IP Library Granted Patent US 9,084,777
Granted Patent B2
US 9,084,777 · App. 12/159,778 · Granted Jul 21, 2015

Stabilized antibody-containing formulations

Inventors: Toshiyuki Morichika (Tokyo, JP); Daisuke Kameoka (Tokyo, JP)
Assignee: CHUGAI SEIYAKU KABUSHIKI KAISHA
A61K39/39591A61K9/19A61K47/183C07K16/2866A61K9/0019A61K2039/505C07K2317/24
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Quick Facts
Patent No.
US 9,084,777
App. No.
12/159,778
Granted
Jul 21, 2015
Kind
B2
Abstract

The present invention relates to antibody-containing lyophilized formulations free from reducing sugars, non-reducing sugars, sugar alcohols or polysaccharides as excipients and including one or more amino acid selected from the group consisting of arginine, histidine, lysine, serine, proline, glycine, alanine and threonine or a salt thereof.

Claims (6)

1. A reconstituted solution obtained by adding water suitable for injection to an antibody-containing lyophilized pharmaceutical formulation free from reducing sugars, non-reducing sugars, sugar alcohols or polysaccharides as fillers and including one or more amino acids selected from the group consisting of arginine, lysine, serine, proline, glycine, alanine and threonine or a salt thereof, wherein the content of the amino acid or a salt thereof is 270 moles or more per mole of the antibody, wherein the antibody concentration in said reconstituted solution is 50 mg/ml or more.

2. The reconstituted solution of claim 1 , wherein the pH of the reconstituted solution is 4-8.

3. The reconstituted solution of claim 2 , wherein the pH of the reconstituted solution is 5.0-7.5.

4. The reconstituted solution of claim 1 , wherein the viscosity of the reconstituted solution is 20 mPa·s or less.

5. The reconstituted solution of claim 4 , wherein the viscosity of the reconstituted solution is 15 mPa·s or less.

6. The reconstituted solution of claim 5 , wherein the viscosity of the reconstituted solution is 12 mPa·s or less.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 5, 2009
From: MORICHIKA, TOSHIYUKI; KAMEOKA, DAISUKE
To: CHUGAI SEIYAKU KABUSHIKI KAISHA
Reel/Frame 022348/0243 →
Continuity (1)
Related Publication 20090291076A1 · Nov 26, 2009