IP Library › Granted Patent US 12,215,103
Granted Patent B2
US 12,215,103 · App. 18/612,631 · Granted Feb 4, 2025

Fused imidazole derivative, preparation method therefor, and medical use thereof

Inventors: Fanglong Yang (Shanghai, CN); Ling Zhang (Shanghai, CN); Liangliang Zheng (Shanghai, CN); Feng He (Shanghai, CN); Weikang Tao (Shanghai, CN)
Assignee: Jiangsu Hengrui Pharmaceuticals Co., Ltd.
C07D417/14A61P1/16C07D405/14C07D471/04C07D495/04
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Quick Facts
Patent No.
US 12,215,103
App. No.
18/612,631
Granted
Feb 4, 2025
Kind
B2
Abstract

Disclosed are fused imidazole derivatives, preparation methods therefor and medical uses thereof. Specifically, the present disclosure relates to a fused imidazole derivative as shown in general formula (IM), a preparation method therefor, a pharmaceutical composition containing the derivative, and the use of same as a therapeutic agent, in particular the use thereof as a GLP-1 receptor agonist, and the use thereof in the preparation of drugs for the treatment and/or prevention of diabetes.

Claims (12)

1. A compound, wherein the compound is selected from the group consisting of:

or a tautomer, racemate, enantiomer or diastereomer thereof or a mixture thereof, or a pharmaceutically acceptable salt thereof.

2. The compound according to claim 1 , wherein the compound is:

or a tautomer, racemate, enantiomer or diastereomer thereof or a mixture thereof, or a pharmaceutically acceptable salt thereof.

3. The compound according to claim 1 , wherein the compound is:

or a tautomer, racemate, enantiomer or diastereomer thereof or a mixture thereof, or a pharmaceutically acceptable salt thereof.

4. A pharmaceutical composition, comprising the compound of claim 1 , or a tautomer, racemate, enantiomer or diastereomer thereof or a mixture thereof, or a pharmaceutically acceptable salt thereof, and one or more pharmaceutically acceptable carriers, diluents or excipients.

5. A pharmaceutical composition, comprising the compound of claim 3 , or a tautomer, racemate, enantiomer or diastereomer thereof or a mixture thereof, or a pharmaceutically acceptable salt thereof, and one or more pharmaceutically acceptable carriers, diluents or excipients.

6. A compound having the structure of:

or a tautomer, racemate, enantiomer or diastereomer thereof or a mixture thereof, or a pharmaceutically acceptable salt thereof.

7. A pharmaceutical composition, comprising the compound of claim 6 , or a tautomer, racemate, enantiomer or diastereomer thereof or a mixture thereof, or a pharmaceutically acceptable salt thereof, and one or more pharmaceutically acceptable carriers, diluents or excipients.

8. A pharmaceutical composition, comprising the compound of claim 2 , or a tautomer, racemate, enantiomer or diastereomer thereof or a mixture thereof, or a pharmaceutically acceptable salt thereof, and one or more pharmaceutically acceptable carriers, diluents or excipients.

Assignments (4)
CORRECTIVE ASSIGNMENT TO CORRECT THE THE NAME OF THE SECOND INVENTOR PREVIOUSLY RECORDED AT REEL: 69335 FRAME: 114. ASSIGNOR(S) HEREBY CONFIRMS THE ASSIGNMENT. Recorded Dec 16, 2024
From: YANG, FANGLONG; ZHANG, LING; ZHENG, LIANGLIANG; HE, FENG; TAO, WEIKANG
To: SHANGHAI HENGRUI PHARMACEUTICAL CO., LTD.
Reel/Frame 070746/0422 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 20, 2024
From: YANG, FANGLONG; CHANG, LING; ZHENG, LIANGLIANG; HE, FENG; TAO, WEIKANG
To: SHANGHAI HENGRUI PHARMACEUTICAL CO., LTD.
Reel/Frame 069335/0114 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 20, 2024
From: SHANGHAI HENGRUI PHARMACEUTICAL CO., INC.
To: JIANGSU HENGRUI PHARMACEUTICALS CO., LTD.
Reel/Frame 069335/0180 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 22, 2024
From: YANG, FANGLONG; ZHANG, LING; ZHENG, LIANGLIANG; HE, FENG; TAO, WEIKANG
To: JIANGSU HENGRUI PHARMACEUTICALS CO., LTD.; SHANGHAI HENGRUI PHARMACEUTICAL CO., LTD.
Reel/Frame 066864/0457 →
Priority Claims (6)
CN 202010905693.4 · Sep 1, 2020 · national
CN 202010984336.1 · Sep 18, 2020 · national
CN 202011124085.6 · Oct 20, 2020 · national
CN 202011253077.1 · Nov 11, 2020 · national
CN 202011407911.8 · Dec 4, 2020 · national
CN 202011627733.X · Dec 31, 2020 · national
Continuity (2)
Continuation 18043508
Related Publication 20240246958A1 · Jul 25, 2024
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