IP Library Granted Patent US 12,521,335
Granted Patent B2
US 12,521,335 · App. 17/749,630 · Granted Jan 13, 2026

Cosmetic compositions containing vitamin C compounds and uses thereof

Inventors: Arthur Pellegrino (Newtown, PA); Fred Khoury (Chatsworth, CA); Ellen Delisle (Hauppauge, NY)
Assignee: RoC OPCO LLC
A61K8/676A61K8/64A61K8/86A61K8/9789A61Q19/08A61K2800/522A61K2800/805
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Quick Facts
Patent No.
US 12,521,335
App. No.
17/749,630
Granted
Jan 13, 2026
Kind
B2
Abstract

Disclosed herein are cosmetic compositions comprising a Vitamin C compound, a peptide, an antioxidant, and a hydrating agent. Also disclosed is a method visibly improving skin by brightening skin, evening skin tone, tightening skin, plumping skin, or improving the appearance of fine lines and wrinkles by topically applying a cosmetic composition comprising Vitamin C compound, a peptide, an antioxidant, and a hydrating agent.

Claims (23)

1 . A cosmetic composition comprising about 0.9 wt. % to about 3.00 wt. % of a Vitamin C compound, about 0.001 wt. % to about 1.0 wt. % of a peptide, about 0.01 wt. % to about 3.00 wt. % of an antioxidant, and up to about 3 wt. % of a hydrating agent;

wherein the Vitamin C compound comprises 3-O-ethyl ascorbic acid, Terminalia ferdinandiana fruit extract, tetrahexyldecyl ascorbate, or a combination thereof,

wherein the antioxidant comprises Cistus monspeliensis flower, leaf, and stem extract, troxerutin, Polygonum aviculare extract, or a combination thereof,

wherein the peptide comprises nonapeptide-1 and

wherein the hydrating agent comprises PPG-24-glycereth-24, Sodium PCA, a plant-based glyceride, a fruit complex, or a combination thereof.

2 . The cosmetic composition of claim 1 , wherein the Vitamin C compound comprises the combination of 3-O-ethyl ascorbic acid and Terminalia ferdinandiana fruit extract.

3 . The cosmetic composition of claim 1 , wherein the antioxidant comprises a combination of Cistus monspeliensis flower, leaf, and stem extract, troxerutin, and Polygonum aviculare extract.

4 . The cosmetic composition of claim 1 , wherein the hydrating agent comprises PPG-24-glycereth-24.

5 . The cosmetic composition of claim 1 , wherein the hydrating agent comprises a plant-based glyceride, a fruit complex, or a combination thereof.

6 . The cosmetic composition of claim 1 , wherein said composition is an oil-in-water emulsion or a gel-cream.

7 . The cosmetic composition of claim 1 , wherein the Vitamin C compound is present in an amount of from about 0.9% to about 1.0% by weight of the composition, the peptide is present in an amount of from about 0.001% to about 0.005% by weight of the composition, the antioxidant is present in an amount of from about 0.01% to about 1% by weight of the composition, and the hydrating agent is present in an amount up to about 1% by weight of the composition.

8 . The cosmetic composition of claim 7 , wherein the Vitamin C compound is present at up to about 1.00% by weight of the composition, the peptide is present at up to about 0.005% by weight of the composition, the antioxidant is present at up to about 0.25% by weight of the composition, and the hydrating agent is present at up to about 1.00% by weight of the composition.

9 . The cosmetic composition of claim 1 , wherein the composition does not cause skin irritation.

10 . A method of improving the skin comprising topically applying the cosmetic composition of claim 1 .

11 . The method of claim 10 , wherein improving the skin comprises visibly brightening the skin, visibly evening skin tone, visibly tightening the skin, or visibly plumping the skin.

12 . The method of claim 10 , wherein improving the skin comprises improving the appearance of fine lines and wrinkles.

13 . The method of claim 10 , wherein the composition is applied to a cleansed face and/or neck.

14 . The method of claim 10 , wherein the composition is applied in the evening.

15 . The cosmetic composition of claim 1 , wherein the vitamin C compound is a combination of 3-O-ethyl ascorbic acid, Terminalia ferdinandiana fruit extract, the peptide is 1-nonapeptide, the antioxidant is a combination of Cistus monspeliensis flower, leaf, and stem extract, troxerutin, Polygonum aviculare extract, and the hydrating agent is PPG-24-glycereth-24.

16 . The cosmetic composition of claim 1 , wherein the vitamin C compound is 3-O-ethyl ascorbic acid, the peptide is 1-nonapeptide, the antioxidant is a combination of Cistus monspeliensis flower, leaf, and stem extract, troxerutin, and Polygonum aviculare extract, and the hydrating agent is a combination of Shea Butter, Citrullus Vulgaris (Watermelon) Fruit Extract, Pyrus Malus (Apple) Fruit Extract, and Lens Esculenta (Lentil) Fruit Extract.

17 . The cosmetic composition of claim 1 , wherein the vitamin C compound is tetrahexyldecyl ascorbate, the peptide further comprises palmitoyl hexapeptide-12, the antioxidant is Cistus monspeliensis flower, leaf, and stem extract, and the hydrating agent is Sodium PCA.

18 . The cosmetic composition of claim 1 , wherein the vitamin C compound is 3-O-ethyl ascorbic acid, the peptide is nonapeptide-1, the antioxidant is a combination of Cistus monspeliensis flower, leaf, and stem extract, troxerutin, and Polygonum aviculare extract, and the hydrating agent is a combination of Citrullus Vulgaris (Watermelon) Fruit Extract, Pyrus Malus (Apple) Fruit Extract, Lens Esculenta (Lentil) Fruit Extract, and Sodium PCA.

19 . The cosmetic composition of claim 1 , wherein the vitamin C compound is 3-O-ethyl ascorbic acid, the peptide is 1-nonapeptide, the antioxidant is a combination of Cistus monspeliensis flower, leaf, and stem extract, troxerutin, Polygonum aviculare extract, and the hydrating agent is a combination of Shea Butter, Citrullus Vulgaris (Watermelon) Fruit Extract, Pyrus Malus (Apple) Fruit Extract, Lens Esculenta (Lentil) Fruit Extract, and Sodium PCA.

Assignments (2)
SECURITY INTEREST Recorded Feb 21, 2024
From: ROC OPCO LLC
To: BAIN CAPITAL CREDIT, LP, AS COLLATERAL AGENT
Reel/Frame 066509/0083 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 27, 2022
From: PELLEGRINO, ARTHUR; KHOURY, FRED; DELISLE, ELLEN
To: ROC OPCO LLC
Reel/Frame 060319/0194 →
Continuity (2)
Provisional Application 63191213 · May 20, 2021
Related Publication 20220370327A1 · Nov 24, 2022
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