IP Library Granted Patent US 12,083,099
Granted Patent B2
US 12,083,099 · App. 17/513,284 · Granted Sep 10, 2024

Methods of treating symptoms of coronavirus infection with viral protease inhibitors

Inventors: Kevin Brown (Philadelphia, PA); Kevin Brogle (Philadelphia, NJ)
Assignee: Accencio LLC
A61K31/407A61K9/0014A61K31/4709
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Quick Facts
Patent No.
US 12,083,099
App. No.
17/513,284
Granted
Sep 10, 2024
Kind
B2
Abstract

The present disclosure relates to a method of reducing or arresting viral load in a subject infected with a coronavirus, the method comprising the step of administering to the subject a therapeutically effective amount of a viral protease inhibitor. In some embodiments, the subject is a human. In one embodiment, the coronavirus is SARS-COV-19 and the viral protease inhibitor is E)-N-(4-(3-(tert-butyl)-5-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-2-methoxystyryl)phenyl)methanesulfonamide; (R)-3-((2S,3S)-2-hydroxy-3-(3-hydroxy-2-methylbenzamido)-4-phenylbutanoyl)-5,5-dimethyl-N-(2-methylbenzyl)thiazolidine-4-carboxamide; R)—N-allyl-3-((2S,3S)-2-hydroxy-3-(3-hydroxy-2-methylbenzamido)-4-phenylbutanoyl)-5,5-dimethylthiazolidine-4-carboxamide; (4-((N-(5-cyclopropyl-2-(4-fluorophenyl)-3-(methylcarbamoyl)benzofuran-6-yl)methylsulfonamido)methyl)-2-fluorophenyl)boronic acid or salts thereof.

Claims (3)

1. A method of treating or alleviating at least one symptom of a coronavirus infection in a subject infected with coronavirus, the method comprising the step of administering to the subject a therapeutically effective amount of the viral protease inhibitor.

2. The method according to claim 1 , wherein the symptom is selected from the group consisting of fever, cough, tiredness, sore throat, diarrhea, conjunctivitis, headache, loss of taste, loss of smell, rash, difficulty breathing, shortness of breath, chest pain, chest pressure, Acute Respiratory Distress Syndrome (ARDS) and organ failure.

3. The method according to claim 1 , wherein the coronavirus is SARS-COV-19.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 22, 2022
From: BROWN, KEVIN; BROGLE, KEVIN
To: ACCENCIO LLC
Reel/Frame 060281/0223 →
Continuity (2)
Provisional Application 63106529 · Oct 28, 2020
Related Publication 20230113114A1 · Apr 13, 2023