IP Library Granted Patent US 10,131,633
Granted Patent B2
US 10,131,633 · App. 15/841,652 · Granted Nov 20, 2018

Cationic lipid

Inventors: Yuta Suzuki (Tsukuba, JP); Kenji Hyodo (Tsukuba, JP); Yohei Tanaka (Nakama, JP)
Assignees: Eisai R&D Management Co., Ltd.; Sogo Pharmaceutical Co., Ltd.
C07D211/62A61K9/5123A61K47/22A61K48/0033C07D205/04C07D207/16C12N15/111C12N15/1137C12N2310/14C12N2320/32
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Quick Facts
Patent No.
US 10,131,633
App. No.
15/841,652
Granted
Nov 20, 2018
Kind
B2
Abstract

The present invention provides a cationic lipid which can be used for nucleic acid delivery to a cytoplasm and which is possible to solve the problem of physical stability of a lipid complex. This cationic lipid is a compound represented by the general formula (3) or a pharmaceutically acceptable salt thereof: wherein, L is an alkyl having 7-12 carbon atoms or an alkenyl having 7-12 carbon atoms, R is an alkyl having 1-2 carbon atoms, and n 1 and n 2 are independently an integer of 1-3.

Claims (6)

1. A cationic lipid which is a compound represented by formula (3) or a pharmaceutically acceptable salt thereof:

wherein L is an alkyl having 7-12 carbon atoms or an alkenyl having 7-12 carbon atoms,

R is an alkyl having 1-2 carbon atoms,

n 1 is 2, and

n 2 is 1.

2. The cationic lipid according to claim 1 , wherein the cationic lipid is a compound represented by the following formula (5) or a pharmaceutically acceptable salt thereof:

Assignments (2)
CORRECTIVE ASSIGNMENT TO CORRECT THE ADDRESS OF THE FIRST LISTED ASSIGNEE PREVIOUSLY RECORDED ON REEL 044832 FRAME 0599. ASSIGNOR(S) HEREBY CONFIRMS THE ASSIGNMENT. Recorded May 21, 2018
From: SUZUKI, YUTA; HYODO, KENJI; TANAKA, YOHEI
To: EISAI R&D MANAGEMENT CO., LTD.; SOGO PHARMACEUTICAL CO., LTD.
Reel/Frame 046963/0756 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 5, 2018
From: SUZUKI, YUTA; HYODO, KENJI; TANAKA, YOHEI
To: EISAI R&D MANAGEMENT CO., LTD.; SOGO PHARMACEUTICAL CO., LTD.
Reel/Frame 044832/0599 →
Continuity (3)
Division 15109512
Provisional Application 61925267 · Jan 9, 2014
Related Publication 20180105493A1 · Apr 19, 2018
Cited By (1)
US 12,667,521