IP Library › Granted Patent US 10,864,212
Granted Patent B2
US 10,864,212 · App. 16/361,810 · Granted Dec 15, 2020

Compositions and methods for treating retinal degradation

Inventors: Jayakrishna Ambati (Lexington, KY); Benjamin Fowler (Lexington, KY)
Assignee: University of Kentucky Research Foundation
A61K31/506A61K31/513A61K31/52A61K31/706A61K31/7052A61K31/7064A61K31/7068A61K31/7072A61K31/7076C07D405/04C07D411/04A61P25/16A61P25/28
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 10,864,212
App. No.
16/361,810
Granted
Dec 15, 2020
Kind
B2
Abstract

The present disclosure relates to compositions and methods for treating retinal damage and/or retinal degradation. More specifically, this disclosure relates to methods for treating degradation of the retinal pigment epithelium by administering compositions comprising a nucleoside and/or a nucleoside or nucleotide reverse transcriptase inhibitor.

Claims (53)

1. A method of treating a condition selected from Parkinson's disease, Alzheimer's disease, and multiple sclerosis comprising administering to a subject in need thereof a compound selected from:

(i) a compound having the structure of formula I

or a pharmaceutically acceptable salt thereof;

(ii) a compound having the structure of formula II

(iii) a compound having the structure of formula III, or a pharmaceutically acceptable salt thereof;

(iv) a compound having the structure of formula IV,

wherein n is 10 to 20;

(v) a compound having the structure of formula V

(vi) stavudine (d4T);

(vii) lamivudine (3TC);

(viii) cordycepin;

(ix) azidothymidine (AZT);

(x) abacavir (ABC); and

(xi) a combination thereof.

2. The method of claim 1 , wherein the compound is selected from:

(i) the compound having the structure of formula I

or a pharmaceutically acceptable salt thereof;

(ii) the compound having the structure of formula II

(iii) the compound having the structure of formula III, or a pharmaceutically acceptable salt thereof;

(iv) the compound having the structure of formula IV,

wherein n is 10 to 20;

(v) a compound having the structure of formula V

(vi) a combination thereof.

3. The method of claim 1 , wherein n is 11.

4. The method of claim 1 , wherein the compound is selected from:

(i) the compound having the structure of formula

or a pharmaceutically acceptable salt thereof;

(ii) the compound having the structure of formula II

and

(iii) a compound having the structure of formula V

and

(iv) a combination thereof.

5. The method of claim 1 , wherein the compound is selected from:

(i) the compound having the structure of formula

or a pharmaceutically acceptable salt thereof;

(ii) a compound having the structure of formula V

and

(iii) a combination thereof.

6. The method of claim 1 , wherein the compound is a compound having the structure of formula I

or a pharmaceutically acceptable salt thereof.

7. The method of claim 1 , wherein the compound is the compound having the structure of formula II:

8. The method of claim 1 , wherein the compound is the compound having the structure of formula V:

9. The method of claim 1 , wherein the compound is selected from

(vi) stavudine (d4T);

(vii) lamivudine (3TC);

(viii) cordycepin;

(ix) azidothymidine (AZT);

(x) abacavir (ABC); and

(xi) a combination thereof.

10. The method of claim 1 , wherein the method comprises administering a composition comprising the compound and a pharmaceutically acceptable carrier.

11. The method of claim 1 , wherein the condition is Parkinson's disease.

12. The method of claim 1 , wherein the condition is Alzheimer's disease.

13. The method of claim 1 , wherein the condition is multiple sclerosis.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 25, 2019
From: AMBATI, JAYAKRISHNA; FOWLER, BENJAMIN
To: UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION
Reel/Frame 048688/0939 →
Continuity (5)
Continuation 15142087 · Apr 29, 2016
Continuation 14450000 · Aug 1, 2014
Provisional Application 61861290 · Aug 1, 2013
Provisional Application 61987612 · May 2, 2014
Related Publication 20190255049A1 · Aug 22, 2019
Cited By (1)
US 12,274,701