IP Library Granted Patent US 10,272,084
Granted Patent B2
US 10,272,084 · App. 15/170,335 · Granted Apr 30, 2019

Histone deacetylase 6 selective inhibitors for the treatment of cisplatin-induced peripheral neuropathy

Inventors: Annemieke Kavelaars (Houston, TX); Cobi J. Heijnen (Houston, TX); Karen Krukowski (San Francisco, CA); Matthew B. Jarpe (Quincy, MA)
Assignees: Regenacy Pharmaceuticals, LLC; Board of Regents, The University of Texas System
A61K31/505A61K33/24
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Quick Facts
Patent No.
US 10,272,084
App. No.
15/170,335
Granted
Apr 30, 2019
Kind
B2
Abstract

Disclosed are methods for treating cisplatin-induced peripheral neuropathy in a subject in need thereof comprising administering to the subject a therapeutically effective amount of a histone deacetylase 6 selective inhibitor.

Claims (7)

1. A method of alleviating numbness associated with cisplatin-induced peripheral neuropathy in a subject in need thereof comprising administering to the subject a therapeutically effective amount of a histone deacetylase 6 selective inhibitor, to thereby alleviate the numbness associated with the cisplatin-induced peripheral neuropathy.

2. The method of claim 1 , wherein the histone deacetylase 6 selective inhibitor is compound 001:

or a pharmaceutically acceptable salt thereof.

3. The method of claim 1 , wherein the histone deacetylase 6 selective inhibitor is co-administered with cisplatin.

4. The method of claim 1 , wherein the histone deacetylase 6 selective inhibitor is administered before or after administering cisplatin.

5. The method of claim 1 , wherein the cisplatin-induced peripheral neuropathy exists in the subject prior to administering the histone deacetylase 6 selective inhibitor.

6. The method of claim 1 , further comprising assessing numbness in the subject following treatment with the histone deacetylase 6 selective inhibitor.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 3, 2017
From: ACETYLON PHARMACEUTICALS INC
To: REGENACY PHARMACEUTICALS, LLC
Reel/Frame 044032/0220 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 22, 2016
From: KAVELAARS, ANNEMIEKE; HEIJNEN, COBI J.; KRUKOWSKI, KAREN
To: BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM
Reel/Frame 040398/0001 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 18, 2016
From: JARPE, MATTHEW B.
To: ACETYLON PHARMACEUTICALS, INC.
Reel/Frame 040371/0442 →
Continuity (2)
Provisional Application 62169528 · Jun 1, 2015
Related Publication 20160346279A1 · Dec 1, 2016
Cited By (1)
US 12,590,084