IP Library Granted Patent US 12,497,600
Granted Patent B2
US 12,497,600 · App. 17/767,764 · Granted Dec 16, 2025

Biosynthesis of cannabinoids from cannabigerolic acid using novel cannabinoid synthases

Inventors: Maybelle Darlene Kho Go (Singapore, SG); Wen Shan Yew (Singapore, SG)
Assignee: National University of Singapore
C12N9/0004C12N15/815C12P17/04C12P17/06C12P17/162C12R2001/84C12R2001/865C12Y121/03007
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Quick Facts
Patent No.
US 12,497,600
App. No.
17/767,764
Granted
Dec 16, 2025
Kind
B2
Abstract

A method for producing a cannabinoid by contacting cannabigerolic acid with a cannabinoid synthase orthologue. The cannabinoid synthase orthologue is from an organism other than Cannabis sativa . Also disclosed is a recombinant cell of Saccharomyces cerevisiae or Pichia pastoris that includes in its genome a nucleic acid encoding the above cannabinoid synthase orthologue. The cannabinoid synthase orthologue is expressed in the recombinant cell in an active form.

Claims (3)

1 . A method for producing one or more cannabinoids, the method comprising contacting cannabigerolic acid (CBGA) with a cannabinoid synthase orthologue, wherein the orthologue includes an amino acid sequence selected from the group consisting of SEQ ID NOs: 16, 23, 47, 57, 87, 107 and 117 and wherein the cannabinoids produced have a molecular weight of 358.5 g/mol, 374.5 g/mol, or 330.5 g/mol.

2 . The method of claim 1 , wherein the cannabinoids produced include cannabielsoic acid and cannabielsoin.

3 . The method of claim 1 , wherein the cannabinoid synthase orthologue is a recombinant enzyme produced in Saccharomyces cerevisiae, Yarrowia lipolytica, Kluyveromyces marxianus , or Pichia pastoris.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 23, 2023
From: GO, MAYBELLE DARLENE KHO; YEW, WEN SHAN
To: NATIONAL UNIVERSITY OF SINGAPORE
Reel/Frame 062452/0899 →
Continuity (2)
Provisional Application 62913991 · Oct 11, 2019
Related Publication 20240084270A1 · Mar 14, 2024
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