IP Library › Granted Patent US 10,188,108
Granted Patent B2
US 10,188,108 · App. 15/565,087 · Granted Jan 29, 2019

Fused bicyclic heterocycle derivatives as pesticides

Inventors: Rüdiger Fischer (Pulheim, DE); David Wilcke (Düsseldorf, DE); Dominik Hager (Monheim, DE); Kerstin Ilg (Köln, DE); Sascha Eilmus (Leichlingen, DE); Ulrich Görgens (Ratingen, DE); Andreas Turberg (Haan, DE)
Assignee: BAYER CROPSCIENCE AKTIENGESELLSCHAFT
A01N43/90C07D471/04C07D519/00
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Quick Facts
Patent No.
US 10,188,108
App. No.
15/565,087
Granted
Jan 29, 2019
Kind
B2
Abstract

The invention relates to novel compounds of the formula (I) in which R 1 , R 2 , R 3 , Q and n have the meanings given above, to their use as acaricides and/or insecticides for controlling animal pests and to processes and intermediates for their preparation.

Claims (106)

1. A compound of formula (I)

wherein

R 1 is ethyl,

R 3 is hydrogen,

Q is

 where the bond from Q to the remainder of the molecule is identified by a wavy line,

n is 0, and

R 2 is selected from the group consisting of H, 8-CF 3 , 8-Cl, 8-SC 2 H 5 , 5-CF 3 and 6-CH 3 ;

or

R 1 is ethyl,

R 3 is hydrogen,

Q is

 where the bond from Q to the remainder of the molecule is identified by a wavy line,

n is 1, and

R 2 is selected from the group consisting of 6-Cl, 6-CF 3 , 7-CF 3 , 5-CF 3 , 8-CF 3 and 6-OCH 3 ;

or

R 1 is ethyl,

R 3 is hydrogen,

Q is

 where the bond from Q to the remainder of the molecule is identified by a wavy line,

n is 2, and

R 2 is selected from the group consisting of H, 8-Cl, 5-CF 3 , 8-CF 3 , 8-SO 2 C 2 H 5 , 6-CH 3 and 6-OCH 3 ;

or

R 1 is ethyl,

R 3 is hydrogen,

Q is

 where the bond from Q to the remainder of the molecule is identified by a wavy line,

n is 0, and

R 2 is selected from the group consisting of H, 5-CH 3 , 5-CF 3 , 6-CF 3 , 6-Cl, 7-CF 3 , 5-SC 2 H 5 , 7-SC 2 H 5 , 7-CH 3 and 6-CH 3 ;

or

R 1 is ethyl,

R 3 is hydrogen,

Q is

 where the bond from Q to the remainder of the molecule is identified by a wavy line,

n is 1, and

R 2 is hydrogen;

or

R 1 is ethyl,

R 3 is hydrogen,

Q is

 where the bond from Q to the remainder of the molecule is identified by a wavy line,

n is 2, and

R 2 is selected from the group consisting of H, 7-CH 3 , 7-CF 3 , 6-CH 3 , 6-CF 3 , 6-Cl and 5-CH 3 ;

or

R 1 is ethyl,

R 3 is hydrogen,

Q is

 where the bond from Q to the remainder of the molecule is identified by a wavy line,

n is 2, and

R 2 is H.

2. The compound formula (I) according to claim 1 , wherein

R 1 is ethyl,

R 3 is hydrogen,

Q is

 where the bond from Q to the remainder of the molecule is identified by a wavy line,

n is 0, and

R 2 is selected from the group consisting of H, 8-CF 3 , 8-Cl, 8-SC 2 H 5 , 5-CF 3 and 6-CH 3 .

3. The compound formula (I) according to claim 1 , wherein

R 1 is ethyl,

R 3 is hydrogen,

Q is

 where the bond from Q to the remainder of the molecule is identified by a wavy line,

n is 1, and

R 2 is selected from the group consisting of 6-Cl, 6-CF 3 , 7-CF 3 , 5-CF 3 , 8-CF 3 and 6-OCH3.

4. The compound formula (I) according to claim 1 , wherein

R 1 is ethyl,

R 3 is hydrogen,

Q is

 where the bond from Q to the remainder of the molecule is identified by a wavy line,

n is 2, and

R 2 is selected from the group consisting of H, 8-Cl, 5-CF 3 , 8-CF 3 , 8-SO 2 C 2 H 5 , 6-CH 3 and 6-OCH 3 .

5. The compound formula (I) according to claim 1 , wherein

R 1 is ethyl,

R 3 is hydrogen,

Q is

 where the bond from Q to the remainder of the molecule is identified by a wavy line,

n is 0, and

R 2 is selected from the group consisting of H, 5-CH 3 , 5-CF 3 , 6-CF 3 , 6-Cl, 7-CF 3 , 5-SC 2 H 5 , 7-SC 2 H 5 , 7-CH 3 and 6-CH 3 .

6. The compound formula (I) according to claim 1 , wherein

R 1 is ethyl,

R 3 is hydrogen,

Q is

 where the bond from Q to the remainder of the molecule is identified by a wavy line,

n is 1, and

R 2 is hydrogen.

7. The compound formula (I) according to claim 1 , wherein

R 1 is ethyl,

R 3 is hydrogen,

Q is

where the bond from Q to the remainder of the molecule is identified by a wavy line,

n is 2, and

R 2 is selected from the group consisting of H, 7-CH 3 , 7-CF 3 , 6-CH 3 , 6-CF 3 , 6-Cl and 5-CH 3 .

8. The compound formula (I) according to claim 1 , wherein

R 1 is ethyl,

R 3 is hydrogen,

Q is

 where the bond from Q to the remainder of the molecule is identified by a wavy line,

n is 2, and

R 2 is H.

9. The compound formula (I) according to claim 4 , wherein

R 2 is hydrogen.

10. A method for controlling one or more animal pests, comprising allowing a compound of the formula (I) according to claim 1 or an agrochemical formulation thereof to act on the animal pests and/or a habitat thereof.

11. An agrochemical formulation comprising one or more compounds according to claim 1 and also one or more extenders and/or surfactants.

12. The agrochemical formulation according to claim 11 , additionally comprising a further agrochemically active compound.

13. The method according to claim 10 , wherein said one or more animal pests comprise insects, arachnids, helminths, nematodes or molluscs.

14. A product comprising a compound of the formula (I) according to claim 1 or an agrochemical formulation thereof for controlling one or more animal pests.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 15, 2018
From: FISCHER, RUEDIGER, DR.; WILCKE, DAVID, DR.; HAGER, DOMINIK, DR.; ILG, KERSTIN, DR.; EILMUS, SASCHA, DR.; GOERGENS, ULRICH; TURBERG, ANDREAS, DR.
To: BAYER CROPSCIENCE AKTIENGESELLSCHAFT
Reel/Frame 044947/0823 →
Priority Claims (1)
EP 15162775 · Apr 8, 2015 · regional
Continuity (1)
Related Publication 20180116222A1 · May 3, 2018
Cited By (1)
US 50,663