IP Library Granted Patent US 11,052,077
Granted Patent B2
US 11,052,077 · App. 17/150,467 · Granted Jul 6, 2021

Methods of treating lung cancer

Inventors: Sundar Srinivasan (Corona Del Mar, CA); Christina Chow (Seattle, WA)
Assignee: BOW RIVER LLC
A61K31/4468A61K9/0019A61K9/0053A61K9/0056A61K9/0078A61K9/0095A61K9/08A61K9/10A61K9/2004A61K9/4841A61K31/00A61K31/397A61K31/407A61K31/454A61K31/4745A61K31/497A61K31/498A61K31/4995A61K31/506A61K31/519A61K31/5383A61K31/5395A61P25/16A61P25/18A61P35/02A61P35/04
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Quick Facts
Patent No.
US 11,052,077
App. No.
17/150,467
Granted
Jul 6, 2021
Kind
B2
Abstract

The present disclosure provides for methods of treating a patient with a CYP3A4 substrate drug, wherein the patient is treated with posaconazole. In some embodiments, the patient stops posaconazole treatment, waits for at least 2 days, and then is treated with the CYP3A4 substrate drug as soon as it is safe to do so. In some embodiments, treatment with the CYP3A4 substrate drug is delayed for about 2-42 days after stopping posaconazole. In some embodiments, the patient is treated with a reduced dose of the CYP3A4 substrate drug for about 2-42 days.

Claims (28)

1. A method of treating lung cancer in a patient in need thereof with an antineoplastic drug which is a CYP3A4 substrate, wherein the patient is treated with posaconazole, comprising:

(a) stopping posaconazole treatment;

(b) delaying administering, for at least 9 days after stopping posaconazole treatment, a dose of the anti-neoplastic drug that the patient would have received based on the patient's age and condition of the patient had not been treated with posaconazole; and then

(c) administering the anti-neoplastic drug.

2. The method of claim 1 , wherein the patient is not obese.

3. The method of claim 1 , wherein the patient has at least one characteristic selected from the group consisting of the following:

i) BMI of at least about 35;

ii) waist size greater than about 42 inches;

iii) % body fat greater than about 40%;

iv) total body fat greater than about 40 kg, and;

v) medically diagnosed as obese.

4. The method of claim 1 , wherein said administering in step (c) is 9-21 days after stopping posaconazole in step (a).

5. The method of claim 1 , wherein said administering in step (c) is 9 days after stopping posaconazole in step (a).

6. The method of claim 1 , wherein said administering in step (c) is 10 days after stopping posaconazole in step (a).

7. The method of claim 1 , wherein said administering in step (c) is 11 days after stopping posaconazole in step (a).

8. The method of claim 1 , wherein said administering in step (c) is 12 days after stopping posaconazole in step (a).

9. The method of claim 1 , wherein said administering in step (c) is 13 days after stopping posaconazole in step (a).

10. The method of claim 1 , wherein said administering in step (c) is 14 days after stopping posaconazole in step (a).

11. The method of claim 1 , wherein said administering of step (c) is at least 21 days after stopping posaconazole in step (a).

12. The method of claim 1 , wherein said administering in step (c) is 9-42 days after stopping posaconazole in step (a).

13. The method of claim 1 , wherein the lung cancer is non-small cell lung cancer.

14. The method of claim 1 , wherein the anti-neoplastic drug is selected from the group consisting of erlotinib, crizotinib, dabrafenib, brigatinib, lorlatinib, and trastuzumab deruxtecan.

15. The method of claim 1 , wherein the anti-neoplastic drug is erlotinib.

16. The method of claim 1 , wherein the anti-neoplastic drug is crizotinib.

17. The method of claim 1 , wherein the anti-neoplastic drug is dabrafenib.

18. The method of claim 1 , wherein the anti-neoplastic drug is brigatinib.

19. The method of claim 1 , wherein the anti-neoplastic drug is lorlatinib.

20. The method of claim 1 , wherein the anti-neoplastic drug is trastuzumab deruxtecan.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 19, 2021
From: SRINIVASAN, SUNDAR; CHOW, CHRISTINA
To: BOW RIVER LLC
Reel/Frame 054949/0430 →
Continuity (4)
Continuation 17082902 · Oct 28, 2020
Continuation 16408931 · May 10, 2019
Continuation In Part 15596585 · May 16, 2017
Related Publication 20210154181A1 · May 27, 2021
Cited By (2)
US 12,318,384 US 12,453,730