IP Library Granted Patent US 11,596,642
Granted Patent B2
US 11,596,642 · App. 16/303,945 · Granted Mar 7, 2023

Therapeutic treatment of breast cancer based on c-MAF status

Inventors: Walter Martin Gregory (West Yorkshire, GB); Juan Carlos Tercero (Madrid, ES); Roger Gomis (Barcelona, ES); Robert E. Coleman (Sheffield, GB)
Assignee: INBIOMOTION S.L.
A61K31/663A61K9/0019A61K9/0053A61K31/47A61P35/04C07K16/2878C12Q1/686C12Q1/6841C12Q1/6874C12Q1/6886C12Q2563/107C12Q2600/106C12Q2600/118C12Q2600/158
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Quick Facts
Patent No.
US 11,596,642
App. No.
16/303,945
Granted
Mar 7, 2023
Kind
B2
Abstract

The present invention relates to the design of a customized therapy for a subject with breast cancer based on the c-MAF expression level and the menopausal status of the subject. In some embodiments, the customized therapy comprises an agent for avoiding or preventing bone degradation. In some embodiments, the agent for avoiding or preventing bone degradation is zoledronic acid.

Claims (25)

1. A method for the treatment of a subject having breast cancer which comprises:

i) quantifying the c-MAF gene copy number, amplification, or gain in a tumor sample of said subject and

ii) comparing the copy number, amplification, or gain obtained in i) with a reference value, wherein the reference value is less than 2.5 copies of the c-MAF gene as measured using FISH,

wherein said subject has not increased copy number, amplification, or gain with respect to said reference value, and administering to said subject a therapy selected from the group consisting of: clodronate, ibandronate, and zoledronic acid.

2. The method of claim 1 , wherein the subject is non-postmenopausal or postmenopausal.

3. The method of claim 1 , wherein the subject is further administered a therapy aiming to prevent and/or treat bone remodeling, improve disease free survival or overall survival.

4. The method according to claim 1 , wherein the therapy is clodronate.

5. The method according to claim 1 , wherein the therapy is zoledronic acid.

6. The method of claim 1 , wherein the breast cancer is selected from the group consisting of: ER+ breast cancer, ER− breast cancer, triple negative breast cancer, of the basal-like subtype, and HER2+ breast cancer.

7. A method for the treatment of bone metastasis in a subject having breast cancer comprising determining that said subject has non increased c-MAF amplification, copy number or gain in a tumor sample with respect to a control sample and administering to said subject an agent capable of preventing or inhibiting bone remodeling or improving disease free survival or overall survival, wherein the agent capable of preventing or inhibiting bone remodeling or improving disease free survival or overall survival is selected from the group consisting of: clodronate, ibandronate, and zoledronic acid, and wherein the control sample has less than 2.5 copies of the c-MAF gene as measured using FISH.

8. The method of claim 7 , wherein the subject is postmenopausal.

9. The method according to claim 7 , wherein the agent is clodronate.

10. The method according to claim 7 , wherein the agent is zoledronic acid.

11. The method of claim 7 , wherein the breast cancer is selected from the group consisting of: ER+ breast cancer, ER− breast cancer, triple negative breast cancer, of the basal-like subtype, and HER2+ breast cancer.

12. A method for the treatment of a subject having breast cancer comprising determining that said subject has non increased c-MAF amplification, copy number, or gain in a tumor sample with respect to a control sample, and administering to said subject an agent selected from the group consisting of: clodronate, ibandronate, and zoledronic acid, and wherein the control sample has less than 2.5 copies of the c-MAF gene as measured using FISH.

13. The method of claim 12 , wherein the subject is non-postmenopausal, premenopausal or postmenopausal.

14. The method of claim 12 , wherein the breast cancer is selected from the group consisting of: ER+ breast cancer, ER− breast cancer, triple negative breast cancer, of the basal-like subtype, and HER2+ breast cancer.

15. The method according to claim 12 , wherein the agent is clodronate.

16. The method according to claim 12 , wherein the agent is zoledronic acid.

17. A method for the identification of a subject having breast cancer who will benefit from treatment with an agent selected from the group consisting of clodronate, ibandronate, and zoledronic acid comprising:

i) quantifying the c-MAF gene copy number, amplification, or gain in a tumor sample of said subject and

ii) comparing the copy number, amplification, or gain obtained in i) with a reference value, wherein the reference value is less than 2.5 copies of the c-MAF gene as measured using FISH,

wherein said subject has not increased copy number, amplification, or gain with respect to said reference value, and administering to said subject a therapy selected from the group consisting of clodronate, ibandronate, and zoledronic acid.

18. The method of claim 17 , wherein the breast cancer is selected from the group consisting of: ER+ breast cancer, ER− breast cancer, triple negative breast cancer, of the basal-like subtype, and HER2+ breast cancer.

19. The method according to claim 17 , wherein the agent is zoledronic acid.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 29, 2019
From: GREGORY, WALTER MARTIN; TERCERO, JUAN CARLOS; GOMIS, ROGER; COLEMAN, ROBERT E.
To: INBIOMOTION S.L.
Reel/Frame 050207/0915 →
Continuity (3)
Provisional Application 62344836 · Jun 2, 2016
Provisional Application 62341333 · May 25, 2016
Related Publication 20190269707A1 · Sep 5, 2019
Cited By (3)
US 12,196,758 US 12,233,077 US 12,312,642