IP Library Granted Patent US 11,007,208
Granted Patent B2
US 11,007,208 · App. 16/863,566 · Granted May 18, 2021

Methods for treating arenaviridae and coronaviridae virus infections

Inventors: Michael O' Neil Hanrahan Clarke (Redwood City, CA); Joy Yang Feng (Hillsborough, CA); Robert Jordan (Foster City, CA); Richard L. Mackman (Millbrae, CA); Adrian S. Ray (Burlingame, CA); Dustin Siegel (Half Moon Bay, CA)
Assignee: Gilead Sciences, Inc.
A61K31/706A61K31/7056
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Quick Facts
Patent No.
US 11,007,208
App. No.
16/863,566
Granted
May 18, 2021
Kind
B2
Abstract

Provided are methods for treating Arenaviridae and Coronaviridae virus infections by administering nucleosides and prodrugs thereof, of Formula I: wherein the 1′ position of the nucleoside sugar is substituted. The compounds, compositions, and methods provided are particularly useful for the treatment of Lassa virus and Junin virus infections.

Claims (14)

1. A method of treating a Coronaviridae infection in a human in need thereof, comprising administering to the human a therapeutically effective amount of a compound having formula:

or a pharmaceutically acceptable salt thereof.

2. The method of claim 1 , comprising administering to the human a therapeutically effective amount of a compound having formula:

3. The method of claim 1 , further comprising administering a pharmaceutically acceptable carrier or excipient.

4. The method of claim 1 , further comprising administering a therapeutically effective amount of at least one other therapeutic agent.

5. The method of claim 4 , wherein the at least one other therapeutic agent is selected from the group consisting of a corticosteroid, an anti-inflammatory signal transduction modulator, β2-adrenoreceptor agonist bronchodilator, an anticholinergic, a mucolytic agent, hypertonic saline, and other drugs for treating a Coronaviridae virus infection; or mixtures thereof.

6. The method of claim 1 , wherein the Coronaviridae infection is caused by a Coronaviridae virus selected from the group consisting of SARS, MERS, 229E, NL63, OC43, and HKU1.

7. The method of claim 1 , wherein the Coronaviridae infection is caused by a SARS virus.

8. The method of claim 1 , wherein the Coronaviridae infection is caused by a MERS virus.

9. The method of claim 1 , wherein the compound, or a pharmaceutically acceptable salt thereof, is administered by oral, rectal, nasal, pulmonary, topical, vaginal, or parenteral administration.

10. The method of claim 9 , wherein the compound, or a pharmaceutically acceptable salt thereof, is administered by parenteral administration.

11. The method of claim 1 , wherein the compound, or a pharmaceutically acceptable salt thereof, is administered by subcutaneous, intramuscular, intravenous, intradermal, intrathecal, or epidural administration.

12. The method of claim 11 , wherein the compound, or a pharmaceutically acceptable salt thereof, is administered by intravenous administration.

13. The method of claim 1 , wherein the compound, or a pharmaceutically acceptable salt thereof, is administered by inhalation administration.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 12, 2020
From: CLARKE, MICHAEL O' NEIL HANRAHAN; FENG, JOY YANG; JORDAN, ROBERT; MACKMAN, RICHARD L.; RAY, ADRIAN S.; SIEGEL, DUSTIN
To: GILEAD SCIENCES, INC.
Reel/Frame 052642/0103 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 30, 2020
From: CLARKE, MICHAEL O' NEIL HANRAHAN; FENG, JOY YANG; JORDAN, ROBERT; MACKMAN, RICHARD L.; RAY, ADRIAN S.; SIEGEL, DUSTIN
To: GILEAD SCIENCES, INC.
Reel/Frame 052542/0593 →
Continuity (5)
Continuation 16265016 · Feb 1, 2019
Continuation 15267433 · Sep 16, 2016
Provisional Application 62219302 · Sep 16, 2015
Provisional Application 62239696 · Oct 9, 2015
Related Publication 20200352967A1 · Nov 12, 2020
Cited By (6)
US 12,297,226 US 12,357,577 US 12,404,289 US 12,448,383 US 12,509,466 US 12,655,172