IP Library Granted Patent US 12,138,490
Granted Patent B2
US 12,138,490 · App. 17/714,964 · Granted Nov 12, 2024

Methods for treating hair loss disorders

Inventors: Angela M. Christiano (Mahwah, NJ); Raphael Clynes (West Nyack, NY)
Assignee: THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK
A61Q7/00A61K8/41A61K8/4953A61K8/64A61K31/137A61K31/277A61K31/407A61K31/437A61K31/506A61K31/519A61K31/52A61K31/529A61K31/5377A61K31/553A61K31/63A61K31/7052A61K31/713A61K2800/782
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Quick Facts
Patent No.
US 12,138,490
App. No.
17/714,964
Granted
Nov 12, 2024
Kind
B2
Abstract

The invention provides for methods for treating a hair loss disorder in a subject by administering a Janus Kinase/Signal Transducers and Activators of Transcription inhibitor.

Claims (16)

1. A method of treating alopecia areata in a human subject in need thereof, the method consisting of orally administering to the human subject an effective amount of a small molecule JAK3 inhibitor, wherein the alopecia areata in the human subject is treated.

2. The method of claim 1 , wherein the small molecule JAK3 inhibitor is selected from Janex 1 (WHI-P131), PF-956980, WHI-P154, tofacitinib (CP690550), VX-509, JAK3 Inhibitor IV (ZM-39923), NSC114792, R348, a pharmaceutically acceptable salt thereof, and a combination thereof.

3. The method of claim 1 , wherein the alopecia areata is selected from patchy alopecia areata, alopecia totalis, and alopecia universalis.

4. The method of claim 1 , wherein the JAK3 inhibitor is administered in a pharmaceutical composition selected from the group consisting of a solution, suspension, capsule, tablet, pill, and troche.

5. The method of claim 1 , wherein administering to the human subject occurs daily.

6. The method of claim 1 , wherein treatment is inducing hair growth.

7. The method of claim 1 , wherein the human subject is an adult.

8. The method of claim 1 , wherein the human subject is a child.

9. The method of claim 7 , wherein the effective amount is about 1 mg/kg body weight of the human subject.

10. The method of claim 7 , wherein the effective amount is selected from about 450 μg/kg body weight of the human subject, about 500 μg/kg body weight of the human subject, about 550 μg/kg body weight of the human subject, about 600 μg/kg body weight of the human subject, about 650 μg/kg body weight of the human subject, about 700 μg/kg body weight of the human subject, about 750 μg/kg body weight of the human subject, about 800 μg/kg body weight of the human subject, about 850 μg/kg body weight of the human subject, about 900 μg/kg body weight of the human subject and about 950 μg/kg body weight of the human subject.

11. The method of claim 7 , wherein treatment is inducing hair growth.

12. A method of treating severe alopecia areata in a human subject in need thereof, the method consisting of orally administering once daily to the human subject an effective amount of a small molecule JAK3 inhibitor, wherein the alopecia areata in the human subject is treated.

13. The method of claim 12 , wherein the small molecule JAK3 inhibitor is selected from Janex 1 (WHI-P131), PF-956980, WHI-P154, tofacitinib (CP690550), VX-509, JAK3 Inhibitor IV (ZM-39923), NSC114792, R348, a pharmaceutically acceptable salt thereof, and a combination thereof.

14. The method of claim 12 , wherein the severe alopecia areata is selected from alopecia totalis and alopecia universalis.

15. The method of claim 12 , wherein the human subject is an adult.

16. The method of claim 12 , wherein the human subject is a child.

Continuity (10)
Continuation 16299382 · Mar 12, 2019
Continuation 15668814 · Aug 4, 2017
Continuation 14821623 · Aug 7, 2015
Continuation 13886252 · May 2, 2013
Continuation In Part PCTUS2013034688 · Mar 29, 2013
Continuation In Part PCTUS2011059029 · Nov 2, 2011
Provisional Application 61645499 · May 10, 2012
Provisional Application 61617225 · Mar 29, 2012
Provisional Application 61409509 · Nov 2, 2010
Related Publication 20230111697A1 · Apr 13, 2023