IP Library Granted Patent US 12,486,249
Granted Patent B2
US 12,486,249 · App. 18/366,218 · Granted Dec 2, 2025

SSTR4 agonist salts

Inventors: David Andrew Coates (New Palestine, IN); David Michael Remick (Fishers, IN)
Assignee: Eli Lilly & Company
C07D401/12C07B2200/13
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Quick Facts
Patent No.
US 12,486,249
App. No.
18/366,218
Granted
Dec 2, 2025
Kind
B2
Abstract

The present invention relates to specific salts of (1S,5R)-(1α,5α,6α)-N-[1,1-dimethyl-2-[(3-methyl-2-pyridyl)oxy]ethyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide, to pharmaceutical compositions comprising said salts, to methods of using said salts to treat physiological disorders, and to intermediates useful in the synthesis of the salts.

Claims (12)

1 . A crystalline compound of the formula:

or a hydrate thereof.

2 . The compound of claim 1 , wherein the compound is a hydrate.

3 . The compound of claim 1 , wherein the compound is a hydrate, wherein the water content at ambient temperature is in the range of 3% to 9% by weight.

4 . The compound of claim 1 , wherein the compound is:

5 . The compound of claim 1 , wherein the compound is:

6 . A pharmaceutical composition comprising the compound of claim 1 and one or more pharmaceutically acceptable carriers, diluents, or excipients.

7 . A method of treating pain in a patient comprising administering to said patient in need of such treatment an effective amount of the compound of claim 1 .

8 . A method of treating chronic back pain in a patient comprising administering to said patient in need of such treatment an effective amount of the compound of claim 1 .

9 . A method of treating neuropathic pain in a patient comprising administering to said patient in need of such treatment an effective amount of the compound of claim 1 .

10 . The method of claim 9 , wherein the neuropathic pain is diabetic peripheral neuropathic pain.

11 . A method of treating pain associated with osteoarthritis in a patient comprising administering to said patient in need of such treatment an effective amount of the compound of claim 1 .

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 7, 2023
From: COATES, DAVID ANDREW; REMICK, DAVID MICHAEL
To: ELI LILLY AND COMPANY
Reel/Frame 064510/0071 →
Continuity (3)
Continuation 17944429 · Sep 14, 2022
Provisional Application 63243785 · Sep 14, 2021
Related Publication 20240067628A1 · Feb 29, 2024
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