IP Library › Granted Patent US 10,093,752
Granted Patent B2
US 10,093,752 · App. 14/304,265 · Granted Oct 9, 2018

Homopolymer nanoparticles by self-emulsion polymerization reaction and preparation method thereof

Inventors: Jae-Suk Lee (Gwangju, KR); Santosh Kumar (Gwangju, KR); Dong Woo Kim (Gwangju, KR); Mohammad Changei (Gwangju, KR); Hong-Joon Lee (Gwangju, KR)
Assignee: GWANGJU INSTITUTE OF SCIENCE AND TECHNOLOGY
C08F2/22A61K9/5138C08F120/06C08F120/20C08F120/42C08F126/06C08F126/10
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Quick Facts
Patent No.
US 10,093,752
App. No.
14/304,265
Granted
Oct 9, 2018
Kind
B2
Abstract

Disclosed herein is a preparation method of homopolymer nanoparticles without using a surfactant. The homopolymer nanoparticles prepared thereby are expected to be widely used not only as a template of a semiconductor metal oxide, a drug delivery system (DDS), an electron transport layer (ETL), and a seed having vertical structural shape, but also in a high precision field such as replacement of an organic device polystyrene bead film.

Claims (18)

1. A preparation method of homopolymer nanoparticles comprising:

(i) preparing a deoxygenated mixture of water and an amphiphilic monomer selected from the group consisting of vinylpyridine, 4-vinylpyridine, acrylic acid, methacrylic acid, styrene sulfonic acid, 4-styrene sulfonic acid, 2-hydroxyethyl methacrylate, hydroxypropyl methacrylate, hydroxybutyl methacrylate, methacrylamide, n-vinylpyrrolidone, acrylonitrile, 4-(4-vinylphenyl)pyridine, and 6-vinylpyridine-3-carbonitrile;

(ii) adding a hydrophilic initiator to said mixture to initiate a surfactant-free polymerization reaction of amphiphilic monomers;

(iii) carrying out the surfactant-free polymerization reaction at constant temperature ranging from 55° C. to 95° C. for 50-160 minutes to form the homopolymer nanoparticles.

2. The preparation method of homopolymer nanoparticles of claim 1 , wherein the homopolymer is represented by one of the following Chemical Formulae 1-7:

wherein n is an integer of 10 to 10,000.

3. The preparation method of homopolymer nanoparticles of claim 1 , wherein the hydrophilic initiator is at least one selected from the group consisting of 2,2′-azobis[2-(2-imidazolin-2-yl)propane]dihydrochloride, 4,4-azobis(4-cyanovaleric acid), ammonium persulfate, potassium persulfate, sodium persulfate, ammonium bisulfate, sodium bisulfate and 1,1-azobis(1-methylbutyronitrile-3-sodium sulfonate).

4. Homopolymer nanoparticles comprising a homopolymer represented by one of the following Chemical Formulae 1-7:

wherein n is an integer of 10 to 10,000; and

wherein said nanoparticles consist of 2-1,000 homopolymers; have a spherical shape having a diameter of 1-800 nm; and have a shell composed of hydrophilic pendants of said homopolymers and an inner layer composed of 70-95 vol % of hydrophobic main chains of said homopolymers and 5-30 vol % of hydrophilic pendants of said homopolymers.

5. The homopolymer nanoparticles of claim 4 prepared by the preparation method of claim 1 .

6. A drug delivery material comprising the homopolymer nanoparticles of claim 4 and a pharmaceutical active material collected in the inner layer of the homopolymer nanoparticles.

7. A preparation method of homopolymer nanoparticles comprising:

(i) preparing a deoxygenated mixture of water and an amphiphilic monomer selected from the group consisting of vinylpyridine, 4-vinylpyridine, acrylic acid, methacrylic acid, styrene sulfonic acid, 4-styrene sulfonic acid, 2-hydroxyethyl methacrylate, hydroxypropyl methacrylate, hydroxybutyl methacrylate, methacrylamide, n-vinylpyrrolidone, acrylonitrile, 4-(4-vinylphenyl)pyridine, and 6-vinylpyridine-3-carbonitrile;

(ii) adding a hydrophilic initiator to said mixture to initiate a surfactant-free polymerization reaction of amphiphilic monomers;

(iii) carrying out a surfactant-free polymerization reaction at constant temperature ranging from 55° C. to 95° C. for 50-160 minutes to form the homopolymer nanoparticles;

(iv) swelling the homopolymer nanoparticles and collecting a pharmaceutical active material in an inner layer of said nanoparticles.

8. The preparation method of homopolymer nanoparticles of claim 7 , wherein the hydrophilic initiator is at least one selected from the group consisting of 2,2′-azobis[2-(2-imidazolin-2-yl)propane]dihydrochloride, 4,4-azobis(4-cyanovaleric acid), ammonium persulfate, potassium persulfate, sodium persulfate, ammonium bisulfate, sodium bisulfate and 1,1-azobis(1-methylbutyronitrile-3-sodium sulfonate).

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 13, 2014
From: LEE, JAE-SUK; KUMAR, SANTOSH; KIM, DONG WOO; CHANGEI, MOHAMMAD; LEE, HONG-JOON
To: GWANGJU INSTITUTE OF SCIENCE AND TECHNOLOGY
Reel/Frame 033164/0459 →
Priority Claims (1)
KR 10-2014-0001067 · Jan 6, 2014 · national
Continuity (2)
Provisional Application 61834436 · Jun 13, 2013
Related Publication 20140370114A1 · Dec 18, 2014