IP Library Granted Patent US 11,807,867
Granted Patent B2
US 11,807,867 · App. 17/816,305 · Granted Nov 7, 2023

Compositions and methods for treating non-age-associated hearing impairment in a human subject

Inventors: Emmanuel John Simons (Boston, MA); Robert Ng (Boston, MA)
Assignee: Akouos, Inc.
C12N15/86A61P27/16C07K14/47A61K48/00C12N2750/14143C12N2750/14144
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Quick Facts
Patent No.
US 11,807,867
App. No.
17/816,305
Granted
Nov 7, 2023
Kind
B2
Abstract

Provided herein are compositions that include at least two different nucleic acid vectors, where each of the at least two different vectors includes a coding sequence that encodes a different portion of an otoferlin protein, and the use of these compositions to treat hearing loss in a subject.

Claims (36)

1. A plurality of recombinant adeno-associated viral (rAAV) vectors comprising:

a) a first rAAV vector comprising a nucleic acid sequence of SEQ ID NO: 96; and

b) a second rAAV vector comprising a nucleic acid sequence of SEQ ID NO: 105.

2. The plurality of rAAV vectors of claim 1 , wherein the first and second rAAV vectors are each encapsulated by an AAV capsid.

3. The plurality of rAAV vectors of claim 2 , wherein the AAV capsid encapsulating the first rAAV vector is a serotype selected from any one of AAV1, AAV2, AAV3, AAV4, AAV5, AAV6, AAV7, AAV8, AAV9, AAVrh8, AAVrh10, AAVrh39, AAVrh43, or Anc80.

4. The plurality of rAAV vectors of claim 2 , wherein the AAV capsid encapsulating the second rAAV vector is a serotype selected from any one of AAV1, AAV2, AAV3, AAV4, AAV5, AAV6, AAV7, AAV8, AAV9, AAVrh8, AAVrh10, AAVrh39, AAVrh43, or Anc80.

5. The plurality of rAAV vectors of claim 2 , wherein the first rAAV vector is encapsulated by an Anc80 capsid and the second rAAV vector is encapsulated by an Anc80 capsid.

6. The plurality of rAAV vectors of claim 5 , wherein the Anc80 capsids comprise the polypeptide sequence of SEQ ID NO: 109.

7. A composition comprising the plurality of rAAV vectors of claim 1 , wherein the composition further comprises one or more pharmaceutically acceptable carriers, diluents, or excipients.

8. The composition of claim 7 , wherein the composition is formulated for intra-cochlear administration.

9. The composition of claim 8 , wherein the composition is formulated to comprise a synthetic perilymph solution.

10. A method of expressing a recombinant full-length otoferlin protein in a mammalian cell, the method comprising administering a plurality of recombinant adeno-associated viral (rAAV) vectors comprising:

a) a first rAAV vector comprising a nucleic acid sequence of SEQ ID NO: 96; and

b) a second rAAV vector comprising a nucleic acid sequence of SEQ ID NO: 105;

to the mammalian cell, wherein the mammalian cell has reduced expression, lack of expression or dysfunction of otoferlin.

11. The method of claim 10 , wherein the mammalian cell is an inner hair cell.

12. The method of claim 10 , wherein the mammalian cell is a human cell.

13. The method of claim 10 , wherein the mammalian cell comprises a defective otoferlin gene.

14. The method of claim 10 , wherein the first and second rAAV vectors are each encapsulated by an AAV capsid.

15. The method of claim 14 , wherein the AAV capsid encapsulating the first rAAV vector is a serotype selected from any one of AAV1, AAV2, AAV3, AAV4, AAV5, AAV6, AAV7, AAV8, AAV9, AAVrh8, AAVrh10, AAVrh39, AAVrh43, or Anc80.

16. The method of claim 14 , wherein the AAV capsid encapsulating the second rAAV vector is a serotype selected from any one of AAV1, AAV2, AAV3, AAV4, AAV5, AAV6, AAV7, AAV8, AAV9, AAVrh8, AAVrh10, AAVrh39, AAVrh43, or Anc80.

17. The method of claim 14 , wherein the first rAAV vector is encapsulated by an Anc80 capsid and the second rAAV vector is encapsulated by an Anc80 capsid.

18. The method of claim 16 , wherein the Anc80 capsids comprise the polypeptide sequence of SEQ ID NO: 109.

19. A method of treating hearing loss in a subject having otoferlin related hearing loss, the method comprising administering a plurality of recombinant adeno-associated viral (rAAV) vectors comprising:

a) a first rAAV vector comprising a nucleic acid sequence of SEQ ID NO: 96; and

b) a second rAAV vector comprising a nucleic acid sequence of SEQ ID NO: 105;

into the cochlea of the subject, wherein the subject has reduced expression, lack of expression, or dysfunction of otoferlin.

20. The method of claim 19 , wherein the subject is a human.

21. The method of claim 19 , wherein the first and second rAAV vectors are each encapsulated by an AAV capsid.

22. The method of claim 21 , wherein the AAV capsid encapsulating the first rAAV vector is a serotype AAV1, AAV2, AAV3, AAV4, AAV5, AAV6, AAV7, AAV8, AAV9, AAVrh8, AAVrh10, AAVrh39, AAVrh43, or Anc80.

23. The method of claim 21 , wherein the AAV capsid encapsulating the second rAAV vector is a serotype AAV1, AAV2, AAV3, AAV4, AAV5, AAV6, AAV7, AAV8, AAV9, AAVrh8, AAVrh10, AAVrh39, AAVrh43, or Anc80.

24. The method of claim 21 , wherein the first rAAV vector is encapsulated by an Anc80 capsid and the second rAAV vector is encapsulated by an Anc80 capsid.

25. The method of claim 24 , wherein the Anc80 capsids comprise the polypeptide sequence of SEQ ID NO: 109.

26. The method of claim 19 , wherein the plurality of rAAV vectors is administered as a single dose.

27. The method of claim 19 , wherein the plurality of rAAV vectors is administered as two or more doses.

28. The method of claim 19 , wherein the subject has a defective otoferlin gene.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 8, 2023
From: SIMONS, EMMANUEL JOHN; NG, ROBERT
To: AKOUOS, INC.
Reel/Frame 063893/0346 →
Continuity (3)
Continuation PCTUS2021018919 · Feb 19, 2021
Provisional Application 62979792 · Feb 21, 2020
Related Publication 20230108913A1 · Apr 6, 2023
Cited By (8)
US 12,188,041 US 12,264,317 US 12,305,191 US 12,359,221 US 12,377,169 US 12,410,442 US 12,589,168 US 12,673,116