IP Library › Granted Patent US 10,828,345
Granted Patent B2
US 10,828,345 · App. 16/159,282 · Granted Nov 10, 2020

Use of a VEGF antagonist to treat angiogenic eye disorders

Inventor: George D. Yancopoulos (Yorktown Heights, NY)
Assignee: REGENERON PHARMACEUTICALS, INC.
A61K38/179A61K9/0048C07K14/71C07K16/22A61K2039/505C07K2319/30C07K2319/32
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Quick Facts
Patent No.
US 10,828,345
App. No.
16/159,282
Granted
Nov 10, 2020
Kind
B2
Abstract

The present invention provides methods for treating angiogenic eye disorders by sequentially administering multiple doses of a VEGF antagonist to a patient. The methods of the present invention include the administration of multiple doses of a VEGF antagonist to a patient at a frequency of once every 8 or more weeks. The methods of the present invention are useful for the treatment of angiogenic eye disorders such as age related macular degeneration, diabetic retinopathy, diabetic macular edema, central retinal vein occlusion, branch retinal vein occlusion, and corneal neovascularization.

Claims (13)

1. A method for treating an angiogenic eye disorder in a patient, said method comprising sequentially administering to the patient a single initial dose of a VEGF antagonist, followed by one or more secondary doses of the VEGF antagonist, followed by one or more tertiary doses of the VEGF antagonist;

wherein each secondary dose is administered 4 weeks after the immediately preceding dose; and wherein each tertiary dose is administered 12 weeks after the immediately preceding dose;

wherein the VEGF antagonist is a receptor-based chimeric molecule comprising an immunoglobin-like (Ig) domain 2 of a first VEGF receptor which is Flt1 and Ig domain 3 of a second VEGF receptor which is Flk1, and a multimerizing component.

2. The method of claim 1 , wherein the VEGF antagonist is aflibercept.

3. The method of claim 1 , wherein all doses of the VEGF antagonist are administered to the patient by intraocular administration.

4. The method of claim 3 , wherein the intraocular administration is intravitreal administration.

5. The method of claim 4 , wherein all doses of the VEGF antagonist comprise from about 0.5 mg to about 2 mg of the VEGF antagonist.

6. The method of claim 5 , wherein all doses of the VEGF antagonist comprise 0.5 mg of the VEGF antagonist.

7. The method of claim 5 , wherein all doses of the VEGF antagonist comprise 2 mg of the VEGF antagonist.

8. The method of claim 5 , wherein the angiogenic eye disorder is selected from the group consisting of: age related macular degeneration, diabetic retinopathy, diabetic macular edema, central retinal vein occlusion, branch retinal vein occlusion, and corneal neovascularization.

9. The method of claim 8 wherein the angiogenic eye disorder is age related macular degeneration.

10. The method of claim 8 wherein the angiogenic eye disorder is diabetic retinopathy.

11. The method of claim 8 , wherein the angiogenic eye disorder is diabetic macular edema.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 4, 2019
From: YANCOPOULOS, GEORGE D.
To: REGENERON PHARMACEUTICALS, INC.
Reel/Frame 047899/0083 →
Continuity (8)
Continuation 15471506 · Mar 28, 2017
Continuation 14972560 · Dec 17, 2015
Continuation 13940370 · Jul 12, 2013
Continuation In Part PCTUS2012020855 · Jan 11, 2012
Provisional Application 61432245 · Jan 13, 2011
Provisional Application 61434836 · Jan 21, 2011
Provisional Application 61561957 · Nov 21, 2011
Related Publication 20190046609A1 · Feb 14, 2019
Cited By (11)
US 1,116,103 US 1,120,314 US 12,268,730 US 12,274,865 US 12,280,093 US 12,571,027 US 12,643,958 US 12,649,031 US 12,691,227 US 12,734,300 US 12,741,098