvate.

4. The pharmaceutical composition of claim 1 comprising the pharmaceutically acceptable salt of compound of Formula I and hydroxypropyl-β-cyclodextrin in a ratio of about 1:10 based on weight.

5. The pharmaceutical composition of claim 1 , wherein the composition is formulated for single dose administration.

6. The pharmaceutical composition of claim 1 , wherein the composition is formulated for oral administration.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 15, 2026
From: AMBIT BIOSCIENCES CORPORATION
To: DAIICHI SANKYO COMPANY, LIMITED
Reel/Frame 074670/0770 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 31, 2012
From: CORRINGHAM, ROBERT E.; O'DONNELL, PATRICK B.
To: AMBIT BIOSCIENCES CORPORATION
Reel/Frame 029546/0220 →
Continuity (3)
Provisional Application 61178472 · May 14, 2009
Provisional Application 61243977 · Sep 18, 2009
Related Publication 20120258081A1 · Oct 11, 2012