IP Library Granted Patent US 10,640,468
Granted Patent B2
US 10,640,468 · App. 15/757,177 · Granted May 5, 2020

1-(4-(2-((1-(3,4-difluorophenyl)-1H-pyrazol-3-Yl)methoxy)ethyl)piperazin-1- Yl)ethanone salts

Inventors: Antoni Torrens-Jover (Barcelona, ES); Carmen Almansa-Rosales (Barcelona, ES)
Assignee: ESTEVE PHARMACEUTICALS, S.A.
C07D231/12C07D403/12C07B2200/13
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Quick Facts
Patent No.
US 10,640,468
App. No.
15/757,177
Granted
May 5, 2020
Kind
B2
Abstract

The present invention relates to 1-(4-(2-((1-(3,4-difluorophenyl)-1H-pyrazol-3-yl)methoxy)ethy)piperazin-1-y)ethanone salts, specifically to the hydrochloride and to the maleate, to pharmaceutical compositions comprising them, and to their use in therapy and/or prophylaxis of sigma receptor associated diseases.

Claims (5)

1. A crystalline salt of 1-(4-(2-((1-(3,4-difluorophenyl)-1H-pyrazol-3-yl)methoxy)ethyl)piperazin-1-yl)ethanone, wherein said salt is selected from hydrochloride, maleate, fumarate, succinate, oxalate and/or hydrobromide.

2. The crystalline salt according to claim 1 wherein the salt is the hydrochloride salt of 1-(4-(2-((1-(3,4-difluorophenyl)-1H-pyrazol-3-yl)methoxy)ethyl)piperazin-1-yl)ethanone.

3. The crystalline salt according to claim 1 wherein the salt is the maleate salt of 1-(4-(2-((1-(3,4-difluorophenyl)-1H-pyrazol-3-yl)methoxy)ethyl)piperazin-1-yl)ethanone.

4. A pharmaceutical composition comprising at least a crystalline salt according to claim 1 .

5. A method for the manufacture of a medicament comprising combining the crystalline salt as defined in claim 1 with a pharmaceutically acceptable excipient.

Assignments (2)
CHANGE OF NAME Recorded Dec 17, 2018
From: LABORATORIOS DEL DR. ESTEVE S.A.
To: ESTEVE PHARMACEUTICALS, S.A.
Reel/Frame 047931/0001 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 2, 2018
From: TORRENS-JOVER, ANTONI; ALMANSA ROSALES, CARMEN
To: LABORATORIOS DEL DR. ESTEVE, S.A.
Reel/Frame 045092/0707 →
Priority Claims (1)
EP 15382436 · Sep 2, 2015 · regional
Continuity (1)
Related Publication 20180251430A1 · Sep 6, 2018