IP Library Granted Patent US 10,865,200
Granted Patent B2
US 10,865,200 · App. 16/209,349 · Granted Dec 15, 2020

Nitrogen-containing heterocyclic compound

Inventors: Masami Yamada (Kanagawa, JP); Shinkichi Suzuki (Kanagawa, JP); Takahiro Sugimoto (Kanagawa, JP); Minoru Nakamura (Kanagawa, JP); Hiroki Sakamoto (Kanagawa, JP); Makoto Kamata (Kanagawa, JP)
Assignee: Takeda Pharmaceutical Company Limited
C07D405/14A61K31/045A61K31/13A61K31/325A61K31/4035A61K31/4155A61K31/445A61K31/4406A61K31/4439A61K31/55C07D209/46C07D401/06C07D401/10C07D401/14C07D403/04C07D403/10C07D405/04C07D471/04
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Quick Facts
Patent No.
US 10,865,200
App. No.
16/209,349
Granted
Dec 15, 2020
Kind
B2
Abstract

The present invention provides a compound having a cholinergic muscarinic M1 receptor positive allosteric modulator activity and useful as an agent for the prophylaxis or treatment of Alzheimer's disease, schizophrenia, pain, sleep disorder, Parkinson's disease dementia, dementia with Lewy bodies, and the like. The present invention relates to a compound represented by the formula (I) or a salt thereof. wherein each symbol is as described in the specification, or a salt thereof.

Claims (3)

1. A method for the treatment of cognitive impairment associated with schizophrenia or Parkinson's disease in a mammal, which comprises administering an effective amount of 2-[(3S,4S)-4-hydroxytetrahydro-2H-pyran-3-yl]-6-(4-methoxybenzyl)-4,5-dimethyl-2,3-dihydro-1H-isoindol-1-one or a salt thereof to the mammal.

2. A method for the treatment of cognitive impairment associated with schizophrenia or Parkinson's disease in a mammal, which comprises administering an effective amount of 4-fluoro-2-[(3S,4S)-4-hydroxytetrahydro-2H-pyran-3-yl]-5-methyl-6-[4-(1H-pyrazol-1-yl)benzyl]-2,3-dihydro-1H-isoindol-1-one or a salt thereof to the mammal.

3. A method for the treatment of cognitive impairment associated with schizophrenia or Parkinson's disease in a mammal, which comprises administering an effective amount of 2-((1 S,2 S)-2-hydroxycyclohexyl)-4,5-dimethyl-6-((6-methylpyridin-3-yl)methyl)isoindolin-1-one or a salt thereof to the mammal.

Priority Claims (1)
JP 2014-089585 · Apr 23, 2014 · national
Continuity (7)
Continuation 15685800 · Aug 24, 2017
Continuation 15608565 · May 30, 2017
Continuation 15488002 · Apr 14, 2017
Continuation 15291769 · Oct 12, 2016
Continuation 15013625 · Feb 2, 2016
Continuation 14693342 · Apr 22, 2015
Related Publication 20190241547A1 · Aug 8, 2019