IP Library › Granted Patent US 10,004,808
Granted Patent B2
US 10,004,808 · App. 15/215,000 · Granted Jun 26, 2018

Methods of treating ulcerative colitis

Inventors: Irving H. Fox (Wellesley, MA); Catherine Scholz (Woburn, MA)
Assignee: MILLENNIUM PHARMACEUTICALS, INC.
A61K47/26A61K9/0019A61K9/19A61K39/39591A61K47/183C07K16/2839A61K2039/505A61K2039/54A61K2039/545C07K2317/14C07K2317/24C07K2317/565C07K2317/92C07K2317/94
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Quick Facts
Patent No.
US 10,004,808
App. No.
15/215,000
Granted
Jun 26, 2018
Kind
B2
Abstract

Methods for inducing clinical remission of ulcerative colitis in a human patient are described comprising administration of an antibody that has binding specificity for human α4β7 integrin using a safe dosing regimen of these antibody formulations that is easy to follow, and which results in a therapeutically effective amount of the anti-α4β7 antibody in vivo.

Claims (5)

1. A method for inducing clinical remission in a human patient having moderately to severely active ulcerative colitis, comprising intravenously administering: a first dose of 300 mg of an antibody that has binding specificity for human α4β7 integrin, a second dose of 300 mg of the antibody two weeks after the first dose, a third dose of 300 mg of the antibody six weeks after the first dose, and then 300 mg of the antibody every eight weeks thereafter, wherein the antibody comprises the heavy chain variable region sequence of amino acids 20 to 140 of SEQ ID NO:2, and the light chain variable region sequence of amino acids 20 to 131 of SEQ ID NO:4, and wherein the human patient had a lack of an adequate response with, lost response to, or was intolerant to a TNFα antagonist.

2. The method of claim 1 , wherein the heavy chain of the antibody comprises amino acids 20 to 470 of SEQ ID NO:2, and the light chain of the antibody comprises amino acids 20 to 238 of SEQ ID NO:4.

3. The method of claim 1 , wherein each dose is intravenously administered as an infusion over about 30 minutes.

4. A method for inducing clinical remission in a human patient having moderately to severely active ulcerative colitis, comprising intravenously administering: a first dose of 300 mg of vedolizumab, a second dose of 300 mg of vedolizumab two weeks after the first dose, a third dose of 300 mg of vedolizumab six weeks after the first dose, and then 300 mg of vedolizumab every eight weeks thereafter,

wherein the human patient had a lack of an adequate response with, lost response to, or was intolerant to a TNFα antagonist.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 25, 2023
From: MILLENNIUM PHARMACEUTICALS, INC.
To: TAKEDA PHARMACEUTICAL COMPANY LIMITED
Reel/Frame 064700/0474 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 23, 2016
From: FOX, IRVING H.; SCHOLZ, CATHERINE
To: MILLENNIUM PHARMACEUTICALS, INC.
Reel/Frame 039841/0506 →
Continuity (5)
Continuation 13462414 · May 2, 2012
Provisional Application 61585859 · Jan 12, 2012
Provisional Application 61550545 · Oct 24, 2011
Provisional Application 61481533 · May 2, 2011
Related Publication 20170002078A1 · Jan 5, 2017
Cited By (13)
US 12,246,064 US 12,286,479 US 12,295,988 US 12,304,956 US 12,391,760 US 12,404,334 US 12,544,445 US 12,551,536 US 12,590,157 US 12,606,627 US 12,622,969 US 12,693,298 US 12,703,749