IP Library Granted Patent US 9,713,599
Granted Patent B2
US 9,713,599 · App. 14/629,938 · Granted Jul 25, 2017

Parenteral formulations of treprostinil

Inventor: Michael Wade (Chapel Hill, NC)
Assignee: United Therapeutics Corporation
A61K31/192A61K31/191A61K31/201A61K31/557A61K31/57
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Quick Facts
Patent No.
US 9,713,599
App. No.
14/629,938
Granted
Jul 25, 2017
Kind
B2
Abstract

The present invention describes novel methods for using Treprostinil or its derivative, or a pharmaceutically acceptable salt thereof, for the treatment and/or prevention of ischemic lesions, such as digital ulcers, in subjects with scleroderma (including systemic sclerosis), Buerger's disease, Raynaud's disease, Raynaud's phenomenon and/or other conditions that cause such lesions. The invention also relates to kits for treatment and/or prevention of ischemic lesions, comprising an effective amount of Treprostinil or its derivative, or a pharmaceutically acceptable salt thereof.

Claims (5)

1. A method of treating pulmonary hypertension comprising parenterally administering to a subject in need thereof a formulation comprising a) 0.1 to 5% w/v of treprostinil or a pharmaceutically acceptable salt thereof and b) a citrate buffer.

2. The method of claim 1 , wherein the parenteral administration is performed intravenously.

3. The method of claim 1 , wherein the formulation is sterile and isotonic with a blood of the subject.

4. The method of claim 1 , wherein the formulation is administered at a rate of 0.625 to 50 ng/kg/min.

5. The method of claim 1 , wherein the formulation is administered at a rate of 10 to 15 ng/kg/min.

Continuity (4)
Continuation 12232611 · Sep 19, 2008
Continuation In Part 11012723 · Dec 16, 2004
Provisional Application 60529622 · Dec 16, 2003
Related Publication 20150164834A1 · Jun 18, 2015