IP Library › Granted Patent US 10,306,874
Granted Patent B2
US 10,306,874 · App. 15/355,392 · Granted Jun 4, 2019

Non-human animals having a humanized lymphocyte-activation gene 3

Inventors: Alexander O. Mujica (Elmsford, NY); Elena Burova (Mount Kisco, NY); Andrew J. Murphy (Croton-on Hudson, NY)
Assignee: REGENERON PHARMACEUTICALS, INC.
A01K67/0278A01K67/0276A61K49/0008C07K14/70503A01K2207/15A01K2217/072A01K2217/075A01K2217/15A01K2227/105A01K2267/01A01K2267/03A01K2267/0331C07H21/04C12N2517/02
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Quick Facts
Patent No.
US 10,306,874
App. No.
15/355,392
Granted
Jun 4, 2019
Kind
B2
Abstract

Non-human animals, and methods and compositions for making and using the same, are provided, wherein the non-human animals comprise a humanization of a Lymphocyte activation gene 3 (Lag3). The non-human animals may be described, in some embodiments, as having a genetic modification to an endogenous Lag3 locus so that the non-human animals express a Lag3 polypeptide that includes a human portion and an endogenous portion (e.g., a non-human portion).

Claims (19)

1. A mouse whose genome comprises a humanized Lymphocyte activation gene 3 (Lag-3) gene at an endogenous Lag-3 locus,

wherein a humanized Lag-3 polypeptide is expressed from the humanized Lag-3 gene on the surface of activated T-lymphocytes in the mouse,

wherein the humanized Lag-3 polypeptide comprises (i) the first two N-terminal immunoglobulin-like domains of a human LAG-3 polypeptide and (ii) the transmembrane and intracellular domains of an endogenous mouse Lag-3 polypeptide, and

wherein the humanized Lag-3 gene is operably linked to the endogenous mouse Lag-3 promoter at the endogenous Lag-3 locus.

2. The mouse of claim 1 , wherein the humanized Lag-3 polypeptide comprises amino acids 29-260 of the human LAG-3 polypeptide, wherein the human LAG-3 polypeptide comprises the amino acid sequence as set forth in SEQ ID No. 6.

3. The mouse of claim 1 , wherein the humanized Lag-3 gene comprises endogenous mouse Lag-3 exons 1, 5, 6, 7 and 8.

4. The mouse of claim 1 , wherein the humanized Lag-3 gene comprises exons 2-4 of a human LAG-3 gene.

5. A humanized Lag-3 polypeptide produced by the mouse of claim 1 .

6. An isolated cell or tissue of the mouse of claim 1 , wherein the genome of the isolated cell or tissue comprises the humanized Lag-3 gene at the endogenous Lag-3 locus.

7. A method of making a mouse comprising

modifying a mouse genome so that the modified genome comprises a humanized Lag-3 gene at an endogenous Lag-3 locus, thereby making the mouse,

wherein a humanized Lag-3 polypeptide is expressed from the humanized Lag-3 gene on the surface of activated T-lymphocytes in the mouse, and

wherein the humanized Lag-3 polypeptide comprises (i) the first two N-terminal immunoglobulin-like domains of a human LAG-3 polypeptide and (ii) the transmembrane and intracellular domains of an endogenous mouse Lag-3 polypeptide, and

wherein the humanized Lag-3 gene is operably linked to the endogenous mouse Lag-3 promoter at the endogenous Lag-3 locus.

8. The method of claim 7 , comprising

(a) integrating a genomic fragment into an endogenous Lag-3 gene in a mouse ES cell, the genomic fragment comprising a nucleotide sequence that encodes the first two N-terminal immunoglobulin-like domains of the human LAG-3 polypeptide, thereby obtaining a genetically modified mouse embryonic stem cell; and,

(c) creating a mouse using the genetically modified mouse ES cell of (a).

9. The method of claim 7 , wherein the humanized Lag-3 gene comprises exons 2-4 of a human LAG-3 gene.

10. The method of claim 7 , wherein the humanized Lag-3 gene encodes at least amino acids 29-260 of the human LAG-3 polypeptide, wherein the human LAG-3 polypeptide comprises the amino acid sequence as set forth in SEQ ID No. 6.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 15, 2017
From: MUJICA, ALEXANDER O.; BUROVA, ELENA; MURPHY, ANDREW J.
To: REGENERON PHARMACEUTICALS, INC.
Reel/Frame 041262/0441 →
Continuity (3)
Provisional Application 62258181 · Nov 20, 2015
Provisional Application 62370430 · Aug 3, 2016
Related Publication 20170142943A1 · May 25, 2017