IP Library › Granted Patent US 12,233,127
Granted Patent B2
US 12,233,127 · App. 17/270,115 · Granted Feb 25, 2025

Human monoclonal antibodies to a new universal influenza A hemagglutinin head domain epitope

Inventor: James E. Crowe, Jr. (Nashville, TN)
Assignee: Vanderbilt University
A61K39/42A61P31/16C07K16/1018G01N33/56983A61K2039/505G01N2333/11
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Quick Facts
Patent No.
US 12,233,127
App. No.
17/270,115
Granted
Feb 25, 2025
Kind
B2
Abstract

The present disclosure is directed to antibodies binding previously undefined epitopes on influenza A virus hemagglutinin and methods for use thereof.

Claims (16)

1. A method of treating a subject infected with influenza A virus or reducing the likelihood of infection of a subject at risk of contracting influenza A virus, comprising administering to said subject an antibody or antibody fragment having heavy chain CDR1-3 sequences and light chain CDR1-3 sequences of SEQ ID NOS: 17-19 and SEQ ID NOS: 29-31, respectively, or administering an RNA or DNA sequence or vector encoding the antibody or antibody fragment.

2. The method of claim 1 , the antibody or antibody fragment is encoded by light and heavy chain variable sequences of SEQ ID NOS: 2 and 1, respectively.

3. The method of claim 1 , the antibody or antibody fragment is encoded by light and heavy chain variable sequences having 95% identity to SEQ ID NOS: 2 and 1, respectively.

4. The method of claim 1 , wherein said antibody or antibody fragment is encoded by light and heavy chain variable sequences having 70%, 80%, or 90% identity to SEQ ID NOS: 2 and 1, respectively.

5. The method of claim 1 , wherein said antibody or antibody fragment comprises light and heavy chain variable sequences according to sequences of SEQ ID NOS: 10 and 9, respectively.

6. The method of claim 1 , wherein said antibody or antibody fragment comprises light and heavy chain variable sequences having 70%, 80% or 90% identity to SEQ ID NOS: 10 and 9, respectively.

7. The method of claim 1 , wherein said antibody or antibody fragment comprises light and heavy chain variable sequences having 95% identity to SEQ ID NOS: 10 and 9, respectively.

8. The method of claim 1 , wherein the antibody fragment is a recombinant scFv (single chain fragment variable) antibody, Fab fragment, F(ab′) 2 fragment, or Fv fragment.

9. The method of claim 1 , wherein said antibody is an IgG, or a recombinant IgG antibody or antibody fragment that comprises an Fc portion mutated to eliminate or enhance FcR interactions, to increase half-life and/or increase therapeutic efficacy, or comprises a glycan modification to eliminate or enhance FcR interactions.

10. The method of claim 1 , wherein said antibody is a chimeric antibody or a bispecific antibody.

11. The method of claim 1 , wherein said antibody or antibody fragment is administered prior to infection or after infection.

12. The method of claim 1 , wherein said subject is a pregnant female, a sexually active female, or a female undergoing fertility treatments.

13. The method of claim 1 , wherein delivering comprises antibody or antibody fragment administration, or genetic delivery with an RNA or DNA sequence or vector encoding the antibody or antibody fragment.

14. The method of claim 1 , wherein said antibody or antibody fragment has an antiviral molecule attached thereto.

15. The method of claim 9 , wherein the mutation to eliminate or enhance FcR interactions, to increase half-life and/or increase therapeutic efficacy is a LALA, N297, GASD/ALIE, YTE or LS mutation.

16. The method of claim 9 , wherein said glycan modification is a result of enzymatic or chemical addition or removal of glycans, or expression in a cell line engineered with a defined glycosylating pattern.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 22, 2024
From: CROWE, JAMES E., JR.
To: VANDERBILT UNIVERSITY
Reel/Frame 069211/0792 →
Continuity (3)
Provisional Application 62848301 · May 15, 2019
Provisional Application 62721675 · Aug 23, 2018
Related Publication 20210252150A1 · Aug 19, 2021
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