IP Library › Granted Patent US 11,787,766
Granted Patent B2
US 11,787,766 · App. 16/639,949 · Granted Oct 17, 2023

Compound having PD-L1 inhibitory activity, preparation method therefor and use thereof

Inventors: Lei Jiang (Shanghai, CN); Jianwen Deng (Shanghai, CN); Xiaoli Lu (Shanghai, CN); Ke Shang (Shanghai, CN); Jianyong Shou (Shanghai, CN); Bing Wang (Shanghai, CN); Danyi Wu (Shanghai, CN); Xueli Xu (Shanghai, CN); Yuan Xu (Shanghai, CN); Yi Zhang (Shanghai, CN); Mingwei Zheng (Shanghai, CN)
Assignee: SHANGHAI ENNOVABIO PHARMACEUTICALS CO., LTD.
C07D213/69A61K31/137A61K31/165A61K31/4155A61K31/437A61K31/44A61K31/444A61K31/4545A61K39/12A61K39/245A61K39/29A61K45/06C07C211/03C07C223/02C07D213/73C07D213/84C07D231/40C07D401/14C07D405/14C07D409/14C07D519/00
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Quick Facts
Patent No.
US 11,787,766
App. No.
16/639,949
Granted
Oct 17, 2023
Kind
B2
Abstract

Provided are a compound for the prevention and treatment of diseases associated with PD-L1, a preparation method therefor and use thereof. Specifically, provided are the compound of formula I, the stereoisomer and the racemate thereof, or pharmaceutically acceptable salts thereof, and also provided is an application thereof in the preparation of a drug for the prevention and treatment of diseases associated with PD-L1.

Claims (150)

1. A compound selected from the following group, or a stereoisomer, a racemate, or a pharmaceutically acceptable salt thereof,

No.

Structure of compound

6

9

17

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2. A compound selected from the following group, or a stereoisomer, a racemate, or a pharmaceutically acceptable salt thereof,

No.

Structure of compound

6

9

20

22

24

26

27

28

30

33

35

37

39

41

42

43

46

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82

3. A compound selected from the following group, or a stereoisomer, a racemate, or a pharmaceutically acceptable salt thereof,

No.

Structure of compound

9

26

27

30

35

36

37

42

43

45

46

47

49

50

51

56

58

60

62

63

65

66

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81

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 25, 2020
From: JIANG, LEI; DENG, JIANWEN; LU, XIAOLI; SHANG, KE; SHOU, JIANYONG; WANG, BING; WU, DANYI; XU, XUELI; XU, YUAN; ZHANG, YI; ZHENG, MINGWEI
To: SHANGHAI ENNOVABIO PHARMACEUTICALS CO., LTD.
Reel/Frame 054467/0590 →
Priority Claims (1)
CN 201710712191.8 · Aug 18, 2017 · national
Continuity (1)
Related Publication 20200392083A1 · Dec 17, 2020