IP Library Granted Patent US 12,258,308
Granted Patent B2
US 12,258,308 · App. 17/544,616 · Granted Mar 25, 2025

Benzene derivative

Inventors: Shoji Nojima (Osaka, JP); Kenji Sasaki (Osaka, JP); Tohru Kambe (Osaka, JP); Takashi Konemura (Osaka, JP); Yoshikazu Goto (Osaka, JP)
Assignee: Ono Pharmaceutical Co., Ltd.
C07C311/21
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Quick Facts
Patent No.
US 12,258,308
App. No.
17/544,616
Granted
Mar 25, 2025
Kind
B2
Abstract

A compound represented by general formula (I) (in the formula, all symbols are as described in the description) or a salt thereof has a potent nerve-protecting and/or -repairing activity, and therefore can be used as a therapeutic agent for neuropathy (e.g., chronic inflammatory demyelinating polyneuropathy, Guillain-Barre syndrome, periarteritis nodosa, allergic vasculitis, diabetic peripheral neuropathy, entrapment neuropathy, peripheral neuropathy associated with the administration of a chemotherapeutic drug, or peripheral neuropathy associated with Charcot-Marie-Tooth disease).

Claims (12)

1. A method of promoting differentiation of a Schwann cell, comprising contacting a cell with 3-[2-[(E)-5-[3-(benzenesulfonamido)phenyl]pent-4-enoxy]phenyl]propanoic acid or a salt thereof.

2. The method according to claim 1 , wherein the cell is contacted with 3-[2-[(E)-5-[3-(benzenesulfonamido)phenyl]pent-4-enoxy]phenyl]propanoic acid.

3. The method according to claim 1 , wherein the cell is contact with a salt of 3-[2-[(E)-5-[3-(benzenesulfonamido)phenyl]pent-4-enoxy]phenyl]propanoic acid.

4. A method for preventing or treating neuropathy, comprising administering an effective amount of 3-[2-[(E)-5-[3-(benzenesulfonamido)phenyl]pent-4-enoxy]phenyl]propanoic acid or a salt thereof to a mammal.

5. The method according to claim 4 , wherein 3-[2-[(E)-5-[3-(benzenesulfonamido)phenyl]pent-4-enoxy]phenyl]propanoic acid is administered.

6. The method according to claim 4 , wherein a salt of 3-[2-[(E)-5-[3-(benzenesulfonamido)phenyl]pent-4-enoxy]phenyl]propanoic acid is administered.

7. The method according to claim 4 , wherein the neuropathy is a peripheral neuropathy.

8. The method according to claim 7 , wherein the peripheral neuropathy is chronic inflammatory demyelinating polyneuropathy, Guillain-Barre syndrome, periarteritis nodosa, allergic vasculitis, diabetic peripheral neuropathy, entrapment neuropathy, peripheral neuropathy associated with Charcot-Marie-Tooth disease, peripheral neuropathy associated with an infectious disease, a drug-induced peripheral neuropathy associated with the administration of an anti-convulsant agent, an anti-microbial agent, a chemotherapeutic drug or a sedative agent, multifocal motor neuropathy or a toxic peripheral neuropathy associated with the ingestion of a heavy metal, an organic solvent, a toxic substance or an alcohol.

9. The method according to claim 4 , wherein the mammal is a human.

10. The method according to claim 8 , wherein the drug-induced peripheral neuropathy is peripheral neuropathy associated with the administration of a chemotherapeutic drug.

11. The method according to claim 4 , wherein the neuropathy is central neuropathy.

12. The method according to claim 11 , wherein the central neuropathy is amyotrophic lateral sclerosis.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 14, 2021
From: NOJIMA, SHOJI; SASAKI, KENJI; KAMBE, TOHRU; KONEMURA, TAKASHI; GOTO, YOSHIKAZU
To: ONO PHARMACEUTICAL CO., LTD.
Reel/Frame 058390/0093 →
Priority Claims (1)
JP 2018-143024 · Jul 31, 2018 · national
Continuity (2)
Continuation 17264603
Related Publication 20220089532A1 · Mar 24, 2022
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