Compositions and methods for type III polyketide production in oleaginous yeast species
View Patent ↗This invention relates to compositions and methods for the production of Type III polyketides using genetically modified oleaginous yeast strains, for example, Yarrowia lipolytica.
1. A genetically modified oleaginous yeast cell comprising a heterologous gene encoding a heterologous Type III polyketide synthase and a gene encoding Acetyl-CoA Carboxylase (AceCarb (ACC1); YALI0C11407g), wherein the oleaginous yeast cell is Yarrowia lipolytica , and wherein the oleaginous yeast cell further comprises the following modifications: the overexpression of Putative Pyruvate Decarboxylase 2 (PDC2; YALI0D06930), Acetyl-CoA Synthetase 1 (ACS1; YALI0F05962), Acetaldehyde Dehydrogenase 5 (ALD5; YALI0D07942), and peroxin 10 (PEX10; YALI0C01023).
2. The yeast cell of claim 1 , wherein the Type III polyketide synthase is selected from the group consisting of a CAA86219.2 gene from Gerbera hybrida , AY517486 gene from Rheum palmatum , JX840717-JX840724 gene from Pseudomonas fluorescens , BOLDU5 gene from Rubus idaeus , B1VLQ8 gene from Streptomyces griseus , SCO1206 from Streptomyces coelicolor , BAB12102.2 gene from Humulus lupulus , or a combination thereof.
3. The yeast cell of claim 1 , wherein the heterologous gene is incorporated into a gene expression cassette comprising a promoter and the heterologous gene, wherein the gene expression cassette is integrated into the genome of the yeast cell.
4. The yeast cell of claim 1 , wherein at least two copies of the heterologous gene are present in the genome of the yeast cell.
5. The yeast cell of claim 1 , wherein the heterologous gene is episomally expressed from a plasmid.
6. The yeast cell of claim 1 , wherein the yeast cell comprises an additional genetic modification.
7. The yeast cell of claim 6 , wherein the additional genetic modification increases the acetyl-CoA or malonyl-CoA levels or fluxes.
8. The yeast cell of claim 7 , wherein the additional genetic modification increases the rate of beta-oxidation to increase the acetyl-CoA or malonyl-CoA levels or fluxes.
9. The yeast cell of claim 8 , wherein the additional genetic modification comprises the elimination or the reduction of Yarrowia lipolytica gene phosphatidate phosphatase (PAH1; YALI0D27016); and/or wherein the additional genetic modification comprises the overexpression of one or more Yarrowia lipolytica genes selected from the group consisting of multifunctional β oxidation protein (oxidoreductase and hydro-lyase) (MFE1; YALI0E15378), primary oleate regulator (POR1; YALI0D12628), or a combination thereof.
10. The yeast cell of claim 6 , wherein the additional genetic modification comprises the elimination or the reduction of one or more Yarrowia lipolytica genes selected from the group consisting of Aspartyl Protease (PEP4; YALI0F27071p), Protease B Vacuolar (PRB1; YALI0B16500p), Protease B Vacuolar (PRB1H; YALI0A06435g), Glucose-starch Glucosyltransferase Isoform 1 (GSY1; YALI0F18502p), Glucose-6-phosphate Dehydrogenase (ZWF1; YALI0E22649p), Pyruvate Carboxylase 1 (PYC1; YALI0C24101p), Phosphoenolpyruvate Carboxykinase (PCK1; YALI0C16995p), Fructose-1,6-bisphosphatase (FBP1; YALI0A15972p), Mitochondrial Carrier (YIA6; YALI0E16478g), Mitochondrial Carrier Protein (RIM2; YALI0F05500g), Alcohol Dehydrogenase 1 (ADH1; YALI0D25630p), Alcohol Dehydrogenase 2 (ADH2; YALI0E17787p), Alcohol Dehydrogenase 3 (ADH3; YALI0A16379p), C1-tetrahydrofolate Synthase (MIS1; YALI0F30745p), C1-THFS Protein C1-Tetrahydrofolate Synthase Precursor Mitochondrial (MTHFD1L; YALI0E01056g), Phosphoglucomutase (PGM2; YALI0E02090p), Glycerol-3-phosphate Dehydrogenase (GPD1; YALI0B02948p), Fatty Acid Synthase Subunit Alpha (FAS2; YALI0B19382p), Fatty Acid Synthase Subunit Beta (FAS1; YALI0B15059p), phosphatidate phosphatase (PAH1; YALI0D27016), or a combination thereof; and/or wherein the additional genetic modification comprises the overexpression of one or more Yarrowia lipolytica genes selected from the group consisting of Pyruvate Decarboxylase (Pyrudecarb (PDC1); YALI0D10131p), Dihydrolipoamide Dehydrogenase (PDE3; YALI0D20768g), Dihydrolipoamide Acetyltransferase (PDE2; YALI0D23683g), Malate Dehydrogenase (MAE1; YALI0E18634p), Acetyl-CoA Synthetase (AceCoA; YALI0F05962g), Pyruvate Dehydrogenase E1 Component Subunit Alpha (PDC-E1; YALI0F20702p), ATP-Citrate Lyase Subunit 1 (ACL1; YALI0E34793p), ATP-Citrate Lyase Subunit 2 (ACL2; YALI0D24431p), AMP Deaminase (AMPD; YALI0E11495p), Acetyl-CoA hydrolase (ACH1; YALI0E30965g), Acetaldehyde Dehydrogenase 1 (ALD1; YALI0B01298), Acetaldehyde Dehydrogenase 2 (ALD2; YALI0C03025), Acetaldehyde Dehydrogenase 3 (ALD3; YALI0E00264), Acetaldehyde Dehydrogenase 4 (ALD4; YALI0F23793), Acetaldehyde Dehydrogenase 6 (ALD6; YALI0F04444), Pyruvate Dehydrogenase E1 Component Subunit Alpha (PDA1; YALI0F20702), Pyruvate Dehydrogenase E1 Component Subunit Beta (PDB1; YALI0E27005), multifunctional β oxidation protein (oxidoreductase and hydro-lyase) (MFE1; YALI0E15378), primary oleate regulator (POR1; YALI0D12628), or a combination thereof.
11. The yeast cell of claim 10 , wherein the additional genetic modification comprises the elimination or the reduction of one or more Yarrowia lipolytica genes selected from the group consisting of Aspartyl Protease (PEP4; YALI0F27071p), Protease B Vacuolar (PRB1; YALI0B16500p), Protease B Vacuolar (PRB1H; YALI0A06435g), Glucose-starch Glucosyltransferase Isoform 1 (GSY1; YALI0F18502p), Glucose-6-phosphate Dehydrogenase (ZWF1; YALI0E22649p), Pyruvate Carboxylase 1 (PYC1; YALI0C24101p), Phosphoenolpyruvate Carboxykinase (PCK1; YALI0C16995p), Fructose-1,6-bisphosphatase (FBP1; YALI0A15972p), Mitochondrial Carrier (YIA6; YALI0E16478g), Mitochondrial Carrier Protein (RIM2; YALI0F05500g), Alcohol Dehydrogenase 1 (ADH1; YALI0D25630p), Alcohol Dehydrogenase 2 (ADH2; YALI0E17787p), Alcohol Dehydrogenase 3 (ADH3; YALI0A16379p), C1-tetrahydrofolate Synthase (MIS1; YALI0F30745p), C1-THFS Protein C1-Tetrahydrofolate Synthase Precursor Mitochondrial (MTHFD1L; YALI0E01056g), Phosphoglucomutase (PGM2; YALI0E02090p), Glycerol-3-phosphate Dehydrogenase (GPD1; YALI0B02948p), Fatty Acid Synthase Subunit Alpha (FAS2; YALI0B19382p), Fatty Acid Synthase Subunit Beta (FAS1; YALI0B15059p), (PAH1; YALI0D27016), or a combination thereof.
12. The yeast cell of claim 10 , wherein the additional genetic modification comprises the overexpression of one or more Yarrowia lipolytica genes selected from the group consisting of Pyruvate Decarboxylase (Pyrudecarb (PDC1); YALI0D10131p), Dihydrolipoamide Dehydrogenase (PDE3; YALI0D20768g), Dihydrolipoamide Acetyltransferase (PDE2; YALI0D23683g), Malate Dehydrogenase (MAE1; YALI0E18634p), Acetyl-CoA Synthetase (AceCoA; YALI0F05962g), Pyruvate Dehydrogenase E1 Component Subunit Alpha (PDC-E1; YALI0F20702p), ATP-Citrate Lyase Subunit 1 (ACL1; YALI0E34793p), ATP-Citrate Lyase Subunit 2 (ACL2; YALI0D24431p), AMP Deaminase (AMPD; YALI0E11495p), Acetyl-CoA hydrolase (ACH1; YALI0E30965g), Acetaldehyde Dehydrogenase 1 (ALD1; YALI0B01298), Acetaldehyde Dehydrogenase 2 (ALD2; YALI0C03025), Acetaldehyde Dehydrogenase 3 (ALD3; YALI0E00264), Acetaldehyde Dehydrogenase 4 (ALD4; YALI0F23793), Acetaldehyde Dehydrogenase 6 (ALD6; YALI0F04444), Pyruvate Dehydrogenase E1 Component Subunit Alpha (PDA1; YALI0F20702), Pyruvate Dehydrogenase E1 Component Subunit Beta (PDB1; YALI0E27005), multifunctional β oxidation protein (oxidoreductase and hydro-lyase) (MFE1; YALI0E15378), primary oleate regulator (POR1; YALI0D12628), or a combination thereof.
13. The yeast cell of claim 1 , wherein the yeast cell is a PO1f strain.
14. The yeast cell of claim 1 , wherein the yeast cell has been preoptimized for lipid overproduction.
15. A method for the production of a Type III polyketide comprising: 1) culturing the oleaginous yeast cell of claim 1 in a growth medium; and 2) isolating said Type III polyketide.
16. A genetically modified oleaginous yeast cell comprising a heterologous gene encoding a heterologous Type III polyketide synthase and a gene encoding Acetyl-CoA Carboxylase (AceCarb (ACC1); YALI0C11407g), wherein the oleaginous yeast cell is Yarrowia lipolytica , and wherein the oleaginous yeast cell further comprises the following modification: the overexpression of peroxin 10 (PEX10; YALI0C01023).
17. The yeast cell of claim 16 , wherein the Type III polyketide synthase is selected from the group consisting of a CAA86219.2 gene from Gerbera hybrida , AY517486 gene from Rheum palmatum , JX840717-JX840724 gene from Pseudomonas fluorescens , B0LDU5 gene from Rubus idaeus , B1VLQ8 gene from Streptomyces griseus , SCO1206 from Streptomyces coelicolor , BAB12102.2 gene from Humulus lupulus , or a combination thereof.
18. The yeast cell of claim 16 , wherein the heterologous gene is incorporated into a gene expression cassette comprising a promoter and the heterologous gene, wherein the gene expression cassette is integrated into the genome of the yeast cell.
19. The yeast cell of claim 16 , wherein at least two copies of the heterologous gene are present in the genome of the yeast cell.
20. The yeast cell of claim 16 , wherein the heterologous gene is episomally expressed from a plasmid.
21. The yeast cell of claim 16 , wherein the yeast cell comprises an additional genetic modification.
22. The yeast cell of claim 21 , wherein the additional genetic modification increases the acetyl-CoA or malonyl-CoA levels or fluxes.
23. The yeast cell of claim 22 , wherein the additional genetic modification increases the rate of beta-oxidation to increase the acetyl-CoA or malonyl-CoA levels or fluxes.
24. The yeast cell of claim 16 , wherein the yeast cell is a PO1f strain.
25. The yeast cell of claim 16 , wherein the yeast cell has been preoptimized for lipid overproduction.
26. A method for the production of a Type III polyketide comprising: 1) culturing the yeast cell of claim 16 in a growth medium; and 2) isolating said Type III polyketide.