IP Library Granted Patent US 10,414,771
Granted Patent B2
US 10,414,771 · App. 15/821,184 · Granted Sep 17, 2019

Compounds useful for inhibiting metastasis from cancer and methods using same

Inventors: Alessandro Fatatis (Penn Valley, PA); Joseph M. Salvino (Chester Springs, PA); Olimpia Meucci (Penn Valley, PA); Whitney L. Gladney (Glenolden, PA)
Assignees: Drexel University; Alliance Discovery, Inc.
C07D487/04A61K31/451A61K31/453A61K31/7088A61K39/3955C07D403/04C07K16/28
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Quick Facts
Patent No.
US 10,414,771
App. No.
15/821,184
Granted
Sep 17, 2019
Kind
B2
Abstract

The present invention includes compositions that are useful in preventing or treating metastasis in a subject diagnosed with cancer. The present invention also includes methods of preventing or treating metastasis in a subject diagnosed with cancer, wherein the method comprises administering to the subject in need thereof an effective amount of a pharmaceutical formulation comprising at least one pharmaceutically acceptable carrier and at least one CX 3 CR1 or fractalkine antagonist.

Claims (14)

1. A compound of Formula (IX):

R A —R B   (IX)

wherein:

R A is selected from the group consisting of:

 and

R B is selected from the group consisting of:

or a pharmaceutically acceptable salt thereof.

2. A pharmaceutical composition comprising a compound of Formula (IX) and at least one pharmaceutically acceptable carrier, wherein the compound of Formula (IX) is:

R A —R B   (IX)

wherein:

R A is selected from the group consisting of:

 and

R B is selected from the group consisting of:

or a pharmaceutically acceptable salt thereof.

Continuity (5)
Continuation 15174227 · Jun 6, 2016
Continuation 13776220 · Feb 25, 2013
Continuation 13312540 · Dec 6, 2011
Provisional Application 61420640 · Dec 7, 2010
Related Publication 20180099972A1 · Apr 12, 2018
Cited By (2)
US 12,605,394 US 12,667,578