IP Library Granted Patent US 11,931,336
Granted Patent B2
US 11,931,336 · App. 17/324,490 · Granted Mar 19, 2024

Enhancing autophagy or increasing longevity by administration of urolithins

Inventors: Christopher L. Rinsch (Lausanne, CH); William Blanco-Bose (La Croix, CH); Bernard Schneider (Pully, CH); Laurent Mouchiroud (Morges, CH); Dongryeol Ryu (Renens, CH); Penelope Andreux (Eclepens, CH); Johan Auwerx (Buchillon, CH)
Assignee: Amazentis SA
A61K31/37A61K31/00A61K31/366A61K31/7048A61K45/06C07D311/80
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Quick Facts
Patent No.
US 11,931,336
App. No.
17/324,490
Granted
Mar 19, 2024
Kind
B2
Abstract

Disclosed are methods, compounds, and compositions useful for increasing autophagy and promoting longevity. The methods, compounds, and compositions relate to urolithins and urolithin precursors and use thereof. Certain urolithins are represented by Formula I, while certain urolithin precursors are represented by Formula IV. The urolithin may be urolithin A, urolithin B, urolithin C, or urolithin D. The urolithin precursor may be ellagic acid or an ellagitannin. The methods include in vivo, ex vivo, and in vitro uses of the compounds and compositions.

Claims (20)

1. A method of treating a disease or condition selected from the group consisting of sarcopenia, sarcopenia of aging, osteoarthritis, muscular atrophy, muscle disuse atrophy, skeletal muscular atrophy, cardiac deterioration, cardiac deterioration with aging, negative consequences linked to aging, improving activity during aging, reducing age-related cataracts, improving balance or coordination, and frailty, comprising administering to a subject in need thereof a therapeutically effective amount of a urolithin, or a pharmaceutically acceptable salt thereof.

2. The method of claim 1 , wherein the disease or condition is sarcopenia.

3. The method of claim 1 , wherein the disease or condition is sarcopenia of aging.

4. The method of claim 1 , wherein the disease or condition is osteoarthritis.

5. The method of claim 1 , wherein the disease or condition is muscular atrophy.

6. The method of claim 1 , wherein the disease or condition is muscle disuse atrophy.

7. The method of claim 1 , wherein the disease or condition is skeletal muscular atrophy.

8. The method of claim 1 , wherein the disease or condition is cardiac deterioration.

9. The method of claim 1 , wherein the disease or condition is cardiac deterioration of aging.

10. The method of claim 1 , wherein the disease or condition is negative consequences linked to aging.

11. The method of claim 1 , wherein the disease or condition is improving activity during aging.

12. The method of claim 1 , wherein the disease or condition is reducing age-related cataracts.

13. The method of claim 1 , wherein the disease or condition is improving balance or coordination.

14. The method of claim 1 , wherein the disease or condition is frailty.

15. The method of claim 1 , wherein the urolithin is administered orally.

16. The method of claim 1 , wherein the urolithin is selected from the group consisting of urolithin A, urolithin B, and any combination thereof.

17. The method of claim 1 , wherein the urolithin is urolithin A.

18. The method of claim 1 , wherein the urolithin is urolithin B.

19. The method of claim 1 , wherein the subject is a human.

20. The method of claim 1 , wherein the urolithin is administered orally; the urolithin is urolithin A; and the subject is a human.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 9, 2021
From: SCHNEIDER, BERNARD; AUWERX, JOHAN; MOUCHIROUD, LAURENT; RYU, DONGRYEOL; ANDREUX, PENELOPE
To: ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (EPFL)
Reel/Frame 056486/0612 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 9, 2021
From: RINSCH, CHRISTOPHER L.; BLANCO-BOSE, WILLIAM
To: AMAZENTIS SA
Reel/Frame 056528/0733 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 9, 2021
From: ECOLE POLYTECHNIQUE FEDERALE DE LAUSANNE (EPFL)
To: AMAZENTIS SA
Reel/Frame 056528/0736 →
Continuity (5)
Continuation 13929455 · Jun 27, 2013
Provisional Application 61791137 · Mar 15, 2013
Provisional Application 61712886 · Oct 12, 2012
Provisional Application 61665137 · Jun 27, 2012
Related Publication 20210353591A1 · Nov 18, 2021
Cited By (3)
US 12,544,358 US 12,576,064 US 12,576,065