IP Library Granted Patent US 11,246,844
Granted Patent B2
US 11,246,844 · App. 15/609,791 · Granted Feb 15, 2022

Methods for inhibiting conversion of choline to trimethylamine (TMA)

Inventors: Stanley Leon Hazen (Pepper Pike, OH); Jose Carlos Garcia-Garcia (Cincinnati, OH); George Franklin Gerberick (West Chester, OH); John August Wos (Mason, OH); Xiaodong Gu (Cleveland, OH); Michael Reilly (Lebanon, OH); Mark Robert Sivik (Mason, OH); Jodie Michelle Reed (Loveland, OH); David Blair Cody (West Harrison, OH)
Assignees: The Procter & Gamble Company; The Cleveland Clinic Foundation
A61K31/14A61K31/04A61K31/205A61K31/275C07C11/02C07C11/22C07C13/04C07C69/003C07C69/01C07C211/62C07C211/63C07C215/40C07C217/40C07C219/08C07C229/12C07C229/22C07C229/30C07C233/02C07C237/06C07C255/07C07C255/24C07D211/46C07D303/04C07D303/36C07D451/02C07C2601/02
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Quick Facts
Patent No.
US 11,246,844
App. No.
15/609,791
Granted
Feb 15, 2022
Kind
B2
Abstract

A method of inhibiting the conversion of choline to trimethylamine (TMA) and lowering TMAO by providing a composition comprising a compound set forth in Formula (I):

Claims (3)

1. A method of inhibiting the conversion of choline to trimethylamine (TMA) and reducing TMAO level in an individual comprising administering to the individual a composition comprising a compound selected from the group consisting of: N-(2,2-dimethoxyethyl)-N,N-dimethylprop-2-yn-1-aminium, N-(2,2-dihydroxyethyl)-N,N-dimethylprop-2-yn-1-aminium, N-(2-hydroxyethyl)-N,N-dimethylbut-3-yn-1-aminium, N-(2,2-diethoxyethyl)-N,N-dimethylprop-2-yn-1-aminium, 4-hydroxy-1-methyl-1-(prop-2-yn-1-yl)piperidin-1-ium, 2-cyano-N,N-dimethyl-N-(prop-2-yn-1-yl)prop-2-en-1-aminium, trimethyl(prop-2-ynyl)ammonium, allyl-(cyanomethyl)-dimethyl-ammonium, or N-(2-hydroxyethyl)-N,N-dimethylprop-2-yn-1-aminium, and a pharmaceutically acceptable salt thereof.

2. The method of claim 1 further comprising administering to the individual a second agent selected from the group consisting of Omega 3 oil, salicylic acid, dimethylbutanol, garlic oil, olive oil, krill oil, Co enzyme Q-10, a probiotic, a prebiotic, dietary fiber, psyllium husk, bismuth salts, phytosterols, grape seed oil, green tea extract, vitamin D, an antioxidant, turmeric, curcumin, and resveratrol.

3. The method of claim 1 , comprising administering the compound to an individual having an elevated level of TMAO in blood, plasma, serum, or urine, and combinations thereof.

Assignments (4)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 8, 2019
From: HAZEN, STANLEY LEON; GU, XIAODONG
To: THE CLEVELAND CLINIC FOUNDATION
Reel/Frame 047925/0480 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 8, 2019
From: GARCIA-GARCIA, JOSE CARLOS; GERBERICK, GEORGE FRANKLIN; WOS, JOHN AUGUST; REILLY, MICHAEL; SIVIK, MARK ROBERT; REED, JODIE MICHELLE; CODY, DAVID BLAIR
To: THE PROCTER & GAMBLE COMPANY
Reel/Frame 047925/0484 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 8, 2019
From: HAZEN, STANLEY LEON; GU, XIAODONG
To: THE CLEVELAND CLINIC FOUNDATION
Reel/Frame 047926/0631 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 7, 2019
From: GARCIA-GARCIA, JOSE CARLOS (NMN); GERBERICK, GEORGE FRANKLIN; WOS, JOHN AUGUST; REILLY, MICHAEL (NMN); SIVIK, MARK ROBERT; REED, JODIE MICHELLE; CODY, DAVID BLAIR
To: THE PROCTER & GAMBLE COMPANY
Reel/Frame 047921/0001 →
Continuity (2)
Provisional Application 62356422 · Jun 29, 2016
Related Publication 20180000754A1 · Jan 4, 2018