IP Library › Granted Patent US 11,679,095
Granted Patent B2
US 11,679,095 · App. 17/323,514 · Granted Jun 20, 2023

Macrophages/microglia in neuro-inflammation associated with neurodegenerative diseases

Inventors: David R. Elmaleh (Newton, MA); Rudolph E. Tanzi (Milton, MA); Timothy M. Shoup (Franklin, MA); Ana Griciuc (Arlington, MA)
Assignee: The General Hospital Corporation
A61K31/352A61K9/0019A61K9/0073A61P25/28C07D311/22C07D311/24A61K45/06
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 11,679,095
App. No.
17/323,514
Granted
Jun 20, 2023
Kind
B2
Abstract

Described herein are methods of treating neuron inflammation conditions, for example, Alzheimer's disease, Parkinson's disease, Huntington's disease, ischemic stroke, and prion disease, comprising administering a therapeutically effective amount of cromolyn or a cromolyn derivative compound.

Claims (18)

1. A method of treating a neuron inflammation condition in a patient in need thereof comprising administering to the patient a therapeutically effective amount of the compound having the following formula:

wherein the neuron inflammation condition is amyotrophic lateral sclerosis (ALS), Huntington's Disease, Parkinson's disease (PD), ischemic stroke, or a condition associated with prion disease.

2. The method of claim 1 , wherein the neuron inflammation condition is ALS.

3. The method of claim 1 , wherein the neuron inflammation is Huntington's Disease.

4. The method of claim 1 , wherein the neuron inflammation is Parkinson's disease.

5. The method of claim 1 , wherein the neuron inflammation condition is ischemic stroke.

6. The method of claim 1 , wherein the neuron inflammation condition is associated with prion disease.

7. The method of claim 2 , wherein the compound is administered intraperitoneally and/or intravenously.

8. The method of claim 1 , wherein the compound is administered transdermally.

9. The method of claim 1 , wherein the compound is administered by inhalation.

10. The method of claim 1 , wherein the compound is administered at a dose between about 1 mg and about 1000 mg per day.

11. The method of claim 1 , where in the compound is administered at a dose of about 10, about 20, about 30, about 50, about 100, or about 500 mg per day.

12. The method of claim 2 , further comprising co-administering a second compound selected from CD4+; siRNA; miRNA that ameliorates ALS; glial morphology modifier; SOD1 control; and Riluzole.

13. The method of claim 2 , further comprising co-administering a second compound selected from an antibody targeting drug that ameliorates ALS and an anti-inflammatory targeting drug that ameliorates ALS.

14. The method of claim 1 , further comprising co-administering a second compound selected from a targeting drug that ameliorates neurodegeneration associated with amyloidosis or tauopathies.

15. The method of claim 4 , further comprising co-administering a second compound selected from an alpha synuclein targeting drug that ameliorates PD and a Parkinson's targeting drug that ameliorates PD.

16. The method of claim 1 , wherein the compound is administered at a dose between about 1 mg and about 70 mg per day.

17. The method of claim 1 , wherein the compound is administered orally.

Assignments (2)
CORRECTIVE ASSIGNMENT TO CORRECT THE INVENTOR NAME LISTED ON THE COVERSHEET FROM DAVID ELMALCH TO DAVID ELMALEH, AND INVENTOR NAME LISTED ON THE ASSIGNMENT FROM ANA GRICLUC TO ANA GRICIUC. PREVIOUSLY RECORDED ON REEL 62943 FRAME 197. ASSIGNOR(S) HEREBY CONFIRMS THE ASSIGNMENT OF ASSIGNOR'S INTEREST. Recorded Jan 20, 2026
From: ELMALEH, DAVID R.; TANZI, RUDOLPH E.; SHOUP, TIMOTHY M.; GRICIUC, ANA
To: THE GENERAL HOSPITAL CORPORATION
Reel/Frame 074903/0004 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 22, 2023
From: ELMALCH, DAVID R.; TANZI, RUDOLPH E.; SHOUP, TIMOTHY M.; GRICLUC, ANA
To: THE GENERAL HOSPITAL CORPORATION
Reel/Frame 062943/0197 →
Continuity (3)
Continuation 16328956
Provisional Application 62382192 · Aug 31, 2016
Related Publication 20220079914A1 · Mar 17, 2022
Cited By (4)
US 12,383,528 US 12,458,622 US 12,605,471 US 12,612,391