Granted Patent
B2
US 11,883,393 · App. 17/126,501 · Granted Jan 30, 2024
Compounds and methods for the targeted degradation of androgen receptor
Assignee:
Arvinas Operations, Inc.
A61K31/496A61K31/167A61K31/277A61K31/337A61K31/417A61K31/4523A61K31/4545A61K31/497A61K31/501A61K31/506A61K31/5377A61K31/5386A61K31/57A61K31/661A61K31/663A61K31/675A61K38/09A61K47/545C07D401/12C07D401/14C07D413/12C07D413/14C07D498/10
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Abstract
This disclosure pertains to compounds, the preparation thereof, and the use of these compounds in the treatment of prostate cancer, including metastatic and/or castrate-resistant prostate cancer, in subjects in need thereof.
Claims (4)
1. A compound that is:
2. A pharmaceutically acceptable salt of a compound that is:
3. A pharmaceutical composition comprising a compound and one or more pharmaceutically acceptable excipients, wherein the compound is:
4. A pharmaceutical composition comprising a pharmaceutically acceptable salt of a compound and one or more pharmaceutically acceptable excipients, wherein the compound is:
Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST
Recorded Feb 4, 2021
From: SNYDER, LAWRENCE B.; CREW, ANDREW P.; WANG, JING; DONG, HANQING
To: ARVINAS OPERATIONS, INC.
Reel/Frame 055140/0837 →
Continuity (4)
Provisional Application
63089497
· Oct 8, 2020
Provisional Application
63032473
· May 29, 2020
Provisional Application
62950815
· Dec 19, 2019
Cited By (3)