IP Library Granted Patent US 11,124,553
Granted Patent B2
US 11,124,553 · App. 16/090,786 · Granted Sep 21, 2021

TDP-43 mitochondrial localization inhibitor for the treatment of neurogenerative disease

Inventor: Xinglong Wang (Cleveland, OH)
Assignee: CASE WESTERN RESERVE UNIVERSITY
C07K14/4713A61P25/28C07K7/06A61K38/00
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Quick Facts
Patent No.
US 11,124,553
App. No.
16/090,786
Granted
Sep 21, 2021
Kind
B2
Abstract

A method of treating a neurodegenerative disease in a subject includes administering to the subject a therapeutically effective amount of a TDP-43 mitochondrial localization inhibitor.

Claims (6)

1. A pharmaceutical composition comprising: a therapeutic agent that includes a synthetic therapeutic peptide of about 5 to about 10 amino acids in length that includes the amino acid sequence selected from the group consisting of SEQ ID NO: 1, SEQ ID NO: 3, and SEQ ID NO: 5 and a transport moiety that is linked to the therapeutic peptide and facilitates uptake of the therapeutic peptides by a cell, wherein the therapeutic peptide inhibits TDP-43 mediated disassembly of mitochondrial respiratory complex 1.

2. The composition of claim 1 , the therapeutic peptide including the amino acid sequence of SEQ ID NO: 1 or SEQ ID NO: 7.

3. The composition of claim 1 , the therapeutic peptide including the amino acid sequence of SEQ ID NO: 3 or SEQ ID NO: 8.

4. The composition of claim 1 , the therapeutic peptide including the amino acid sequence of SEQ ID NO: 5 or SEQ ID NO: 9.

5. The composition of claim 1 , the transport moiety comprising a TAT peptide.

6. The composition of claim 1 , the therapeutic agent having the amino acid sequence selected from the group consisting of SEQ ID NOs: 12-17.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 22, 2019
From: WANG, XINGLONG
To: CASE WESTERN RESERVE UNIVERSITY
Reel/Frame 049250/0197 →
Continuity (3)
Provisional Application 62319580 · Apr 7, 2016
Provisional Application 62328484 · Apr 27, 2016
Related Publication 20190211070A1 · Jul 11, 2019