IP Library Granted Patent US 10,149,839
Granted Patent B2
US 10,149,839 · App. 15/657,395 · Granted Dec 11, 2018

Chemical compounds

Inventors: James Stewart Scott (Cambridge, GB); Thomas Andrew Moss (Cambridge, GB); Daniel Hillebrand O'Donovan (Cambridge, GB); Johannes Wilhelmus Maria Nissink (Cambridge, GB); Samantha Jayne Hughes (Cambridge, GB); Bernard Christophe Barlaam (Cambridge, GB); Dan Anders Broo (Mölndal, SE); Bin Yang (Waltham, MA); Jeffrey Gilbert Varnes (Waltham, MA); Dedong Wu (Waltham, MA)
Assignee: AstraZeneca AB
A61K31/437A61K31/407A61K31/495A61K31/506C07D471/04G01N23/20075G01N25/4866
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Quick Facts
Patent No.
US 10,149,839
App. No.
15/657,395
Granted
Dec 11, 2018
Kind
B2
Abstract

The specification relates to compounds of Formula (I): and pharmaceutically acceptable salts thereof, to processes and intermediates used for their preparation, pharmaceutical compositions containing them and their use in the treatment of cell proliferative disorders.

Claims (8)

1. A compound, or a pharmaceutically acceptable salt thereof, wherein the compound is N-(2-((5-((1R,3R)-2-(2,2-difluoroethyl)-3-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-4-methoxypyridin-2-yl)oxy)ethyl)-3-fluoropropan-1-amine, which compound has the following structure:

2. A pharmaceutical composition, which comprises the compound according to claim 1 , or a pharmaceutically acceptable salt thereof, in association with a pharmaceutically-acceptable excipient.

3. A compound, wherein the compound is N-(2-((5-(1R,3R)-2-(2,2-difluoroethyl)-3-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-4-methoxypyridin-2-yl)oxy)ethyl)-3-fluoropropan-1-amine.

4. A pharmaceutical composition, which comprises the compound according to claim 3 , in association with a pharmaceutically-acceptable excipient.

5. A pharmaceutically acceptable salt of N-(2-((5-((1R,3R)-2-(2,2-difluoroethyl)-3-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-4-methoxypyridin-2-yl)oxy)ethyl)-3-fluoropropan-1-amine.

6. A pharmaceutical composition, which comprises the salt according to claim 5 , in association with a pharmaceutically-acceptable excipient.

7. A pharmaceutically acceptable salt, wherein the pharmaceutically acceptable salt is the 2-methoxybenzoate salt of N-(2-((5-((1R,3R)-2-(2,2-difluoroethyl)-3-methyl-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)-4-methoxypyridin-2-yl)oxy)ethyl)-3-fluoropropan-1-amine.

8. A pharmaceutical composition, which comprises the salt according to claim 7 , in association with a pharmaceutically-acceptable excipient.

Assignments (11)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 26, 2018
From: YANG, BIN
To: ASTRAZENECA PHARMACEUTICALS LP
Reel/Frame 045716/0708 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 27, 2018
From: BROO, DAN ANDERS
To: ASTRAZENECA AB
Reel/Frame 045044/0204 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 27, 2018
From: HUGHES, SAMANTHA JAYNE
To: ASTRAZENECA UK LIMITED
Reel/Frame 045448/0475 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 27, 2018
From: YANG, BIN; VARNES, JEFFREY GILBERT
To: ASTRAZENECA PHARMACEUTICALS LP
Reel/Frame 045464/0120 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 31, 2018
From: BROO, DAN ANDERS
To: ASTRAZENECA AB
Reel/Frame 045204/0355 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 25, 2018
From: HUGHES, SAMANTHA JAYNE
To: ASTRAZENECA UK LIMITED
Reel/Frame 045141/0248 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 25, 2018
From: BROO, DAN ANDERS
To: ASTRAZENECA AB
Reel/Frame 045141/0194 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 25, 2018
From: WU, DEDONG
To: ASTRAZENECA PHARMACEUTICALS LP
Reel/Frame 044723/0761 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 25, 2018
From: ASTRAZENECA PHARMACEUTICALS LP
To: ASTRAZENECA UK LIMITED
Reel/Frame 044723/0784 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 25, 2018
From: ASTRAZENECA UK LIMITED
To: ASTRAZENECA AB
Reel/Frame 044723/0808 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 25, 2018
From: SCOTT, JAMES STEWART; MOSS, THOMAS ANDREW; O'DONOVAN, DANIEL HILLEBRAND; NISSINK, JOHANNES WILHELMUS, MARIA; BARLAAM, BERNARD CHRISTOPHE
To: ASTRAZENECA UK LIMITED
Reel/Frame 044723/0627 →
Continuity (5)
Provisional Application 62366173 · Jul 25, 2016
Provisional Application 62382909 · Sep 2, 2016
Provisional Application 62429951 · Dec 5, 2016
Provisional Application 62472852 · Mar 17, 2017
Related Publication 20180021316A1 · Jan 25, 2018