IP Library › Granted Patent US 12,516,384
Granted Patent B2
US 12,516,384 · App. 17/760,869 · Granted Jan 6, 2026

Methods and kit for analyzing responsiveness of patients to CD19 immunotherapy

Inventors: Charles G. Mullighan (Memphis, TN); Kathryn G. Roberts (Memphis, TN); Chunxu Qu (Memphis, TN); Yaqi Zhao (Memphis, TN)
Assignee: St. Jude Children's Research Hospital, Inc.
C12Q1/6886A61K35/28A61K38/1709A61P35/02C07K16/2803C07K2317/31C12Q1/6869C12Q2600/106C12Q2600/158
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Quick Facts
Patent No.
US 12,516,384
App. No.
17/760,869
Filed
Mar 16, 2022
Granted
Jan 6, 2026
Kind
B2
Art Unit
1642
USPC
424/136.1
Abstract

Kits and methods for determining resistance of a B-cell malignancy to blinatumomab immunotherapy and selecting a treatment for a subject with a B-cell malignancy based upon the expression level of an exon 2 intra-exonic splice variant of CD19 are provided.

Claims (14)

1 . A kit comprising a thermostable polymerase and a pair of primer oligonucleotides for amplifying a nucleic acid of SEQ ID NO:3, and optionally a probe that hybridizes to the exon 2 splice junction of SEQ ID NO:3, wherein the pair of primer oligonucleotides comprise:

(a) SEQ ID NO:4 and SEQ ID NO:5;

(b) SEQ ID NO:6 and SEQ ID NO:7;

(c) SEQ ID NO:8 and SEQ ID NO:9; or

(d) SEQ ID NO:10 and SEQ ID NO:11, and

the pair of primer oligonucleotides or probe comprises a reporter moiety.

2 . The kit of claim 1 , wherein the probe comprises SEQ ID NO:12.

3 . A method for selecting a treatment for a subject with a B-cell malignancy, comprising:

(a) measuring CD19 exon2del transcript expression levels in a sample of malignant B-cells from a subject using the kit of claim 1 ;

(b) comparing the levels of CD19 exon2del transcript expression obtained in step (a) with a reference level of CD19 exon2del transcript or wild-type CD19 transcript expression; and

(c) treating the subject with a CD19-independent treatment when the levels of CD19 exon2del transcript expression are elevated in the sample compared to the reference level.

4 . The method of claim 3 , wherein the reference level of CD19 exon2del transcript or wild-type CD19 transcript expression is obtained from a pool of subjects that have positively responded to treatment with a CD19 immunotherapeutic.

5 . The method of claim 3 , wherein the subject has acute lymphoblastic leukemia.

6 . The method of claim 3 , wherein the CD19-independent treatment comprises bone marrow transplantation or administration of an anti-CD22 immunotherapeutic, a BH3 mimetic or chemotherapeutic.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 17, 2022
From: MULLIGHAN, CHARLES G.; ROBERTS, KATHRYN G.; QU, CHUNXU; ZHAO, YAQI
To: ST. JUDE CHILDREN'S RESEARCH HOSPITAL, INC.
Reel/Frame 059294/0687 →
Continuity (2)
Provisional Application 62901951 · Sep 18, 2019
Related Publication 20220356531A1 · Nov 10, 2022
References Cited (11)
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Fischer, J. et al. (2017) “CD19 Isoforms Enabling Resistance to CART-19 Immunotherapy Are Expressed in B-ALL Patients at Initial Diagnosis,” Journal of Immunotherapy 40(5):187-195. [cited by applicant]
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Jazirehi, A.R., et al. (2017) “Clinical Implications of Anti-CD19 Chimeric Antigen Receptors (CAR) T Cell Therapy in Acute Lymphoblastic Leukemia (ALL),” Immunotherapy 3(2):1000142. [cited by applicant]
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Maude, S.L., et al. (2015) “CD19-targeted chimeric antigen receptor T-cell therapy for acute lymphoblastic leukemia,” Blood 125(25):4017-4023. [cited by applicant]
Sotillo, E., et al. (2015) “Convergence of Acquired Mutations and Alternative Splicing of CD19 Enables Resistance to CART-19 Immunotherapy ,” Cancer Discovery 5(12):1282-95. [cited by applicant]