IP Library › Granted Patent US 11,129,867
Granted Patent B2
US 11,129,867 · App. 16/264,702 · Granted Sep 28, 2021

Method of treating cancer cells

Inventors: Hui-Ching Wang (Hsinchu, TW); Dah-Tsyr Chang (Hsinchu, TW); Yu-Hsuen Tu (Hsinchu, TW); Ping-Hsueh Kuo (Hsinchu, TW)
Assignee: National Tsing Hua University
A61K38/08A61K31/352A61K41/0057A61K47/545A61K47/64A61P35/00A63F13/60A63F13/67G06N3/126G06T1/20A63F2300/60
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Quick Facts
Patent No.
US 11,129,867
App. No.
16/264,702
Granted
Sep 28, 2021
Kind
B2
Abstract

The present invention discloses a method of treating cancer cells. The method comprises administrating a composition comprises a rhodamine or rhodamine derivative conjugated to a peptide comprises an amino acid sequence of SEQ ID NO: 1 to a subject in need, and activate the composition with light.

Claims (12)

1. A method of treating head and neck squamous cell carcinoma, comprising:

administering a composition comprising a rhodamine or rhodamine derivative conjugated to a peptide comprising an amino acid sequence of SEQ ID NO: 1 to a subject suffering from head and neck squamous cell carcinoma, and

activating the composition with light, wherein the rhodamine or the rhodamine derivative is selected from the group consisting of: Carboxytetramethylrhodamine (TAMRA), Tetramethylrhodamine (TMR) and 5/6-tetramethyl-rhodamine isothiocyanate (TRITC).

2. The method of claim 1 , wherein the composition is administered into a mass of cancer cells of the head and neck squamous cell carcinoma.

3. The method of claim 1 , wherein the composition induces apoptosis of the cancer cells of the head and neck squamous cell carcinoma.

4. The method of claim 3 , wherein the apoptosis is independent of caspase activation.

5. The method of claim 1 , wherein the composition induces mitochondria fragmentation of the cancer cells of the head and neck squamous cell carcinoma.

6. The method of claim 1 , wherein the composition induces reactive oxygen species (ROS) generation of the cancer cells of the head and neck squamous cell carcinoma.

7. The method of claim 1 , wherein the composition induces DNA damage of the cancer cells of the head and neck squamous cell carcinoma.

8. The method of claim 1 , wherein the light is with a wavelength of 380 nm to 750 nm.

9. The method of claim 8 , wherein the light is with a wavelength of 400 nm to 620 nm.

10. The method of claim 9 , wherein the light is with a wavelength of 470 nm to 580 nm.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 1, 2019
From: WANG, HUI-CHING; CHANG, DAH-TSYR; TU, YU-HSUEN; KUO, PING-HSUEH
To: NATIONAL TSING HUA UNIVERSITY
Reel/Frame 048215/0050 →
Continuity (2)
Provisional Application 62576050 · Oct 23, 2017
Related Publication 20190151402A1 · May 23, 2019