IP Library › Granted Patent US 11,065,220
Granted Patent B2
US 11,065,220 · App. 16/485,735 · Granted Jul 20, 2021

Anti-pathogenic therapeutic compositions

Inventors: Weston J. Hale (Missoula, MT); Thomas F. Rau (Heidelberg Heights, AU)
Assignee: Wintermute Biomedical, Inc.
A61K31/198A61K9/0014A61K31/192A61K31/201A61K47/10A61P31/04
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Quick Facts
Patent No.
US 11,065,220
App. No.
16/485,735
Granted
Jul 20, 2021
Kind
B2
Abstract

Therapeutic compounds useful for the treatment of pathogens including bacteria (gram positive and gram negative, mycobacteria), some fungi and viruses. The compounds described herein may include a mixture of therapeutically-effective amounts of a polar amino acid, a CI 1 fatty acid, and an anthraquinone. The invention further provides for the administration of the therapeutic compounds to a patient (e.g., a human) suffering from an infection.

Claims (17)

1. An anti-pathogenic therapeutic composition comprising a mixture of L-Arginine, undecylenic acid and cassic acid, wherein the cassic acid is encapsulated in the undecylenic acid, and wherein the percentage of cassic acid in the mixture is greater than 0.03% w/w of the mixture.

2. The composition of claim 1 , wherein the percentage of cassic acid in the mixture is between 0.03% and 2.3% w/w of the mixture.

3. The composition of claim 1 , wherein the percentage of cassic acid in the mixture is between 0.1% and 1.0% w/w of the mixture.

4. The composition of claim 1 , wherein the percentage of L-Arginine in the mixture is between 47% and 73% w/w of the mixture.

5. The composition of claim 1 , wherein the percentage of undecylenic acid in the mixture is between 26% and 53% w/w of the mixture.

6. The composition of claim 1 , wherein the percentage of L-Arginine in the mixture is about 62% w/w of the mixture, and the percentage of undecylenic acid is about 37.6% w/w of the mixture, and the percentage of cassic acid is about 0.4% w/w of the mixture.

7. The composition of claim 1 , further comprising an excipient, diluent, or carrier.

8. The composition of claim 7 , wherein said excipient, diluent, or carrier comprises cetyl alcohol and water.

9. The composition of claim 7 , wherein said excipient, diluent, or carrier is configured for topical application.

10. The composition of claim 7 , wherein said excipient, diluent, or carrier comprises an emulsifying agent.

11. The composition of claim 1 , further comprising a cooling or heating additive.

12. The composition of claim 1 , wherein the concentration of cassic acid in the composition is greater than 0.1 mg/ml.

13. The composition of claim 1 , wherein the composition is configured as a liquid or emulsion in a form suitable for topical administration to a human.

14. The composition of claim 1 , wherein the composition is configured for one or more of: oral, parenteral, intraperitoneal, transmucosal, transdermal, rectal, inhalable, and topical administration.

15. The composition of claim 1 , wherein the composition is configured for coating a medical device.

16. An anti-pathogenic therapeutic composition effective against gram negative bacteria, the composition comprising a mixture of L-Arginine, undecylenic acid and cassic acid, wherein the cassic acid is encapsulated in the undecylenic acid, and wherein the percentage of cassic acid in the mixture is between 0.03% and 2.3% w/w of the mixture, the percentage of L-Arginine is between 47% and 73% w/w of the mixture, and the percentage of undecylenic acid in the mixture is between 26% and 53% w/w of the mixture.

17. An anti-pathogenic therapeutic composition effective against gram negative bacteria, the composition comprising a mixture of L-Arginine, undecylenic acid and cassic acid, wherein the cassic acid is encapsulated in the undecylenic acid, and wherein the percentage of cassic acid in the mixture is less than 5% w/w of the mixture, the percentage of L-Arginine is between 47% and 73% w/w of the mixture, and the percentage of undecylenic acid in the mixture is between 26% and 53% w/w of the mixture, further wherein the mixture is combined with an excipient, diluent, or carrier and the concentration of cassic acid in the composition is 0.1 mg/ml or greater.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 21, 2020
From: HALE, WESTON J.; RAU, THOMAS F.
To: WINTERMUTE BIOMEDICAL, INC.
Reel/Frame 051893/0246 →
Continuity (2)
Provisional Application 62458140 · Feb 13, 2017
Related Publication 20200046666A1 · Feb 13, 2020
Cited By (3)
US 12,186,293 US 12,324,797 US 12,383,524