IP Library Granted Patent US 9,556,101
Granted Patent B2
US 9,556,101 · App. 14/328,062 · Granted Jan 31, 2017

Compositions and methods relating to proliferative diseases

Inventors: Gavin P. Robertson (Hummelstown, PA); Raghavendra Gowda Chandagalu D. (Hershey, PA); Subbarao V. Madhunapantula (East Godavari District, IN); Gajanan S. Inamdar (Hindalga, IN); Omer F. Kuzu (Harrisburg, PA)
Assignee: The Penn State Research Foundation
C07C61/29A61K9/0019A61K9/1271A61K31/135A61K31/136A61K31/137A61K31/155A61K31/17A61K31/19A61K31/195A61K31/215A61K31/26A61K45/06C07C211/31C07C229/38C07C265/08C07C275/24C07C279/04C07C331/24C07C335/02
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Quick Facts
Patent No.
US 9,556,101
App. No.
14/328,062
Granted
Jan 31, 2017
Kind
B2
Abstract

Anti-cancer compositions and methods are described herein. In particular, compositions including one or more of leelamine, a leelamine derivative, abietylamine, an abietylamine derivative, and an abietic acid derivative are described. Methods for treatment of pathological conditions particularly cancer, in a subject using one or more of leelamine, a leelamine derivative, abietylamine, an abietylamine derivative, and an abietic acid derivative are described herein.

Claims (7)

1. An anti-cancer pharmaceutical composition, comprising:

N-methylabietylamine/GPR-7 {[(1R,4aR)-1,4a-dimethyl-7-(propan-2-yl)-1,2,3,4,4a,4b,5,6,10,10a-decahydrophenanthren-1-yl]methyl}(methyl)amine; and a pharmaceutically acceptable carrier.

2. The composition of claim 1 , wherein the pharmaceutically acceptable carrier comprises liposomes.

3. A method of treating a subject having cancer, comprising: administering a therapeutically effective amount of the anti-cancer pharmaceutical composition of claim 1 to the subject.

4. The method of claim 3 , wherein the anti-cancer pharmaceutical composition is effective to preferentially inhibit the PI3K, MAPK and STAT pathways in a cancer cell compared to a non-cancer cell.

5. The method of claim 3 , wherein the subject is human.

6. The method of claim 3 , further comprising administration of an adjunct anti-cancer treatment.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 14, 2016
From: ROBERTSON, GAVIN P.; RAGHAVENDRA GOWDA, CHANDAGALU D.; MADHUNAPANTULA, SUBBARAO; KUZU, OMER F.; INAMDAR, GAJANA S.
To: THE PENN STATE RESEARCH FOUNDATION
Reel/Frame 037731/0332 →
CONFIRMATORY LICENSE Recorded Apr 7, 2015
From: PENNSYLVANIA STATE UNIVERSITY
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 035379/0741 →
Continuity (4)
Division 13312682 · Dec 6, 2011
Provisional Application 61466572 · Mar 23, 2011
Provisional Application 61420094 · Dec 6, 2010
Related Publication 20140322304A1 · Oct 30, 2014