IP Library Granted Patent US 11,046,774
Granted Patent B2
US 11,046,774 · App. 16/285,118 · Granted Jun 29, 2021

Method of treating or ameliorating metabolic disorders using binding proteins for gastric inhibitory peptide receptor (GIPR) in combination with GLP-1 agonists

Inventors: Junming Yie (Warren, NJ); Donghui Shi (Thousand Oaks, CA); David J. Lloyd (Thousand Oaks, CA); Jinghong Wang (Palo Alto, CA); Glenn N. Sivits, Jr. (Newbury Park, CA); Murielle M. Veniant-Ellison (Thousand Oaks, CA); Renee Komorowski (Ventura, CA); Neeraj Agrawal (Thousand Oaks, CA); Darren L. Bates (Oak Park, CA); Brandon C. P. Clavette (Coquitlam, CA); Ian N. Foltz (Burnaby, CA); Shu-yin Ho (Thousand Oaks, CA); Christopher Murawsky (Roberts Creek, CA); Xiaoshan Min (Burlingame, CA); Zhulun Wang (Palo Alto, CA)
Assignee: AMGEN INC.
C07K16/2869A61K9/0019A61K38/1703A61K38/26A61K39/3955A61K2039/505A61K2039/54C07K2299/00C07K2317/21C07K2317/32C07K2317/33C07K2317/41C07K2317/52C07K2317/71C07K2317/76C07K2317/92
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Quick Facts
Patent No.
US 11,046,774
App. No.
16/285,118
Granted
Jun 29, 2021
Kind
B2
Abstract

Methods of treating metabolic diseases and disorders using an antigen binding protein specific for the GIPR polypeptide are provided. In various embodiments the metabolic disease or disorder is type 2 diabetes, obesity, dyslipidemia, elevated glucose levels, elevated insulin levels and diabetic nephropathy. In certain embodiments the antigen binding protein is administered in combination with a GLP-1 receptor agonist.

Claims (18)

1. A method of treating a subject with a metabolic disorder, the method comprising administering to the subject a therapeutically effective amount of an antigen binding protein that specifically binds to a polypeptide comprising amino acids 1-139 of human Gastric Inhibitory Peptide Receptor (“GIPR”), wherein said antigen binding protein is an antibody and is an antagonist of GIPR.

2. The method of claim 1 , wherein said metabolic disorder is a disorder of glucose metabolism.

3. The method of claim 2 , wherein said glucose metabolism disorder comprises hyperglycemia and wherein said administering reduces plasma glucose in said subject.

4. The method of claim 2 , wherein said glucose metabolism disorder comprises hyperinsulinemia and wherein said administering reduces plasma insulin in said subject.

5. The method of claim 2 , wherein said glucose metabolism disorder comprises glucose intolerance and wherein said administering increases glucose tolerance in said subject.

6. The method of claim 2 , wherein said disorder of glucose metabolism comprises insulin resistance and wherein said administering decreases insulin resistance in said subject.

7. The method of claim 2 , wherein said glucose metabolism disorder comprises diabetes mellitus.

8. The method of claim 2 , wherein said subject is obese.

9. The method of claim 8 , wherein said administering reduces body weight in said subject.

10. The method of claim 8 , wherein said administering reduces body weight gain in said subject.

11. The method of claim 8 , where said administering reduces fat mass in said subject.

12. The method of claim 8 , wherein said disorder of glucose metabolism comprises insulin resistance and wherein said administering reduces insulin resistance in said subject.

13. The method of claim 8 , wherein said subject has increased liver steatosis, and wherein said administering reduces liver steatosis in said subject.

14. The method of claim 8 , wherein said subject has increased liver fat content, and wherein said administering reduces liver fat content in said subject.

15. The method of claim 1 , wherein said subject is a mammal.

16. The method of claim 1 , wherein said subject is human.

17. The method of claim 1 , wherein said administering is by parenteral injection.

18. The method of claim 1 , wherein said administering is by subcutaneous injection.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 7, 2019
From: YIE, JUNMING; SHI, DONGHUI; LLOYD, DAVID J; WANG, JINGHONG; SIVITS, JR., GLENN N; VENIANT-ELLISON, MURIELLE M; KOMOROWSKI, RENEE; AGRAWAL, NEERAJ; BATES, DARREN L; CLAVETTE, BRANDON C. P.; FOLTZ, IAN N; HO, SHU-YIN; MURAWSKY, CHRISTOPHER; MIN, XIAOSHAN; WANG, ZHULUN
To: AMGEN INC.
Reel/Frame 048535/0301 →
Continuity (5)
Division 15387542 · Dec 21, 2016
Provisional Application 62420415 · Nov 10, 2016
Provisional Application 62337799 · May 17, 2016
Provisional Application 62387486 · Dec 23, 2015
Related Publication 20190276546A1 · Sep 12, 2019
Cited By (4)
US 12,214,051 US 12,252,540 US 12,435,149 US 12,465,652