IP Library Granted Patent US 10,646,580
Granted Patent B2
US 10,646,580 · App. 15/801,892 · Granted May 12, 2020

Oligosaccharide conjugates for targeting bacteria and uses related thereto

Inventors: Niren Murthy (Berkeley, CA); Eric Seth Gilbert (Decatur, GA); Xinghai Ning (Athens, GA); Mark Goodman (Atlanta, GA); Bryan Stubblefield (Atlanta, GA)
Assignees: Emory University; Georgia Tech Research Corporation; Georgia State University Research Foundation, Inc.
A61K47/61A61K31/496A61K45/06A61K49/0021A61K49/0032A61K49/0054A61K51/06A61K51/065C08B31/00C08L3/04
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Quick Facts
Patent No.
US 10,646,580
App. No.
15/801,892
Granted
May 12, 2020
Kind
B2
Abstract

This disclosure relates to conjugates for targeting bacteria and related uses. In certain embodiments, the disclosure relates to methods of transferring a molecule of interest into bacteria comprising mixing bacteria with a non-naturally occurring conjugate under conditions such that the conjugate is transported across the bacterial cell wall. Typically, the conjugate comprises an oligosaccharide and a molecule of interest. In certain embodiments, the molecule of interest may be a tracer or an antibiotic.

Claims (12)

1. An imaging method for a bacterial infection comprising a) administering a tracer molecule comprising a radionuclide or fluorescent molecule conjugated to maltodextrin to a subject; and b) determining whether the subject has a bacterial infection by scanning the subject and detecting a positron emitting or single photon emitting radionuclide or fluorescent molecule with an emission wavelength between 400 nm and 1200 nm.

2. The imaging method of claim 1 , further comprising the step of creating an image highlighting the location of the tracer molecule conjugated to maltodextrin in the subject.

3. The method of claim 1 , wherein the tracer molecule comprises a radionuclide, wherein the radionuclide is a positron-emitting radionuclide.

4. The method of claim 3 , wherein the positron-emitting radionuclide is selected from carbon-11, nitrogen-13, oxygen-15, fluorine-18, rubidium-82, and strontium-82.

5. The method of claim 1 , wherein the tracer molecule is a fluorescent molecule.

6. The method of claim 5 , wherein the fluorescent molecule is a fluorescent dye.

7. The method of claim 1 , wherein the maltodextrin comprises 2, 3, 4, 5, or 6 sugar oligomers.

8. The method of claim 1 , wherein the maltodextrin comprises greater than 2 glucose oligomers.

9. The method of claim 1 , wherein the tracer molecule comprises a positron-emitting radionuclide.

10. The method of claim 1 , wherein the tracer molecule conjugated to maltodextrin is

11. An imaging method for a bacterial infection comprising a) administering a tracer molecule comprising a radionuclide or fluorescent molecule conjugated to an oligosaccharide linked by an alpha 1, 4-covalent bond to a subject; and b) determining whether the subject has a bacterial infection by scanning the subject and detecting a positron emitting or single photon emitting radionuclide or fluorescent molecule with an emission wavelength between 400 nm and 1200 nm.

12. The method of claim 1 , wherein the tracer molecule comprises a radionuclide, wherein the radionuclide is a single photon emitting computed tomography radionuclide.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 7, 2018
From: GILBERT, ERIC SETH; STUBBLEFIELD, BRYAN
To: GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION, INC.
Reel/Frame 045732/0323 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 7, 2018
From: GOODMAN, MARK
To: EMORY UNIVERSITY
Reel/Frame 045732/0327 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 7, 2018
From: MURTHY, NIREN; NING, XINGHAI
To: GEORGIA TECH RESEARCH CORPORATION
Reel/Frame 045732/0333 →
Continuity (4)
Division 14190928 · Feb 26, 2014
Continuation 13979382
Provisional Application 61432668 · Jan 14, 2011
Related Publication 20180125991A1 · May 10, 2018