IP Library Granted Patent US 9,616,140
Granted Patent B2
US 9,616,140 · App. 14/493,489 · Granted Apr 11, 2017

Fluorescent phospholipid ether compounds, compositions, and methods of use

Inventors: Anatoly Pinchuk (Madison, WI); Jamey P. Weichert (Fitchburg, WI); Marc Longino (Verona, WI); Irawati Kandela (Madison, WI); William R. Clarke (Colgate, WI)
Assignee: CELLECTAR BIOSCIENCES, INC.
A61K49/0021A61K49/0032A61K49/0052C07F9/5728C07F9/6561C07F9/65583A61K49/0017
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Quick Facts
Patent No.
US 9,616,140
App. No.
14/493,489
Granted
Apr 11, 2017
Kind
B2
Abstract

The invention generally relates to novel fluorescent phospholipid compounds, compositions comprising these compounds, and diagnostic methods utilizing these compounds. A preferred compound of the present invention has the following structural formula:

Claims (22)

1. A method of determining cancer in a subject, comprising:

administering to a subject a composition comprising a phospholipid ether compound selected from the group consisting of:

and

determining cancer in the subject by detecting the phospholipid ether compound in the subject.

2. The method of claim 1 , wherein the phospholipid ether compound has a structure:

3. The method of claim 1 , wherein the phospholipid ether compound has a structure:

4. The method of claim 1 , wherein the phospholipid ether compound has a structure:

5. The method of claim 1 , wherein the composition comprises a pharmaceutically acceptable carrier.

6. The method of claim 1 , wherein the subject is human.

7. The method of claim 1 , wherein the cancer is selected from the group consisting of melanoma, colorectal adenocarcinoma, uterine carcinoma, pancreatic carcinoma, ovarian adenocarcinoma, glioblastoma, clear cell carcinoma, and prostate adenocarcinoma.

8. The method of claim 1 , wherein the phospholipid ether compound is detected using fluorescence.

9. A method of detection of a phospholipid ether compound within a subject, comprising:

administering to a subject a composition comprising a phospholipid ether compound selected from the group consisting of:

and

detecting retention of the phospholipid ether compound within an organ within the subject.

10. The method of claim 9 , wherein the phospholipid ether compound has a structure

11. The method of claim 9 , wherein the phospholipid ether compound has a structure:

12. The method of claim 9 , wherein the phospholipid ether compound has a structure:

13. The method of claim 9 , wherein the composition comprises a pharmaceutically acceptable carrier.

14. The method of claim 9 , wherein the subject is human.

15. The method of claim 9 , wherein retention of the phospholipid ether compound is detected using fluorescence.

16. The method of claim 9 , wherein the organ is selected from the group consisting of colon, rectum, small bowel, esophagus, stomach, duodenum, uterus, pancreas and common bile duct, bronchi, sinus, lung, bladder, kidney, abdominal cavity, and thoracic cavity.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 7, 2014
From: PINCHUK, ANATOLY; WEICHERT, JAMEY P.; LONGINO, MARC; KANDELA, IRAWATI; CLARKE, WILLIAM R.
To: CELLECTAR, INC.
Reel/Frame 033899/0405 →
Continuity (7)
Continuation 13318546
Continuation 12463998 · May 11, 2009
Continuation 12463983 · May 11, 2009
Continuation 12463978 · May 11, 2009
Continuation 12463970 · May 11, 2009
Continuation 12463990 · May 11, 2009
Related Publication 20150044142A1 · Feb 12, 2015