IP Library Granted Patent US 10,654,900
Granted Patent B2
US 10,654,900 · App. 15/282,111 · Granted May 19, 2020

Method for treating prostatitis utilizing the pore-forming protein proaerolysin PRX302

Inventor: J. Curtis Nickel (Kingston, CA)
Assignee: Sophiris Bio, Corp.
C07K14/195A61K38/164A61K45/06A61K47/60A61K47/6425A61K47/6869C07K16/28A61K38/00C07K2319/30C07K2319/33
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Quick Facts
Patent No.
US 10,654,900
App. No.
15/282,111
Granted
May 19, 2020
Kind
B2
Abstract

The present disclosure includes methods and compositions for treating any condition involving prostatitis and similar diseases and/or conditions. These methods and compositions involve the use of targeted modified pore-forming proteins, including variant proaerolysin proteins.

Claims (13)

1. A method of treating prostatitis in a subject having prostatitis, said method comprising intraprostatically administering to said subject a therapeutically effective amount of PRX302,

wherein the PRX302 comprises an amino acid sequence having greater than 98% sequence identity to the amino acid sequence shown in SEQ ID NO:4 and which maintains the ability to selectively target and kill normal prostate cells, wherein the PRX302 comprises a polyhistidine tag;

wherein said administering of the PRX302 results in a reduction in prostate volume.

2. The method of claim 1 , wherein administration results in at least a 10% reduction in prostate volume.

3. The method of claim 1 , wherein administration results in at least a 50% reduction in prostate volume.

4. The method of claim 1 , wherein the prostatitis is chronic prostatitis.

5. The method of claim 1 , further comprising administering an additional therapeutic agent for treating prostatitis.

6. The method of claim 5 , wherein the additional therapeutic agent comprises an α-1-adrenoreceptor antagonist, an antibiotic, an anti-inflammatory agent, a 5α reductase inhibitor, a phytotherapy, or any combination thereof.

7. The method of claim 1 , wherein the subject has one or more signs of prostatitis comprising a prostate volume of 30 to 100 mL, prostate specific antigen blood levels of 4-10 ng/mL, or a combination thereof.

8. The method of claim 1 , wherein the polyhistidine tag comprises six histidine residues at the C-terminal end of PRX302 (SEQ ID NO:4).

9. A method of treating prostatitis in a subject having prostatitis, said method comprising intraprostatically administering to said subject a therapeutically effective amount of PRX302,

wherein the PRX302 comprises an amino acid sequence having greater than 98% sequence identity to the amino acid sequence shown in SEQ ID NO:4 and which maintains the ability to selectively target and kill normal prostate cells, and a C-terminal polyhistidine tag that includes six histidine residues;

wherein said administering of the PRX302 results in a reduction in prostate volume.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 20, 2016
From: NICKEL, CURTIS, DR
To: PROTOX THERAPEUTICS, INC.
Reel/Frame 040695/0680 →
CHANGE OF NAME Recorded Dec 20, 2016
From: PROTOX THERAPEUTICS, INC.
To: SOPHIRIS BIO INC.
Reel/Frame 040695/0820 →
Continuity (5)
Continuation 14537429 · Nov 10, 2014
Continuation 13608995 · Sep 10, 2012
Continuation 13139928
Provisional Application 61122709 · Dec 15, 2008
Related Publication 20170081370A1 · Mar 23, 2017