IP Library Granted Patent US 10,377,761
Granted Patent B2
US 10,377,761 · App. 16/045,371 · Granted Aug 13, 2019

Pyrrolo[1,2-f][1,2,4]triazines useful for treating respiratory syncitial virus infections

Inventors: Michael O'Neil Hanrahan Clarke (Redwood City, CA); Edward Doerffler (Foster City, CA); Richard L. Mackman (Millbrae, CA); Dustin Siegel (Half Moon Bay, CA)
Assignee: Gilead Sciences, Inc.
C07D487/04C07D405/04C07D405/14C07F9/6561C07H7/06
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Quick Facts
Patent No.
US 10,377,761
App. No.
16/045,371
Granted
Aug 13, 2019
Kind
B2
Abstract

Provided herein are formulations, methods and substituted tetrahydrofuranyl-pyrrolo[1,2-f][1,2,4]triazine-4-amine compounds of Formula (I) for treating Pneumovirinae virus infections, including respiratory syncytial virus infections, as well as methods and intermediates for synthesis of tetrahydrofuranyl-pyrrolo[1,2-f][1,2,4]triazine-4-amine compounds.

Claims (18)

1. A compound of formula:

or a pharmaceutically acceptable salt thereof.

2. A compound of formula:

or a pharmaceutically acceptable salt thereof.

3. A compound of formula:

4. A compound of formula:

5. A pharmaceutical composition comprising the compound or the pharmaceutically acceptable salt of claim 1 .

6. A pharmaceutical composition comprising the compound or the pharmaceutically acceptable salt of claim 2 .

7. A pharmaceutical composition comprising the compound of claim 3 .

8. A pharmaceutical composition comprising the compound of claim 4 .

9. A method of treating a Pneumovirinae virus infection in a human, the method comprising administering to the human a therapeutically effective amount of the compound or the pharmaceutically acceptable salt of claim 1 .

10. The method of claim 9 , wherein the Pneumovirinae virus infection in the human is a human respiratory syncytial virus infection.

11. A method of treating a Pneumovirinae virus infection in a human, the method comprising administering to the human a therapeutically effective amount of the compound or the pharmaceutically acceptable salt of claim 2 .

12. The method of claim 11 , wherein the Pneumovirinae virus infection in the human is a human respiratory syncytial virus infection.

13. A method of treating a Pneumovirinae virus infection in a human, the method comprising administering to the human a therapeutically effective amount of the compound of claim 3 .

14. The method of claim 13 , wherein the Pneumovirinae virus infection in the human is a human respiratory syncytial virus infection.

15. A method of treating a Pneumovirinae virus infection in a human, the method comprising administering to the human a therapeutically effective amount of the compound of claim 4 .

16. The method of claim 15 , wherein the Pneumovirinae virus infection in the human is a human respiratory syncytial virus infection.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 17, 2018
From: HANRAHAN CLARKE, MICHAEL O'NEIL; DOERFFLER, EDWARD; MACKMAN, RICHARD L.; SIEGEL, DUSTIN
To: GILEAD SCIENCES, INC.
Reel/Frame 046852/0645 →
Continuity (5)
Continuation 15610104 · May 31, 2017
Continuation 15182529 · Jun 14, 2016
Continuation 14534715 · Nov 6, 2014
Provisional Application 61902544 · Nov 11, 2013
Related Publication 20190055253A1 · Feb 21, 2019
Cited By (8)
US 12,264,173 US 12,297,226 US 12,357,577 US 12,404,289 US 12,448,383 US 12,509,466 US 12,655,172 US 12,723,057