IP Library › Granted Patent US 12,624,341
Granted Patent B2
US 12,624,341 · App. 19/037,555 · Granted May 12, 2026

Mammalian cell population and medicaments for cell therapies in humans and improved cell cultivation methods

Inventors: Antoine Lafont (Paris, FR); Mathieu Castela (Clamart, FR)
Assignee: SCARCELL Therapeutics
C12N5/0632A61K9/08A61K35/28A61K35/33A61K35/38A61K45/06A61P19/00C12N5/0656C12N5/0692C12N2500/32C12N2500/84C12N2501/115C12N2501/2301C12N2509/00
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Quick Facts
Patent No.
US 12,624,341
App. No.
19/037,555
Granted
May 12, 2026
Kind
B2
Abstract

Compositions of matter, including cell populations and medicaments, are provided that are derived from human gingival fibroblasts and have cell phenotypes that occur in proportions not found in natural gum tissue, but rather, are preferentially are selected to express proteins favoring angiogenesis and anti-inflammatory effects, while reducing cell populations that promote tumorigenicity and/or formation of metalloproteinases that inhibit tissue regeneration. Methods of generating such compositions are provided that increase proliferation many-fold compared to previously known methods, and methods of using such compositions in a wide range of human cell therapies are provided.

Claims (34)

1 . A pharmaceutical dose for treating a human ailment comprising:

an injectable volume of about 1.0 ml to 2.5 ml containing:

a medium comprising 10% dimethyl sulfoxide, 88% DMEM, and 1% non-essential amino acids; and

between 2 and 40 million viable cultured human gingival fibroblast cells having phenotypes such that at least about 90% of the cell population expresses CD90 and CD63 and about 10% or less of the cell population expresses CD146,

wherein the viable cultured human gingival fibroblast cells are cultured by a process comprising the steps of:

obtaining a population of viable gingival fibroblast cells representative of naturally occurring gingival fibroblast cells in human gum tissue;

culturing the viable gingival fibroblast cells through four passages in a culture medium that includes at least 20% fetal bovine serum (FBS) and basic fibroblast growth factor (bFGF), without isolating gingival fibroblast cell subpopulations, wherein during the first two passages, the population of viable gingival fibroblast cells monotonically increases; and

culturing the viable gingival fibroblast cells to a fifth passage, wherein during the fifth passage, omitting the 20% FBS and bFGF from the culture medium and adding interleukin 1β in a concentration of 0.1 ng/ml to 10 ng/ml,

wherein by completion of the fifth passage, the gingival fibroblast cells correspond to cell phenotypes cultivated so that at least about 90% of the cell population expresses CD90 and CD63 and about 10% or less of the cell population expresses CD146.

2 . The pharmaceutical dose of claim 1 , wherein a duration of the first of the four passages of culturing the viable gingival fibroblast cells is about 6 days.

3 . The pharmaceutical dose of claim 2 , wherein each of the second, the third, and the fourth passage of the four passages of culturing the viable gingival fibroblast cells has a duration of about 6 days.

4 . The pharmaceutical dose of claim 1 , wherein during at least the fifth passage of culturing the viable gingival fibroblast cells, non-essential amino acids are added to the culture medium.

5 . The pharmaceutical dose of claim 1 , wherein culturing the viable gingival fibroblast cells during each of the five passages expands the cells more than six-fold.

6 . The pharmaceutical dose of claim 1 , wherein the pharmaceutical dose contains between 10 and 20 million viable cultured human gingival fibroblast cells.

7 . The pharmaceutical dose of claim 1 , wherein about 10% or less of the cell population expresses at least one mRNA selected from the group consisting of MCAM, VCAM1, CD19, ITGAM, CD3D, CD4, FZD9, NGFR, NANOG, POU5F1, SOX2, KLF4, MYC, TNF, IL1A, IL1B, IL17A, IL23A, OSM, IF127, IFI44L, RSAD2, IFIT1, IFNA1 and IFNG mRNAs.

8 . The pharmaceutical dose of claim 1 , wherein about 50% or more of the cell population expresses at least one mRNA selected from the group consisting of TIMP1, CD9, CD81, THY, ITGB1, FST, and COL1A2 mRNAs.

9 . The pharmaceutical dose of claim 1 , wherein the viable human gingival fibroblast cells are allogeneic.

10 . A pharmaceutical dose for treating a human ailment comprising:

an injectable volume of about 1.0 ml to 2.5 ml containing:

a medium comprising 10% dimethyl sulfoxide, 88% DMEM, and 1% non-essential amino acids; and

at least 2 million viable cultured human gingival fibroblast cells having phenotypes such that at least about 90% of the cell population expresses CD90 and CD63 and about 10% or less of the cell population expresses CD146,

wherein the viable cultured human gingival fibroblast cells are cultured by a process comprising the steps of:

obtaining a population of viable gingival fibroblast cells representative of naturally occurring gingival fibroblast cells in human gum tissue;

culturing the population of viable gingival fibroblast cells through four passages in a culture medium that includes at least 20% fetal bovine serum (FBS) and basic fibroblast growth factor (bFGF), without isolating gingival fibroblast cell subpopulations, wherein during the first two passages, the population of viable gingival fibroblast cells monotonically increases; and

culturing the population of viable gingival fibroblast cells to a fifth passage, wherein during the fifth passage, omitting the 20% FBS and bFGF from the culture medium and adding interleukin 1β in a concentration of 0.1 ng/ml to 10 ng/ml and nonessential amino acids,

wherein by completion of the fifth passage, the gingival fibroblast cells correspond to cell phenotypes cultivated so that at least about 90% of the cell population expresses CD90 and CD63 and about 10% or less of the cell population expresses CD146.

11 . The pharmaceutical dose of claim 10 , wherein a duration of the first of the four passages of culturing the viable gingival fibroblast cells is about 6 days.

12 . The pharmaceutical dose of claim 10 , wherein each of the second, the third, and the fourth passage of the four passages of culturing the viable gingival fibroblast cells has a duration of about 6 days.

13 . The pharmaceutical dose of claim 10 , wherein culturing the viable gingival fibroblast cells during each of the five passages expands the cells more than six-fold.

14 . The pharmaceutical dose of claim 10 , wherein the pharmaceutical dose contains up to 40 million cells.

15 . The pharmaceutical dose of claim 10 , wherein about 10% or less of the cell population expresses at least one mRNA selected from the group consisting of MCAM, VCAM1, CD19, ITGAM, CD3D, CD4, FZD9, NGFR, NANOG, POU5F1, SOX2, KLF4, MYC, TNF, IL1A, IL1B, IL17A, IL23A, OSM, IF127, IFI44L, RSAD2, JFIT1, IFNA1 and IFNG mRNAs.

16 . The pharmaceutical dose of claim 10 , wherein about 50% or more of the cell population expresses at least one mRNA selected from the group consisting of TIMP1, CD9, CD81, THY, ITGB1, FST, and COL1A2 mRNAs.

17 . The pharmaceutical dose of claim 10 , wherein the viable human gingival fibroblast cells are allogeneic.

18 . The pharmaceutical dose of claim 10 , wherein the pharmaceutical dose is configured for injection with a syringe.

Priority Claims (1)
EP 23305350 · Mar 15, 2023 · regional
Continuity (3)
Division 18301839 · Apr 17, 2023
Provisional Application 63490489 · Mar 15, 2023
Related Publication 20250207093A1 · Jun 26, 2025
References Cited (37)
US 7951593B2 · Gogly et al. · 2011 [cited by applicant]
US 8303948B2 · Gogly et al. · 2012 [cited by applicant]
US 8609085B2 · Lafont et al. · 2013 [cited by applicant]
US 10300279B2 · Fraga et al. · 2019 [cited by applicant]
US 10624838B2 · Lafont et al. · 2020 [cited by applicant]
US 11229670B2 · Lafont et al. · 2022 [cited by applicant]
US 20110097421A1 · Gogly et al. · 2011 [cited by applicant]
US 20160008342A1 · Chiamvimonat · 2016 [cited by applicant]
US 20160151274A1 · Lafont · 2016 [cited by examiner]
US 20160256496A1 · Gogly et al. · 2016 [cited by applicant]
US 20180028571A1 · Gogly et al. · 2018 [cited by applicant]
US 20200268805A1 · Lafont et al. · 2020 [cited by applicant]
US 20200306174A1 · Lafont et al. · 2020 [cited by applicant]
US 20210156778A1 · Gadea Ramos et al. · 2021 [cited by applicant]
US 20210238542A1 · Kitano et al. · 2021 [cited by applicant]
US 20240307454A1 · Lafont et al. · 2024 [cited by applicant]
US 20240309323A1 · Lafont et al. · 2024 [cited by applicant]
AU 2008201328A1 · 2008 [cited by examiner]
WO 2023007244A1 · 2023 [cited by applicant]
Diar-Bakirly et al., Saudi J. Biol. Sci., 2021, vol. 28:2518-2526. [cited by examiner]
Wu et al., Med. Sci. Monit., 2018, vol. 24:1112-1123. [cited by examiner]
Palmqvist et al., J. Dent. Res., 2008, vol. 87(6):558-563. [cited by examiner]
Ahangar et al. “Human gingival fibroblast secretome accelerates wound healing through anti-inflammatory and pro-angiogenic mechanisms,” Regenerative Medicine, 5(24): 1-10 (2020). [cited by applicant]
Brown et al., “Ability of the Canine Brief Pain Inventory to detect response to treatment in dogs with osteoarthritis,” J Am Vet Med Assoc., 233(8):1278-1283 (Oct. 2008). [cited by applicant]
Diar-Bakirly et al., “Human gingival fibroblasts: Insolation, characterization, and evaluation of CD146 expression,” Saudi Journal of Biological Sciences, 28:2518-2526 (Jan. 2021). [cited by applicant]
Ferre et al. “Formation of Cartilage and Synovial Tissue by Human Gingival Stem Cells,” Stem Cells and Development, 23(23): 2895-2907 (Jul. 2014). [cited by applicant]
Forough et al. “Overexpression of tissue inhibitor of matrix metalloproteinase-1 inhibits vascular smooth muscle cell functions in vitro and in vivo,” Circ Res. Oct. 1996;79(4):812-20. [cited by applicant]
Fournier et al. “Multipotent progenitor cells in gingival connective tissue” Tissue Engineering Part A, 2010 vol. 16, No. 9, pp. 2891-2899, 2010. [cited by applicant]
Grindberg et al., “RNA-sequencing from single nuclei,” PNAS, 110(49):19802-19807 (Dec. 2013). [cited by applicant]
Guo et al., “Tissue inhibitors of metalloproteinases-(TIMP-1) and -2(TIMP-2) are major serum factors that stimulate the TIMP-1 gene in human gingival fibroblasts” Biochim. Biophys. Aceta, 2006, vol. 1763(3):296-304. [cited by applicant]
Hou et al., “Autologous Transplantation of Gingival Fibroblast-Like Cells and a Hydroxylapatite Complex Graft in the Treatment of Periodontal Osseous Defects: Cell Cultivation and Long-Term Report of Cases,” Cell Transp… [cited by applicant]
Linard et al., “Therapeutic Potential of Gingival Fibroblasts for Cutaneous Radiation Syndrome: Comparison to Bone Marrow-Mesenchymal Stem Cell Grafts,” Stem Cells and Development, 24(10):1182-1193 (Jan. 2015). [cited by applicant]
Magne et al. “IL-1β-Primed mesenchymal stromal cells improve epidermal substitute engraftment and wound healing via matrix metalloproteinases and transforming growth factor-β1”, Journal of Investigative Dermatology, 202… [cited by applicant]
Mao et al. “Gingiva-Derived Mesenchymal stem cell-extracellular vesicles activate schwann cell repair phenotype and promote nerve regeneration”, Tissue Engineering: Part A, 2019, vol. 25(11-12): 887-900. [cited by applicant]
Medical Dictionary, definition for heterogeneous, https://medical-dictionary.thedreedictionary.com/heterogeneous, 2012 p. 1. [cited by applicant]
Palkowitz et al. Biofunctionalization of Dental Abutment Surfaces by crosslinked ECM proteins strongly enhances adhesion and proliferation of gingival fibroblast: Advanced. Healthcare Materials, 2022. 10(10), pp. 1-12, … [cited by applicant]
Rajan et al. Conditioned medium from human gingival mesenchymal stem cells protects motor-neuron-like NSC-34 cells against scratch-injury-induced cell death Int. J. Immunopathol. Pharmacol., 2017, vol. 30(4):383-394. [cited by applicant]