IP Library Granted Patent US 9,931,397
Granted Patent B2
US 9,931,397 · App. 11/917,709 · Granted Apr 3, 2018

Immunogenic composition

Inventors: Ralph Leon Biemans (Rixensart, BE); Dominique Boutriau (Rixensart, BE); Carine Capiau (Rixensart, BE); Philippe Denoel (Rixensart, BE); Pierre Duvivier (Rixensart, BE); Jan Poolman (Rixensart, BE)
Assignee: GLAXOSMITHKLINE BIOLOGICALS S.A.
A61K39/385A61K39/0017A61K39/0018A61K39/05A61K39/08A61K39/092A61K39/095A61K39/099A61K39/102A61K39/116A61K39/145A61K39/292C07H3/00C12N7/00A61K39/12A61K2039/545A61K2039/55A61K2039/575A61K2039/6037A61K2039/62A61K2039/627A61K2039/70C12N2730/10134C12N2760/16234C12N2760/16271C12N2770/32634
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Quick Facts
Patent No.
US 9,931,397
App. No.
11/917,709
Granted
Apr 3, 2018
Kind
B2
Abstract

The present application relates to an immunogenic composition comprising at least 2 conjugates of N. meningitidis capsular saccharide and protein carrier, wherein said conjugates comprise at least 2 different N. meningitidis capsular saccharides selected from the group consisting of MenA, MenC, MenY and MenW, wherein at least one capsular saccharide is conjugated to a protein carrier with a saccharide:protein ratio (w/w) between 1:2-1:5, and wherein at least one different capsular saccharide is conjugated to a protein carrier with a saccharide:protein ratio (w/w) between 5:1-1:1.99.

Claims (17)

1. An immunogenic composition comprising conjugates of a plurality of N. meningitidis capsular saccharides and carrier protein, wherein said conjugates comprise a first N. meningitidis capsular saccharide which is N. meningitidis serogroup A capsular saccharide (MenA) or N. meningitidis serogroup C capsular saccharide (MenC), wherein the first N. meningitidis capsular saccharide is conjugated to a first carrier protein with a saccharide to carrier protein ratio (w/w) ranging from 1:2-1:5, and a second different N. meningitidis capsular saccharide conjugated to a second carrier protein with a saccharide to carrier protein ratio (w/w) ranging from 5:1-1:1.99, wherein the second different capsular saccharide is a N. meningitidis serogroup Y capsular saccharide (MenY), a N. meningitidis serogroup W capsular saccharide (MenW) or a N. meningitidis serogroup C capsular saccharide (MenC), wherein the first N. meningitidis capsular saccharide is conjugated to a linker with 1-cyano-4-dimethylamino pyridinium tetrafluoroborate (CDAP) chemistry, wherein the first carrier protein is conjugated to the linker with carbodiimide chemistry, optionally using 1-ethyl-3-(3-dimethylaminopropyl) carbodiimide (EDAC), and wherein the composition does not include an adjuvant.

2. The immunogenic composition of claim 1 , wherein the first N. meningitidis capsular saccharide is N. meningitidis serogroup A capsular saccharide (MenA) and the second different N. meningitidis capsular saccharide is N. meningitidis serogroup W capsular saccharide (MenW) and the ratio of the MenW capsular saccharide to the carrier protein ranges from 5:1-1:1.99, 2:1-1:1.99, 1.5:1-1:1.8, 1:1-1:1.7, 1:1.2-1:1.6, or 1:1.4-1:1.5 (w/w).

3. The immunogenic composition of claim 1 , wherein the second N. meningitidis capsular saccharide is N. meningitidis serogroup Y capsular saccharide (MenY) and the ratio of the MenY capsular saccharide to the carrier protein ranges from 5:1-1:1.99, 2:1-1:1.99, 1.5:1-1:1.9, 1:1-1:1.8, 1:1.1-1:1.6, or 1:1.3-1:1.4 (w/w).

4. The immunogenic composition of claim 2 , wherein the ratio of the N. meningitidis serogroup A capsular saccharide (MenA) to the carrier protein ranges from 1:2-1:5, 1:2.4-1:4, 1:2.7-1:3.5, or 1:2.9-1:3.1 (w/w).

5. The immunogenic composition of claim 1 , wherein the first N. meningitidis capsular saccharide is N. meningitidis serogroup A capsular saccharide (MenA) and the second different N. meningitidis capsular saccharide is N. meningitidis serogroup C capsular saccharide (MenC) and the ratio of the MenC capsular saccharide to carrier protein ranges from 5:1-1:1.99, 2:1-1:1.99, 1.5;1-1:1.8, 1.3:1-1:1.6, 1.2:1-1:1.4, or 1.1:1-1:1.2 (w/w).

6. The immunogenic composition of claim 1 , wherein the first N. meningitidis capsular saccharide is N. meningitidis serogroup C capsular saccharide (MenC) and the ratio of the MenC capsular saccharide to carrier protein ranges from 1:2-1:5, 1:2.5-1:4.5, 1:2.7-1:4.3, 1:3-1:4, or 1:3.3-1:3.5 (w/w).

7. The immunogenic composition of claim 1 , wherein the second different N. meningitidis capsular saccharide is directly conjugated to the second carrier protein.

8. The immunogenic composition of claim 1 wherein the first and second carrier proteins are independently selected from the group consisting of tetanus toxoid (TT), diphtheria toxoid (DT), cross-reacting material 197 (CRM197), fragment C of tetanus toxoid (TT) and protein D.

9. The immunogenic composition of claim 8 wherein the first N. meningitidis capsular saccharide is conjugated to the first carrier protein and the second different N. meningitidis capsular saccharide is conjugated to the second carrier protein, wherein the first and second carrier proteins are the same carrier protein.

10. The immunogenic composition of claim 1 , wherein the first N. meningitidis capsular saccharide is separately conjugated to the first carrier protein and the second different N. meningitidis capsular saccharide is separately conjugated to the second carrier protein.

11. The immunogenic composition of claim 1 , further comprising a H. influenzae b capsular saccharide (Hib) conjugated to a carrier protein.

12. The immunogenic composition of claim 11 wherein the H. influenzae b capsular saccharide (Hib) conjugate is present in a lower dose than the dose of each of the first capsular saccharide and the second different capsular saccharide conjugates.

13. The immunogenic composition of claim 1 comprising a N. meningitidis serogroup B outer membrane vesicle preparation or capsular saccharide.

14. A vaccine comprising the immunogenic composition of claim 1 and a pharmaceutically acceptable excipient.

15. A vaccine kit for concomitant or sequential administration comprising two multi-valent immunogenic compositions for conferring protection in a host against disease caused by Bordetella pertussis, Clostridium tetani, Corynebacterium diphtheriae, Haemophilus influenzae and Neisseria meningitidis , said kit comprising a first container comprising tetanus toxoid (TT), diphtheria toxoid (DT), and whole-cell or acellular pertussis components and a second container comprising the immunogenic composition of claim 1 .

16. A process for making the vaccine of claim 14 comprising the step of mixing the immunogenic composition of claim 1 with a pharmaceutically acceptable excipient.

17. A method of immunizing a human host against disease caused by Neisseria meningitidis infection comprising administering to the host an immunoprotective dose of the immunogenic composition of claim 1 .

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 15, 2008
From: BIEMANS, RALPH LEON; BOUTRIAU, DOMINIQUE; CAPIAU, CARINE; DENOEL, PHILIPPE; DUVIVIER, PIERRE; POOLMAN, JAN
To: GLAXOSMITHKLINE BIOLOGICALS S.A.
Reel/Frame 020520/0267 →
Priority Claims (6)
GB 0513069.5 · Jun 27, 2005 · national
GB 0513071.1 · Jun 27, 2005 · national
GB 0515556.9 · Jul 28, 2005 · national
GB 0524204.5 · Nov 28, 2005 · national
GB 0526040.1 · Dec 21, 2005 · national
GB 0526041.9 · Dec 21, 2005 · national
Continuity (1)
Related Publication 20090252759A1 · Oct 8, 2009