IP Library › Granted Patent US 12,208,092
Granted Patent B2
US 12,208,092 · App. 18/615,512 · Granted Jan 28, 2025

Compositions and methods for administering paltusotine to patients with hepatic impairment

Inventors: Lance Goulet (Poway, CA); William Humphreys (Lawrenceville, NJ); Ajay Madan (San Diego, CA); Sha Luo (San Diego, CA)
Assignee: CRINETICS PHARMACEUTICALS, INC.
A61K31/4709A61K9/0053A61K9/2013A61K9/2018A61K9/2027A61K9/2054A61K9/2813A61K9/2866
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Quick Facts
Patent No.
US 12,208,092
App. No.
18/615,512
Granted
Jan 28, 2025
Kind
B2
Abstract

Provided are compositions and methods for administering paltusotine, or a pharmaceutically acceptable salt thereof, to a patient having hepatic impairment.

Claims (30)

1. A method comprising administering a therapeutically effective amount of paltusotine, or a pharmaceutically acceptable salt thereof, to a patient, wherein the patient has hepatic impairment, and wherein the therapeutically effective amount of paltusotine, or a pharmaceutically acceptable salt thereof, is the same amount that would be administered to a patient who does not have hepatic impairment, wherein the paltusotine is administered to the patient to treat acromegaly, carcinoid syndrome and/or neuroendocrine tumor.

2. A method comprising:

(a) administering to a patient a therapeutically effective amount of paltusotine, or a pharmaceutically acceptable salt thereof;

(b) subsequently determining that the patient has hepatic impairment; and

(c) administering the same therapeutically effective amount of paltusotine, or a pharmaceutically acceptable salt thereof, to the patient without dose adjustment, wherein the paltusotine is administered to the patient to treat acromegaly, carcinoid syndrome and/or neuroendocrine tumor.

3. The method of claim 1 , wherein the patient has mild, moderate, or severe hepatic impairment.

4. The method of claim 3 , wherein the patient has mild hepatic impairment.

5. The method of claim 3 , wherein the patient has moderate hepatic impairment.

6. The method of claim 3 , wherein the patient has severe hepatic impairment.

7. The method of claim 1 , wherein the patient has a Child-Pugh Score of 5-6, 7-9, or 10-15.

8. The method of claim 7 , wherein the patient has a Child-Pugh Score of 4-5.

9. The method of claim 7 , wherein the patient has a Child-Pugh Score of 6-8.

10. The method of claim 7 , wherein the patient has a Child-Pugh Score of 10-15.

11. The method of claim 1 , wherein the patient has acromegaly.

12. The method of claim 11 , wherein the paltusotine, or a pharmaceutically acceptable salt thereof, is administered in an amount equivalent to about 40 mg of paltusotine free base.

13. The method of claim 11 , wherein the paltusotine, or a pharmaceutically acceptable salt thereof, is administered in an amount equivalent to about 60 mg of paltusotine free base.

14. The method of claim 2 , wherein the paltusotine, or a pharmaceutically acceptable salt thereof, is administered to the patient to treat acromegaly.

15. The method of claim 1 , wherein the patient has carcinoid syndrome and/or NETs.

16. The method of claim 15 , wherein the paltusotine, or a pharmaceutically acceptable salt thereof, is administered in an amount equivalent to about 40 mg of paltusotine free base.

17. The method of claim 15 , wherein the paltusotine, or a pharmaceutically acceptable salt thereof, is administered in an amount equivalent to about 80 mg of paltusotine free base.

18. The method of claim 15 , wherein the paltusotine, or a pharmaceutically acceptable salt thereof, is administered in an amount equivalent to about 120 mg of paltusotine free base.

19. The method of claim 2 , wherein the paltusotine, or a pharmaceutically acceptable salt thereof, is administered to the patient to treat carcinoid syndrome and/or NETs.

20. The method of claim 1 , wherein the paltusotine, or a pharmaceutically acceptable salt thereof, is administered daily.

21. The method of claim 1 , wherein the paltusotine, or a pharmaceutically acceptable salt thereof, is administered once daily.

22. The method of claim 1 , wherein the paltusotine, or a pharmaceutically acceptable salt thereof, is administered orally.

23. The method of claim 1 , wherein the paltusotine, or a pharmaceutically acceptable salt thereof, is administered in one or more oral dosage forms.

24. The method of claim 23 , wherein the oral dosage form is a tablet.

25. The method of claim 1 , wherein the paltusotine, or a pharmaceutically acceptable salt thereof, is a hydrochloride salt of paltusotine.

26. The method of claim 25 , wherein the hydrochloride salt of paltusotine is amorphous.

27. The method of claim 1 , wherein the patient with hepatic impairment has equivalent exposure of paltusotine free base as in a patient with normal hepatic function who is administered the same amount of paltusotine, or a pharmaceutically acceptable salt thereof.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 26, 2024
From: GOULET, LANCE; HUMPHREYS, WILLIAM; MADAN, AJAY; LUO, SHA
To: CRINETICS PHARMACEUTICALS, INC.
Reel/Frame 069052/0958 →
Continuity (2)
Provisional Application 63455193 · Mar 28, 2023
Related Publication 20240325376A1 · Oct 3, 2024
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