IP Library Granted Patent US 10,953,026
Granted Patent B2
US 10,953,026 · App. 16/417,488 · Granted Mar 23, 2021

N-acetyl mannosammine as a therapeutic agent

Inventors: Marjan Huizing (Santa Cruz, CA); William A. Gahl (Kensington, MD); Irini Manoli (Rockville, MD); Enriko Klootwijk (London, GB)
Assignee: The United States of America, as represented by the Secretary, Department of Health and Human Services
A61K31/7008A61K31/7012A61P3/10A61P9/12A61P21/00
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Quick Facts
Patent No.
US 10,953,026
App. No.
16/417,488
Granted
Mar 23, 2021
Kind
B2
Abstract

The invention relates to compositions and methods for treating kidney and muscle dysfunction that involves use of therapeutic amounts of N-acetyl mannosamine.

Claims (24)

1. A method of treating a condition or disease in a mammal in need thereof comprising

selecting a mammal with the condition or disease; and

administering to the mammal an effective amount of N-acetyl mannosamine or a derivative thereof, wherein the derivative consists of Formula I:

wherein R 1 , R 3 , R 4 , or R 5 is hydrogen, lower alkanoyl, carboxylate or lower alkyl; R 2 is lower alkyl, lower alkanoylalkyl, lower alkyl alkanoyloxy; and the condition or disease is muscular dystrophy, high blood pressure, or diabetes.

2. A method of treating a condition or disease in a mammal in need thereof comprising

selecting a mammal with the condition or disease; and

administering to the mammal a therapeutically effective amount of N-acetyl mannosamine to the mammal, wherein the condition or disease is muscular atrophy, muscular dystrophy, high blood pressure, or diabetes.

3. The method of claim 2 , wherein the therapeutic amount is about 0.1 g to about 50 g N-acetyl mannosamine per day.

4. The method of claim 2 , wherein the therapeutic amount is administered in a unit dosage of about 0.01 g to about 50 g N-acetyl mannosamine per unit dosage.

5. The method of claim 1 , comprising sustained release of the N-acetyl mannosamine or a derivative thereof.

6. The method of claim 1 , comprising topical administration of N-acetyl mannosamine or a derivative thereof.

7. The method of claim 1 , wherein the method reduces hematuria and/or proteinuria in the mammal.

8. A method of reducing proteinuria in a mammal in need thereof comprising:

selecting a mammal with a condition or disease, and

administering to the mammal an effective amount of N-acetyl mannosamine or a derivative thereof, to the mammal, wherein the derivative consists of Formula I:

wherein R 1 , R 3 , R 4 , or R 5 is hydrogen, lower alkanoyl, carboxylate or lower alkyl; R 2 is lower alkyl, lower alkanoylalkyl, lower alkyl alkanoyloxy; and wherein the condition or disease is high blood pressure, diabetes, or diabetic nephropathy, thereby reducing proteinuria in the mammal.

9. The method of claim 8 , comprising administering a therapeutic amount of N-acetyl mannosamine to the mammal.

10. The method of claim 9 , wherein the therapeutic amount is about 0.1 g to about 50 g N-acetyl mannosamine per day.

11. The method of claim 9 , wherein the therapeutic amount is administered in a unit dosage of about 0.01 g to about 50 g N-acetyl mannosamine per unit dosage.

12. The method of claim 8 , comprising sustained release of the N-acetyl mannosamine or a derivative thereof.

13. The method of claim 8 , comprising topical administration of the N-acetyl mannosamine or a derivative thereof.

14. The method of claim 9 , wherein the N-acetyl mannosamine is administered orally to the mammal.

15. The method of claim 9 , wherein the N-acetyl mannosamine is microencapsulated.

16. The method of claim 1 , comprising oral administration of N-acetyl mannosamine or a derivative thereof.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 29, 2019
From: HUIZING, MARJAN; GAHL, WILLIAM A.; MANOLI, IRINI; KLOOTWIJK, ENRIKO
To: GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES
Reel/Frame 049309/0064 →
CHANGE OF NAME Recorded May 29, 2019
From: GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES
To: THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES
Reel/Frame 049309/0206 →
Continuity (6)
Continuation 15702529 · Sep 12, 2017
Continuation 14754304 · Jun 29, 2015
Division 13791576 · Mar 8, 2013
Continuation 12530433
Provisional Application 60932451 · May 31, 2007
Related Publication 20190374561A1 · Dec 12, 2019