IP Library › Granted Patent US 12,083,168
Granted Patent B2
US 12,083,168 · App. 17/719,580 · Granted Sep 10, 2024

Treatment and detection of inherited neuropathies and associated disorders

Inventors: Stephan L. Zuchner (Miami, FL); Adriana Rebelo (Miami, FL); Andrea Cortese (London, GB); Rong Grace Zhai (Miami, FL); David N. Herrmann (Rochester, NY)
Assignees: University of Miami; University of Rochester; UCL Business LTD
A61K38/443A61K31/198A61K31/352A61K31/4184A61K31/4188A61K31/426A61K31/428A61K31/473A61K31/499A61K31/502A61K31/517A61K31/7105A61K38/465A61K48/005A61P25/28C12N9/0006C12N15/1137C12N15/86C12Q1/6883C12Y101/01014G01N33/66C12N2310/11C12N2750/14143C12Q2600/156
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Quick Facts
Patent No.
US 12,083,168
App. No.
17/719,580
Granted
Sep 10, 2024
Kind
B2
Abstract

The present disclosure relates to methods of detecting and treating inherited neuropathy.

Claims (14)

1. A method for treating inherited neuropathy associated with a mutation in the sorbitol dehydrogenase (SORD) gene in a mammalian subject, comprising administering to the subject an effective amount of an inhibitor of aldose reductase.

2. The method of claim 1 , wherein the inhibitor of aldose reductase is selected from the group consisting of Alrestatin, Epalrestat, Diepalrestat, Fidarestat, Imirestat, Lidorestat, Minalrestat, Ponalrestat, Ranirestat, Salfredin B11, Sorbinil, Tolrestat, Zenarestat, and Zopolrestat.

3. The method of claim 1 , wherein the inhibitor of aldose reductase is Epalrestat.

4. The method of claim 1 , wherein the inhibitor of aldose reductase is Zopolrestat.

5. The method of claim 1 , wherein the inhibitor of aldose reductase is Ranirestat.

6. The method of claim 1 , wherein the mutation in the sorbitol dehydrogenase (SORD) gene is selected from the group consisting of c.329G>C; p.Arg110Pro, c.298C>T; p.Arg100Ter, and c.458C>A; p. Ala 153 Asp, wherein the mutations are defined with reference to the nucleotide sequence of SEQ ID NO: 45 and the amino acid sequence of SEQ ID NO: 46.

7. The method of claim 1 , wherein the mutation in the sorbitol dehydrogenase (SORD) gene selected from the group consisting of c.28C>T; p.Leu10Phe, c.316_425+165del; p.Cys106Ter, c.895C>T; p.Arg299Ter, and c.964G>A; p. Val322Ile, wherein the mutations are defined with reference to the nucleotide sequence of SEQ ID NO: 45 and the amino acid sequence of SEQ ID NO: 46.

8. The method of claim 1 , wherein the effective amount of an aldose reductase inhibitor reduces the level of intracellular sorbitol in the subject.

9. The method of claim 1 , further comprising detecting the mutation in the sorbitol dehydrogenase gene of the subject.

10. The method of claim 1 , further comprising measuring the level of sorbitol in a subject, wherein a sorbitol level of greater than about 10 mg/L in blood indicates that the subject has neuropathy associated with the mutation in the sorbitol dehydrogenase (SORD) gene.

11. The method of claim 1 , wherein the subject has a deletion of individual or multiple coding exons that encode the amino acid of SEQ ID NO:46 or a deletion of the entire SORD gene that encodes the amino acid of SEQ ID NO:46.

12. The method of claim 1 , wherein the mutation in the SORD gene leads to hypomorphic function of SORD.

13. The method of claim 1 , wherein the mutation in the SORD gene leads to loss of function of SORD.

14. The method of claim 1 , wherein the mutation in the sorbitol dehydrogenase (SORD) gene is c.757delG; p.Ala253GlnfsTer27, wherein the mutation is defined with reference to the nucleotide sequence of SEQ ID NO: 45 and the amino acid sequence of SEQ ID NO: 46.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 16, 2023
From: ZUCHNER, STEPHAN L.; REBELO, ADRIANA; ZHAI, RONG GRACE
To: UNIVERSITY OF MIAMI
Reel/Frame 063970/0136 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 16, 2023
From: CORTESE, ANDREA
To: UCL BUSINESS LTD
Reel/Frame 063970/0177 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 16, 2023
From: HERRMANN, DAVID N.
To: UNIVERSITY OF ROCHESTER
Reel/Frame 064012/0596 →
Continuity (6)
Continuation 17517227 · Nov 2, 2021
Continuation PCTUS2020031708 · May 6, 2020
Provisional Application 62987151 · Mar 9, 2020
Provisional Application 62844370 · May 7, 2019
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